Brief Information of the Compound and Protein
Compound Name
 Compound Info 
(+/-)-1-[2-(4-fluorophenyl)-2-(1-methylpiperidin-4-yl)ethyl]-4-[4-(1-naphthyl)butyl]piperazine tri hydrochloride
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 PubChem ID
CID: 45263492
Canonical SMILES
CN1CCC(C(CN2CCN(CCCCc3cccc4ccccc34)CC2)c2ccc(F)cc2)CC1.Cl
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Compound Formula C32H43ClFN3
Compound Structure
Protein Name
 Protein Info 
Melanocortin receptor 4
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
>
Peptide receptor (family A GPCR)
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Short peptide receptor (family A GPCR)
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Melanocortin receptor
Uniprot ID
P32245
Gene Name
MC4R
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000053 COS-7
 Cell Line Info 
Chlorocebus aethiops (Green monkey)  1
1
IC50 = 333 nM
   TI
   LI
   LO
   TS