Brief Information of the Compound and Protein
Compound Name
(+/-)-1-cyclohexyl-4-(1-(4-fluorophenyl)-2-{4-[4-(1-naphthyl)butyl]piperazin-1-yl}ethyl)piperazine
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PubChem ID
CID: 44423433
Canonical SMILES
Fc1ccc(cc1)C(CN1CCN(CCCCc2cccc3ccccc23)CC1)N1CCN(CC1)C1CCCCC1
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Compound Formula C36H49FN4
Compound Structure
Protein Name
Melanocortin receptor 4
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Short peptide receptor (family A GPCR)
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Melanocortin receptor
Uniprot ID
P32245
Gene Name
MC4R
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000109 COS-1 Chlorocebus aethiops (Green monkey)  1
1
IC50 = 241 nM
   TI
   LI
   LO
   TS