Brief Information of the Compound and Protein
Compound Name
 Compound Info 
(+/-)-1-[2-(4-fluorophenyl)-2-(4-isopropylpiperazin-1-yl)ethyl]-4-[3-(3-methoxybiphenyl-2-yl)propyl]piperazine
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 PubChem ID
CID: 44423460
Canonical SMILES
COc1cccc(-c2ccccc2)c1CCCN1CCN(CC(N2CCN(CC2)C(C)C)c2ccc(F)cc2)CC1
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Compound Formula C35H47FN4O
Compound Structure
Protein Name
 Protein Info 
Melanocortin receptor 4
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
>
Peptide receptor (family A GPCR)
>
Short peptide receptor (family A GPCR)
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Melanocortin receptor
Uniprot ID
P32245
Gene Name
MC4R
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000109 COS-1
 Cell Line Info 
Chlorocebus aethiops (Green monkey)  1
1
IC50 = 15.2 nM
   TI
   LI
   LO
   TS