Brief Information of the Compound and Protein
Compound Name
(+/-)-1-[2-(4-fluorophenyl)-2-(4-isopropylpiperazin-1-yl)ethyl]-4-[3-(40-methylbiphenyl-2-yl)propyl]piperazine
    Show/Hide
PubChem ID
CID: 44423465
Canonical SMILES
CC(C)N1CCN(CC1)C(CN1CCN(CCCc2ccccc2-c2ccc(C)cc2)CC1)c1ccc(F)cc1
    Show/Hide
Compound Formula C35H47FN4
Compound Structure
Protein Name
Melanocortin receptor 4
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
>
Peptide receptor (family A GPCR)
>
Short peptide receptor (family A GPCR)
>
Melanocortin receptor
Uniprot ID
P32245
Gene Name
MC4R
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000109 COS-1 Chlorocebus aethiops (Green monkey)  1
1
IC50 = 41.8 nM
   TI
   LI
   LO
   TS