Brief Information of the Compound and Protein
Compound Name
N-[(2R)-4-[6-(4-chlorophenyl)sulfanyl-2-(4-methoxyphenyl)-3-oxopyridazin-4-yl]butan-2-yl]-4-(4-fluorophenyl)-N-methylpiperidine-3-carboxamide
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PubChem ID
CID: 44397355
Canonical SMILES
COc1ccc(cc1)-n1nc(Sc2ccc(Cl)cc2)cc(CC[C@@H](C)N(C)C(=O)C2CNCCC2c2ccc(F)cc2)c1=O
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Compound Formula C34H36ClFN4O3S
Compound Structure
Protein Name
Melanocortin receptor 4
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Short peptide receptor (family A GPCR)
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Melanocortin receptor
Uniprot ID
P32245
Gene Name
MC4R
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
IC50 = 93 nM
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