Brief Information of the Compound and Protein
Compound Name
2-{5-[4-(2-Diethylamino-ethoxy)-phenyl]-pyrimidin-2-yl}-3-(2,3-dihydro-benzofuran-5-yl)-1,2,3,4-tetrahydro-pyrrolo[3,4-b]quinolin-9-one
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PubChem ID
CID: 11028215
SID: 16091201
Canonical SMILES
CCN(CC)CCOc1ccc(cc1)-c1cnc(nc1)N1Cc2c(nc3ccccc3c2O)C1c1ccc2OCCc2c1
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Compound Formula C35H35N5O3
Compound Structure
Protein Name
cGMP-specific 3',5'-cyclic phosphodiesterase
Protein Classification
Enzyme
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Phosphodiesterase
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Phosphodiesterase 5
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Phosphodiesterase 5A
Uniprot ID
O54735
Gene Name
PDE5A
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000070 RFL-6 Rattus norvegicus (Rat)  1
1
Ki = 0.53 nM
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