Brief Information of the Compound and Protein
Compound Name
 Compound Info 
methyl 1-[2-[[3-(4-methyl-6-morpholin-4-yl-1H-benzimidazol-2-yl)-2-oxo-1H-pyridin-4-yl]amino]ethyl]pyrazole-4-carboxylate
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 PubChem ID
CID: 136036563
Canonical SMILES
COC(=O)c1cnn(CCNc2cc[nH]c(=O)c2-c2nc3c(C)cc(cc3[nH]2)N2CCOCC2)c1
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Compound Formula C24H27N7O4
Compound Structure
Protein Name
 Protein Info 
Insulin-like growth factor 1 receptor
Protein Classification
Enzyme
>
Kinase
>
Protein Kinase
>
TK protein kinase group
>
Tyrosine protein kinase InsR family
Uniprot ID
P08069
Gene Name
IGF1R
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000766 SAL1
 Cell Line Info 
Homo sapiens (Human)  1
1
IC50 = 711 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 IC50 = 91 nM