Brief Information of the Compound and Protein
Compound Name
N-[1-(1,3-benzodioxol-5-ylmethyl)piperidin-4-yl]-2-(2-propan-2-yloxyethylamino)-5-thiophen-2-ylpyridine-3-carboxamide
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PubChem ID
CID: 44403535
Canonical SMILES
CC(C)OCCNc1ncc(cc1C(=O)NC1CCN(Cc2ccc3OCOc3c2)CC1)-c1cccs1
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Compound Formula C28H34N4O4S
Compound Structure
Protein Name
Melanin-concentrating hormone receptor 1
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Short peptide receptor (family A GPCR)
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MCH receptor
Uniprot ID
Q99705
Gene Name
MCHR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000016 IMR-32 Homo sapiens (Human)  1
1
IC50 = 190 nM
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