Brief Information of the Compound and Protein
Compound Name
 Compound Info 
RESINIFERATOXIN
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 PubChem ID
CID: 44564218
Canonical SMILES
COc1cc(CC(=O)OCC2=C[C@H]3[C@H]4OC5(Cc6ccccc6)O[C@@]4(C[C@@H](C)[C@]3(O5)[C@@H]3C=C(C)C(=O)[C@@]3(O)C2)C(C)=C)ccc1O
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Compound Formula C37H40O9
Compound Structure
Protein Name
 Protein Info 
Transient receptor potential cation channel subfamily V member 1
Protein Classification
Ion channel
>
Voltage-gated ion channel
>
Transient receptor potential channel
Uniprot ID
O35433
Gene Name
TRPV1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO
 Cell Line Info 
Cricetulus griseus (Chinese hamster)  3
1
EC50 = 0.27 nM
   TI
   LI
   LO
   TS
2
Ki = 0.043 nM
   TI
   LI
   LO
   TS
3
Ki = 0.13 nM
   TI
   LI
   LO
   TS
CL001009 CHO/VR1
 Cell Line Info 
Cricetulus griseus (Chinese hamster)  1
1
Ki = 0.0426 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 IC50 = 180 nM
2 Ki = 0.023 nM