Brief Information of the Compound and Protein
Compound Name
N-(piperidin-2-ylmethyl)-4-[4-(trifluoromethyl)phenyl]-2-[4-[3-(trifluoromethyl)pyridin-2-yl]piperazin-1-yl]-1H-imidazole-5-carboxamide
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PubChem ID
CID: 11548759
SID: 16650887
Canonical SMILES
FC(F)(F)c1ccc(cc1)-c1nc([nH]c1C(=O)NCC1CCCCN1)N1CCN(CC1)c1ncccc1C(F)(F)F
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Compound Formula C27H29F6N7O
Compound Structure
Protein Name
Transient receptor potential cation channel subfamily V member 1
Protein Classification
Ion channel
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Voltage-gated ion channel
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Transient receptor potential channel
Uniprot ID
O35433
Gene Name
TRPV1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  2
1
IC50 = 2950 nM
   TI
   LI
   LO
   TS
2
IC50 > 4000 nM
   TI
   LI
   LO
   TS