Brief Information of the Compound and Protein
Compound Name
3-[4-(4-Amino-butyl)-5-quinolin-2-yl-4H-[1,2,4]triazol-3-ylsulfanyl]-1-(7-methyl-1H-indol-3-yl)-propan-1-one
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PubChem ID
CID: 11705763
SID: 16810448
Canonical SMILES
Cc1cccc2c(c[nH]c12)C(=O)CCSc1nnc(-c2ccc3ccccc3n2)n1CCCCN
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Compound Formula C27H28N6OS
Compound Structure
Protein Name
Somatostatin receptor type 5
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Short peptide receptor (family A GPCR)
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Somatostatin receptor
Uniprot ID
P35346
Gene Name
SSTR5
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000026 CHO-K1 Cricetulus griseus (Chinese hamster)  1
1
EC50 = 2.3 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 Ki = 0.38 nM