Brief Information of the Compound and Protein
Compound Name
(E)-N-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-3-(2-morpholin-4-yl-6-trifluoromethyl-pyridin-3-yl)-acrylamide
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PubChem ID
CID: 10194869
SID: 15191228
Canonical SMILES
FC(F)(F)c1ccc(\C=C\C(=O)Nc2ccc3OCCOc3c2)c(n1)N1CCOCC1
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Compound Formula C21H20F3N3O4
Compound Structure
Protein Name
Transient receptor potential cation channel subfamily V member 1
Protein Classification
Ion channel
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Voltage-gated ion channel
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Transient receptor potential channel
Uniprot ID
Q8NER1
Gene Name
TRPV1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  2
1
IC50 = 15 nM
   TI
   LI
   LO
   TS
2
IC50 = 40 nM
   TI
   LI
   LO
   TS