Brief Information of the Compound and Protein
Compound Name
 Compound Info 
Biphenyl-2-carboxylic acid [2-(4-[1,4']bipiperidinyl-1'-yl-4-oxo-butoxy)-4-(5,6,7,8-tetrahydro-thieno[3,2-b]azepine-4-carbonyl)-phenyl]-amide
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 PubChem ID
CID: 11239468
SID: 16323412
Canonical SMILES
O=C(CCCOc1cc(ccc1NC(=O)c1ccccc1-c1ccccc1)C(=O)N1CCCCc2sccc12)N1CCC(CC1)N1CCCCC1
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Compound Formula C42H48N4O4S
Compound Structure
Protein Name
 Protein Info 
Vasopressin V2 receptor
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Short peptide receptor (family A GPCR)
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Vasopressin and oxytocin receptor
Uniprot ID
P30518
Gene Name
AVPR2
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO
 Cell Line Info 
Cricetulus griseus (Chinese hamster)  1
1
IC50 = 30 nM
   TI
   LI
   LO
   TS