Brief Information of the Compound and Protein
Compound Name
7-fluoro-N-[1-[[3-fluoro-4-(2-pyrrolidin-1-ylethylcarbamoyl)phenyl]methyl]piperidin-4-yl]-4-oxochromene-2-carboxamide
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PubChem ID
CID: 16739263
SID: 26698089
Canonical SMILES
Fc1ccc2c(c1)oc(cc2=O)C(=O)NC1CCN(Cc2ccc(C(=O)NCCN3CCCC3)c(F)c2)CC1
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Compound Formula C29H32F2N4O4
Compound Structure
Protein Name
Melanin-concentrating hormone receptor 1
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Short peptide receptor (family A GPCR)
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MCH receptor
Uniprot ID
Q99705
Gene Name
MCHR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000016 IMR-32 Homo sapiens (Human)  2
1
IC50 = 29 nM
   TI
   LI
   LO
   TS
2
IC50 = 420 nM
   TI
   LI
   LO
   TS