Brief Information of the Compound and Protein
Compound Name
7-fluoro-N-[1-[[3-fluoro-4-[(2E)-2-methoxyiminoethoxy]phenyl]methyl]piperidin-4-yl]-4-oxochromene-2-carboxamide
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PubChem ID
CID: 44438747
Canonical SMILES
CO\N=C\COc1ccc(CN2CCC(CC2)NC(=O)c2cc(=O)c3ccc(F)cc3o2)cc1F
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Compound Formula C25H25F2N3O5
Compound Structure
Protein Name
Melanin-concentrating hormone receptor 1
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Short peptide receptor (family A GPCR)
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MCH receptor
Uniprot ID
Q99705
Gene Name
MCHR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000016 IMR-32 Homo sapiens (Human)  2
1
IC50 = 31 nM
   TI
   LI
   LO
   TS
2
IC50 = 480 nM
   TI
   LI
   LO
   TS