Brief Information of the Compound and Protein
Compound Name
3-[6-(dimethylamino)-4-methylpyridin-3-yl]-2,5-dimethyl-N-(naphthalen-2-ylmethyl)-N-propylpyrazolo[1,5-a]pyrimidin-7-amine
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PubChem ID
CID: 11375016
SID: 16468288
Canonical SMILES
CCCN(Cc1ccc2ccccc2c1)c1cc(C)nc2c(c(C)nn12)-c1cnc(cc1C)N(C)C
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Compound Formula C30H34N6
Compound Structure
Protein Name
Corticotropin-releasing factor receptor 1
Protein Classification
Membrane receptor
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Family B G protein-coupled receptor
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Peptide receptor (family B GPCR)
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Corticotropin releasing factor receptor
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Corticotropin releasing factor receptor
Uniprot ID
P34998
Gene Name
CRHR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
Ki = 15 nM
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