Brief Information of the Compound and Protein
Compound Name
3-[6-(dimethylamino)-4-methylpyridin-3-yl]-2,5-dimethyl-N-(5-methylhexan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
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PubChem ID
CID: 11280879
SID: 16367797
Canonical SMILES
CC(C)CCC(C)Nc1cc(C)nc2c(c(C)nn12)-c1cnc(cc1C)N(C)C
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Compound Formula C23H34N6
Compound Structure
Protein Name
Corticotropin-releasing factor receptor 1
Protein Classification
Membrane receptor
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Family B G protein-coupled receptor
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Peptide receptor (family B GPCR)
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Corticotropin releasing factor receptor
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Corticotropin releasing factor receptor
Uniprot ID
P34998
Gene Name
CRHR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
Ki = 13 nM
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