Brief Information of the Compound and Protein
Compound Name
 Compound Info 
2-[({2-[(1E)-3-(diethylamino)-1-propenyl]phenyl}sulfonyl)-amino]-5,6,7,8-tetrahydro-1-naphthalenecarboxylic acid
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 PubChem ID
CID: 11546119
SID: 16648296
Canonical SMILES
CN(C)C/C=C/c1ccccc1S(=O)(=O)Nc1ccc2c(c1C(=O)O)CCCC2
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Compound Formula C22H26N2O4S
Compound Structure
Protein Name
 Protein Info 
Methionine aminopeptidase 2
Protein Classification
Enzyme
>
Protease
>
Metallo protease
>
Metallo protease MG clan
>
Metallo protease M24A subfamily
Uniprot ID
P50579
Gene Name
METAP2
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000156 HT-1080
 Cell Line Info 
Homo sapiens (Human)  1
1
EC50 = 3000 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 IC50 = 27 nM
2 IC50 = 410 nM