Brief Information of the Compound and Protein
Compound Name
(R)-6-(4-chlorophenyl)-3-(2-(cyclopentylmethyl)-2,3-dihydrobenzo[b][1,4]dioxin-6-yl)thieno[3,2-d]pyrimidin-4(3H)-one
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PubChem ID
CID: 11995445
SID: 17494568
Canonical SMILES
Clc1ccc(cc1)-c1cc2ncn(-c3ccc4O[C@H](CN5CCCC5)COc4c3)c(=O)c2s1
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Compound Formula C25H22ClN3O3S
Compound Structure
Protein Name
Melanin-concentrating hormone receptor 1
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Short peptide receptor (family A GPCR)
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MCH receptor
Uniprot ID
Q99705
Gene Name
MCHR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
IC50 = 7 nM
   TI
   LI
   LO
   TS