Brief Information of the Compound and Protein
Compound Name
N-[1-(1,3-benzodioxol-5-ylmethyl)piperidin-4-yl]-4-oxo-7-(trifluoromethyl)chromene-2-carboxamide
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PubChem ID
CID: 11974030
SID: 17425879
Canonical SMILES
FC(F)(F)c1ccc2c(c1)oc(cc2=O)C(=O)NC1CCN(Cc2ccc3OCOc3c2)CC1
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Compound Formula C24H21F3N2O5
Compound Structure
Protein Name
Melanin-concentrating hormone receptor 1
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Short peptide receptor (family A GPCR)
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MCH receptor
Uniprot ID
Q99705
Gene Name
MCHR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000016 IMR-32 Homo sapiens (Human)  2
1
IC50 = 178 nM
   TI
   LI
   LO
   TS
2
IC50 = 3070 nM
   TI
   LI
   LO
   TS