Brief Information of the Compound and Protein
Compound Name
2-Benzyl-8-(2-{1-[4-(4,5-dihydro-1H-imidazol-2-yl)-benzyl]-piperidin-4-yl}-ethoxy)-2,3,4,5-tetrahydro-benzo[c]azepin-1-one
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PubChem ID
CID: 9828622
SID: 14787820
Canonical SMILES
O=C1N(Cc2ccccc2)CCCc2ccc(OCCC3CCN(Cc4ccc(cc4)C4=NCCN4)CC3)cc12
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Compound Formula C34H40N4O2
Compound Structure
Protein Name
Melanin-concentrating hormone receptor 1
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Short peptide receptor (family A GPCR)
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MCH receptor
Uniprot ID
Q99705
Gene Name
MCHR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
IC50 = 300 nM
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