Brief Information of the Compound and Protein
| Compound Name |
9-cis-retinoic acid (9cRA)
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PubChem ID | |||||
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Compound Structure |
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| Protein Name |
Retinoic acid receptor RXR-alpha
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Protein Classification |
Transcription factor
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Nuclear receptor
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Nuclear hormone receptor subfamily 2
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Nuclear hormone receptor subfamily 2 group B
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Nuclear hormone receptor subfamily 2 group B member 1
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| Uniprot ID | Gene Name | RXRA |
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Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
| Cell Line ID | Cell Line Name | Cell Line Organism | |
| CL000044 | CV-1 | Chlorocebus aethiops (Green monkey) | 2 |
| 1 |
EC50 = 900 nM
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TI
LI
LO
TS
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| 2 |
EC50 = 1015 nM
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TI
LI
LO
TS
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Biochemical Assays
| 1 | EC50 = 430 nM | ||
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| 2 | EC50 = 900 nM | ||
| 3 | EC50 > 10000 nM | ||
| 4 | IC50 > 1000 nM | ||
| 5 | Kd = 9 nM | ||
| 6 | Kd = 53 nM | ||
| 7 | Kd > 200 nM | ||
| 8 | Ki = 0.4 nM | ||
| 9 | Ki = 350 nM | ||