Brief Information of the Compound and Protein
Compound Name
1-(17-chloro-3-oxa-2-azatetracyclo[12.4.0.02,6.07,12]octadeca-1(14),7,9,11,15,17-hexaen-4-yl)-N,N-dimethylmethanamine
    Show/Hide
PubChem ID
CID: 10381889
SID: 15396992
Canonical SMILES
CN(C)CC1CC2N(O1)c1cc(Cl)ccc1Cc1ccccc21
    Show/Hide
Compound Formula C19H21ClN2O
Compound Structure
Protein Name
5-hydroxytryptamine receptor 2A
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
>
Small molecule receptor (family A GPCR)
>
Monoamine receptor
>
Serotonin receptor
Uniprot ID
P28223
Gene Name
HTR2A
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000309 NCTC clone 929 Mus musculus (Mouse)  1
1
IC50 = 3.467 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 IC50 = 3.467 nM