Brief Information of the Compound and Protein
Compound Name
 Compound Info 
5-(2,4-Dioxo-thiazolidin-5-ylmethyl)-2-methoxy-N-(4-trifluoromethyl-benzyl)-benzamide
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 PubChem ID
CID: 151183
SID: 22395193
Canonical SMILES
COc1ccc(CC2SC(=O)NC2=O)cc1C(=O)NCc1ccc(C(F)(F)F)cc1
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Compound Formula C20H17F3N2O4S
Compound Structure
Protein Name
 Protein Info 
Peroxisome proliferator-activated receptor gamma
Protein Classification
Transcription factor
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Nuclear receptor
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Nuclear hormone receptor subfamily 1
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Nuclear hormone receptor subfamily 1 group C
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Nuclear hormone receptor subfamily 1 group C member 3
Uniprot ID
P37231
Gene Name
PPARG
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000026 CHO-K1
 Cell Line Info 
Cricetulus griseus (Chinese hamster)  1
1
EC50 = 800 nM
   TI
   LI
   LO
   TS
CL000044 CV-1
 Cell Line Info 
Chlorocebus aethiops (Green monkey)  1
1
EC50 = 900 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 EC50 = 800 nM
2 EC50 = 850 nM
3 EC50 = 1090 nM
4 IC50 = 463 nM
5 Kd = 326 nM
6 Kd = 330 nM
7 Ki = 330 nM