Brief Information of the Compound and Protein
Compound Name
1-{4-[3-(3-Chloro-5-fluoro-phenyl)-prop-2-ynyloxy]-[1,2,5]thiadiazol-3-yl}-4-aza-tricyclo[2.2.1.0*2,6*]heptane
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PubChem ID
CID: 44303408
Canonical SMILES
Fc1cc(Cl)cc(c1)C#CCOc1nsnc1C12CN3CC1C2C3
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Compound Formula C17H13ClFN3OS
Compound Structure
Protein Name
Muscarinic acetylcholine receptor M2
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Acetylcholine receptor
Uniprot ID
P08172
Gene Name
CHRM2
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL001014 CHO-CHRM2 Cricetulus griseus (Chinese hamster)  1
1
EC50 = 1480 nM
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