Brief Information of the Compound and Protein
Compound Name
1-{4-[3-(3,5-Dichloro-phenyl)-prop-2-ynylsulfanyl]-[1,2,5]thiadiazol-3-yl}-4-aza-tricyclo[2.2.1.0*2,6*]heptane
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PubChem ID
CID: 44303293
Canonical SMILES
Clc1cc(Cl)cc(c1)C#CCSc1nsnc1C12CN3CC1C2C3
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Compound Formula C17H13Cl2N3S2
Compound Structure
Protein Name
Muscarinic acetylcholine receptor M2
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Acetylcholine receptor
Uniprot ID
P08172
Gene Name
CHRM2
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL001014 CHO-CHRM2 Cricetulus griseus (Chinese hamster)  1
1
EC50 = 528 nM
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