Brief Information of the Compound and Protein
Compound Name
 Compound Info 
5-Amino-1H-[1,2,4]triazole-3-carboxylic acid ((S)-1-{(S)-1-[((S)-carbamoyl-phenyl-methyl)-carbamoyl]-4-guanidino-butylcarbamoyl}-2-cyclohexyl-ethyl)-amide
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 PubChem ID
CID: 44280768
Canonical SMILES
NC(=N)NCCC[C@H](NC(=O)[C@H](CC1CCCCC1)NC(=O)c1nnc(N)[nH]1)C(=O)N[C@H](C(N)=O)c1ccccc1
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Compound Formula C26H39N11O4
Compound Structure
Protein Name
 Protein Info 
Proteinase-activated receptor 1
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
>
Peptide receptor (family A GPCR)
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Protease-activated receptor
>
Protease-activated receptor
Uniprot ID
P25116
Gene Name
F2R
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000812 CHRF
 Cell Line Info 
Homo sapiens (Human)  1
1
IC50 = 7000 nM
   TI
   LI
   LO
   TS