General Information of the Protein
Protein ID
PT06764
Protein Name
Taste receptor type 2 member 10
Secondarily
Protein Name
Taste receptor family B member 2
Gene Name
TAS2R10
Sequence
MLRVVEGIFIFVVVSESVFGVLGNGFIGLVNCIDCAKNKLSTIGFILTGLAISRIFLIWIIITDGFIQIFSPNIYASGNLIEYISYFWVIGNQSSMWFATSLSIFYFLKIANFSNYIFLWLKSRTNMVLPFMIVFLLISSLLNFAYIAKILNDYKTKNDTVWDLNMYKSEYFIKQILLNLGVIFFFTLSLITCIFLIISLWRHNRQMQSNVTGLRDSNTEAHVKAMKVLISFIILFILYFIGMAIEISCFTVRENKLLLMFGMTTTAIYPWGHSFILILGNSKLKQASLRVLQQLKCCEKRKNLRVT
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Organism
Homo sapiens, Human
Protein Classification
Membrane receptor
>
Taste family G protein-coupled receptor
>
Taste receptor (taste family GPCR)
Function
Gustducin-coupled strychnine receptor implicated in the perception of bitter compounds in the oral cavity and the gastrointestinal tract. Signals through PLCB2 and the calcium-regulated cation channel TRPM5.
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Uniprot ID
Primary ID:
Q9NYW0

Secondarily ID:
Q3MIM9
Q6NTD9
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HGNC ID
HGNC:14918
Subcellular Location
Membrane
Map of Molecular Bioactivity Related to the Protein
Map of Molecular Bioactivity Related to the Protein

Protein
Cell Line
Compound

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Protein
Cell Line ID: CL000025 , HEK-293T
Compound ID Compound Name Compound Formula
CP0850084
3-Betahydroxy dihydro costunolide
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C15H22O3
 4
1
EC50 = 2740 nM
   TI
   LI
   LO
   TS
2
EC50 = 5390 nM
   TI
   LI
   LO
   TS
3
EC50 = 21720 nM
   TI
   LI
   LO
   TS
4
EC50 = 25200 nM
   TI
   LI
   LO
   TS
CP0866307
3-beta-hydroxy dihydro costunolide
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C15H22O3
 1
1
EC50 = 25200 nM
   TI
   LI
   LO
   TS