General Information of the Protein
Protein ID
PT06703
Protein Name
Tachykinin-3
Secondarily
Protein Name
ZNEUROK1
Neuromedin-K
Gene Name
TAC3
Secondarily
Gene Name
NKNB
UNQ585/PRO1155
Sequence
MRIMLLFTAILAFSLAQSFGAVCKEPQEEVVPGGGRSKRDPDLYQLLQRLFKSHSSLEGLLKALSQASTDPKESTSPEKRDMHDFFVGLMGKRSVQPDSPTDVNQENVPSFGILKYPPRAE
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Organism
Homo sapiens, Human
Protein Classification
Secreted protein
Function
Tachykinins are active peptides which excite neurons, evoke behavioral responses, are potent vasodilators and secretagogues, and contract (directly or indirectly) many smooth muscles (By similarity). Is a critical central regulator of gonadal function.
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Uniprot ID
Primary ID:
Q9UHF0

Secondarily ID:
Q6IAG2
Q71BC6
Q71BC9
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Ensembl ID
ENSG00000166863
HGNC ID
HGNC:11521
Subcellular Location
Secreted
Map of Molecular Bioactivity Related to the Protein
Map of Molecular Bioactivity Related to the Protein

Protein
Cell Line
Compound

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Protein
Cell Line ID: CL000228 , IM-9
Compound ID Compound Name Compound Formula
CP0411506
US8470816, 30
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C27H30Cl3N3O3
 1
1
IC50 = 23 nM
   TI
   LI
   LO
   TS
CP0420222
US8470816, 18
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C27H30BrCl2N3O3
 1
1
IC50 = 24 nM
   TI
   LI
   LO
   TS
CP0415706
US8470816, 24
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C28H33Cl2N3O3
 1
1
IC50 = 49 nM
   TI
   LI
   LO
   TS
CP0472579
US8470816, 21
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C28H33Cl2N3O4
 1
1
IC50 = 130 nM
   TI
   LI
   LO
   TS
CP0411371
US8470816, 31
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C33H35Cl2N3O3
 1
1
IC50 = 160 nM
   TI
   LI
   LO
   TS
CP0429693
US8470816, 91
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C29H29Cl2F6N3O3
 1
1
IC50 = 330 nM
   TI
   LI
   LO
   TS