General Information of the Protein
Protein ID
PT02841
Protein Name
Envelope glycoprotein gp160
Secondarily
Protein Name
Env polyprotein
Glycoprotein 120
Glycoprotein 41
Gene Name
ENV
Sequence
MRATEIRKNYQHLWKGGTLLLGMLMICSAAEQLWVTVYYGVPVWKEATTTLFCASDAKAYDTEVHNVWATHACVPTDPNPQEVKLENVTENFNMWKNNMVEQMHEDIISLWDQSLKPCVKLTPLCVTLNCTDLRNATNTTSSSWETMEKGEIKNCSFNITTSIRDKVQKEYALFYNLDVVPIDNASYRLISCNTSVITQACPKVSFEPIPIHYCAPAGFAILKCNDKKFNGTGPCTNVSTVQCTHGIRPVVSTQLLLNGSLAEEEIVIRSENFTNNAKTIIVQLNESVVINCTRPNNNTRKSINIGPGRALYTTGEIIGDIRQAHCNLSKTQWENTLEQIAIKLKEQFGNNKTIIFNPSSGGDPEIVTHSFNCGGEFFYCNSTQLFTWNDTRKLNNTGRNITLPCRIKQIINMWQEVGKAMYAPPIRGQIRCSSNITGLLLTRDGGKDTNGTEIFRPGGGDMRDNWRSELYKYKVVKIEPLGVAPTKAKRRVVQREKRAVGLGALFLGFLGAAGSTMGAASITLTVQARQLLSGIVQQQNNLLRAIEAQQHLLQLTVWGIKQLQARVLAVERYLRDQQLLGIWGCSGKLICTTTVPWNTSWSNKSLNEIWDNMTWMKWEREIDNYTHIIYSLIEQSQNQQEKNEQELLALDKWASLWNWFDITKWLWYIKIFIMIVGGLIGLRIVFVVLSIVNRVRQGYSPLSFQTHLPAQRGPDRPDGIEEEGGERDRDRSGPLVDGFLAIIWVDLRSLCLFSYHRLRDLLLIVTRIVELLGRRGWGVLKYWWNLLQYWIQELKNSAVSLLNATAIAVAEGTDRVIEILQRAFRAVLHIPVRIRQGLERALL
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Organism
Human immunodeficiency virus type 1 group M subtype B (isolate YU-2), HIV-1
Protein Classification
Surface antigen
Function
Oligomerizes in the host endoplasmic reticulum into predominantly trimers. In a second time, gp160 transits in the host Golgi, where glycosylation is completed. The precursor is then proteolytically cleaved in the trans-Golgi and thereby activated by cellular furin or furin-like proteases to produce gp120 and gp41.
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Uniprot ID
P35961
Subcellular Location
Virion membrane
Host cell membrane
Host endosome membrane
Map of Molecular Bioactivity Related to the Protein
Map of Molecular Bioactivity Related to the Protein

Protein
Cell Line
Compound

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Protein
Cell Line ID: CL000442 , Cf2Th-CCR5
 Cell Line Info 
Compound ID Compound Name Compound Formula
CP0282815
 Compound Info 
N'-(4-chloro-3-fluorophenyl)-N-[[2-(morpholin-4-ylmethyl)phenyl]methyl]oxamide
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C20H21ClFN3O3
  1
1
IC50 = 20500 nM
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CP0296385
 Compound Info 
N'-(4-chloro-3-fluorophenyl)-N-[2-(1-propan-2-ylpiperidin-2-yl)ethyl]oxamide
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C18H25ClFN3O2
  1
1
IC50 = 27000 nM
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CP0296382
 Compound Info 
N'-(4-chloro-3-fluorophenyl)-N-[[1-(2-hydroxyethyl)piperidin-3-yl]methyl]oxamide
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C16H21ClFN3O3
  1
1
IC50 = 27600 nM
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CP0283382
 Compound Info 
N'-(4-chloro-3-fluorophenyl)-N-[(2,2,6,6-tetramethylpiperidin-4-yl)methyl]oxamide
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C18H25ClFN3O2
  1
1
IC50 = 33000 nM
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CP0283381
 Compound Info 
N'-(4-chloro-3-fluorophenyl)-N-[(1-cyclopropylpyrrolidin-3-yl)methyl]oxamide
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C16H19ClFN3O2
  1
1
IC50 = 33500 nM
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CP0144831
 Compound Info 
N-(5-azaspiro[3.5]nonan-8-yl)-N'-(4-chloro-3-fluorophenyl)oxamide
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C16H19ClFN3O2
  1
1
IC50 = 38500 nM
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CP0293020
 Compound Info 
N'-(4-chloro-3-fluorophenyl)-N-(1,2,3,4-tetrahydroisoquinolin-1-ylmethyl)oxamide
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C18H17ClFN3O2
  1
1
IC50 = 50400 nM
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CP0228422
 Compound Info 
N'-(4-chloro-3-fluorophenyl)-N-(1-cyclohexylpyrrolidin-3-yl)oxamide
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C18H23ClFN3O2
  1
1
IC50 = 57100 nM
 Bioactivity Info 
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CP0144833
 Compound Info 
N'-(4-chloro-3-fluorophenyl)-N-(1-propylpiperidin-3-yl)oxamide
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C16H21ClFN3O2
  1
1
IC50 = 58000 nM
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CP0282782
 Compound Info 
(R)-N1-(1-benzylpyrrolidin-3-yl)-N2-(4-chloro-3-fluorophenyl)oxalamide
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C19H19ClFN3O2
  1
1
IC50 = 58500 nM
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CP0293019
 Compound Info 
N'-(4-chlorophenyl)-N-[(1-ethylpyrrolidin-2-yl)methyl]oxamide
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C15H20ClN3O2
  1
1
IC50 = 58600 nM
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CP0297492
 Compound Info 
N'-(4-chloro-3-fluorophenyl)-N-[2-(4-chlorophenyl)-2-pyrrolidin-1-ylethyl]oxamide
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C20H20Cl2FN3O2
  1
1
IC50 = 61400 nM
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CP0108705
 Compound Info 
N'-(4-chloro-3-fluorophenyl)-N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]oxamide
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C14H14ClFN4O2
  1
1
IC50 = 64500 nM
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CP0304542
 Compound Info 
N'-(4-chloro-3-fluorophenyl)-N-(1,2,2,6,6-pentamethylpiperidin-4-yl)oxamide
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C18H25ClFN3O2
  1
1
IC50 = 65800 nM
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CP0144832
 Compound Info 
N-[[(3aS,6aS)-2,3,4,5,6,6a-hexahydro-1H-cyclopenta[c]pyrrol-3a-yl]methyl]-N'-(4-chloro-3-fluorophenyl)oxamide
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C16H19ClFN3O2
  1
1
IC50 = 68300 nM
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CP0049276
 Compound Info 
N'-(4-chloro-3-fluorophenyl)-N-[2-(2-chlorophenyl)-2-(4-methylpiperazin-1-yl)ethyl]oxamide
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C21H23Cl2FN4O2
  1
1
IC50 = 73600 nM
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CP0214321
 Compound Info 
N'-(4-chlorophenyl)-N-(2,2,6,6-tetramethylpiperidin-4-yl)oxamide
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C17H24ClN3O2
  1
1
IC50 = 73700 nM
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CP0282807
 Compound Info 
N'-(4-chloro-3-fluorophenyl)-N-(2,2,6,6-tetramethylpiperidin-4-yl)oxamide
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C17H23ClFN3O2
  1
1
IC50 = 74800 nM
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CP0282780
 Compound Info 
N'-(4-chloro-3-fluorophenyl)-N-[2-[(2S,6R)-2,6-dimethylpiperidin-1-yl]ethyl]oxamide
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C17H23ClFN3O2
  1
1
IC50 = 75500 nM
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CP0282779
 Compound Info 
N-[[(4S,5S)-5-(aminomethyl)-2,2-dimethyl-1,3-dioxolan-4-yl]methyl]-N'-(4-chloro-3-fluorophenyl)oxamide
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C15H19ClFN3O4
  1
1
IC50 = 76600 nM
 Bioactivity Info 
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CP0228423
 Compound Info 
N'-(4-chloro-3-fluorophenyl)-N-[(1-ethylpyrrolidin-2-yl)methyl]oxamide
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C15H19ClFN3O2
  1
1
IC50 = 85200 nM
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CP0049251
 Compound Info 
N-(4-bromophenyl)-5-(pyrrolidin-1-ylmethyl)-1,2-oxazole-3-carboxamide
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C15H16BrN3O2
  1
1
IC50 > 100000 nM
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CP0049265
 Compound Info 
1-(4-chlorophenyl)-3-[[2-(5-methyl-2-propan-2-ylphenoxy)acetyl]amino]urea
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C19H22ClN3O3
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0049277
 Compound Info 
N-(4-chloro-3-fluorophenyl)-N'-[1-(2-chlorophenyl)-1-morpholin-4-ylpropan-2-yl]oxamide
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C21H22Cl2FN3O3
  1
1
IC50 > 100000 nM
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CP0049278
 Compound Info 
N-(4-chlorophenyl)-3-(1,2,4-triazol-4-yl)-1H-pyrazole-5-carboxamide
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C12H9ClN6O
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0049279
 Compound Info 
N-(4-chlorophenyl)-7-hydroxy-2-iminochromene-3-carboxamide
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C16H11ClN2O3
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0049396
 Compound Info 
N-[(2-aminopyrimidin-5-yl)methyl]-N'-(4-chloro-3-fluorophenyl)oxamide
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C13H11ClFN5O2
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0049397
 Compound Info 
N-(4-chloro-3-fluorophenyl)-N'-(3-cyano-5,5,7,7-tetramethyl-4,6-dihydrothieno[2,3-c]pyridin-2-yl)oxamide
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C20H20ClFN4O2S
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0049398
 Compound Info 
N'-(4-chloro-2-fluorophenyl)-N-(2,2,6,6-tetramethylpiperidin-4-yl)oxamide
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C17H23ClFN3O2
  1
1
IC50 > 100000 nM
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CP0049399
 Compound Info 
N-[[(1S,9aR)-2,3,4,6,7,8,9,9a-octahydro-1H-quinolizin-1-yl]methyl]-N'-(4-chloro-3-fluorophenyl)oxamide
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C18H23ClFN3O2
  1
1
IC50 > 100000 nM
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CP0049400
 Compound Info 
N-(4-chloro-3-fluorophenyl)-N'-[1-(2-ethyl-1,2,4-triazol-3-yl)ethyl]oxamide
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C14H15ClFN5O2
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0049401
 Compound Info 
N'-(4-chloro-3-fluorophenyl)-N-[[4-(dimethylamino)-1-methylpiperidin-4-yl]methyl]oxamide
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C17H24ClFN4O2
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0049402
 Compound Info 
N'-(4-chloro-3-fluorophenyl)-N-[2-(2,6-dimethylmorpholin-4-yl)ethyl]oxamide
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C16H21ClFN3O3
  1
1
IC50 > 100000 nM
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CP0049403
 Compound Info 
4-(2-(4-chloro-3-fluorophenylamino)-2-oxoacetamido)-1,2,2,6,6-pentamethylpiperidine 1-oxide
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C18H25ClFN3O3
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0049404
 Compound Info 
N'-(4-chloro-3-fluorophenyl)-N-(3,3,5,5-tetramethylcyclohexyl)oxamide
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C18H24ClFN2O2
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0055745
 Compound Info 
2,2,6,6-tetramethyl-4-(2-methyl-3-oxo-3,4-dihydro-2H-benzo[b][1,4]thiazine-7-carboxamido)piperidinium
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C19H27N3O2S
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0081497
 Compound Info 
N-(4-bromophenyl)-3-(4-propan-2-ylpiperidin-1-yl)propanamide
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C17H25BrN2O
  1
1
IC50 > 100000 nM
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CP0081499
 Compound Info 
(3S)-1-(3-(4-chlorophenylamino)-3-oxopropyl)-3-methylpiperidinium
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C15H21ClN2O
  1
1
IC50 > 100000 nM
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CP0083290
 Compound Info 
N'-(4-chloro-3-fluorophenyl)-N-[2-(dimethylamino)-2-pyrrolidin-1-ylethyl]oxamide
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C16H22ClFN4O2
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0083292
 Compound Info 
N-(4-chlorophenyl)-2-[(6-methyl-2-oxo-1H-pyrimidin-4-yl)sulfanyl]acetamide
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C13H12ClN3O2S
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0098492
 Compound Info 
4-(2-(4-chlorophenethylamino)-2-oxoacetamido)-2,2,6,6-tetramethylpiperidinium
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C19H28ClN3O2
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0108700
 Compound Info 
N'-(4-chloro-2-phenylmethoxyphenyl)-N-(2,2,6,6-tetramethylpiperidin-4-yl)oxamide
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C24H30ClN3O3
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0108701
 Compound Info 
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-N'-(4-chloro-3-fluorophenyl)oxamide
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C16H18ClFN4O2
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0108795
 Compound Info 
N'-(4-chloro-3-fluorophenyl)-N-(piperidin-4-ylmethyl)oxamide
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C14H17ClFN3O2
  1
1
IC50 > 100000 nM
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CP0108796
 Compound Info 
N'-(4-bromophenyl)-N-(2,2,6,6-tetramethylpiperidin-4-yl)butanediamide
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C19H28BrN3O2
  1
1
IC50 > 100000 nM
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CP0117351
 Compound Info 
(S)-3-(3-(4-chlorophenoxy)-2-hydroxypropyl)-5,5-dimethylimidazolidine-2,4-dione
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C14H17ClN2O4
  1
1
IC50 > 100000 nM
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CP0117353
 Compound Info 
(R)-N1-(1,4-dioxaspiro[4.4]nonan-2-ylmethyl)-N2-(4-chlorophenyl)oxalamide
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C16H19ClN2O4
  1
1
IC50 > 100000 nM
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CP0117355
 Compound Info 
4-(2-(4-bromophenylamino)-2-oxoethyl)-N-ethylpiperazine-1-carbimidothioic acid
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C15H21BrN4OS
  1
1
IC50 > 100000 nM
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CP0144840
 Compound Info 
N'-(3-propan-2-ylphenyl)-N-(2,2,6,6-tetramethylpiperidin-4-yl)oxamide
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C20H31N3O2
  1
1
IC50 > 100000 nM
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CP0144841
 Compound Info 
(R)-2-(6-amino-4-oxo-1,4-dihydropyrimidin-2-ylthio)-N-(4-chlorophenyl)propanamide
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C13H13ClN4O2S
  1
1
IC50 > 100000 nM
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CP0145109
 Compound Info 
N-(4-bromophenyl)-2-[(5-oxo-1,2-dihydropyrazol-3-yl)methylsulfanyl]acetamide
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C12H12BrN3O2S
  1
1
IC50 > 100000 nM
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CP0145111
 Compound Info 
1-(but-1-en-2-yl)-2-(5-(2-ethylcyclopentyl)-2,3-dimethylenepentyl)-3,4-dimethylcyclopenta-1,3-diene
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C17H25N3O4S
  1
1
IC50 > 100000 nM
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CP0162780
 Compound Info 
N-(4-bromophenyl)-3-[3-(hydroxymethyl)anilino]butanamide
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C17H19BrN2O2
  1
1
IC50 > 100000 nM
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CP0162781
 Compound Info 
1-[3-(4-bromoanilino)-3-oxopropyl]piperidine-4-carboxamide
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C15H20BrN3O2
  1
1
IC50 > 100000 nM
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CP0214324
 Compound Info 
N'-(4-chloro-3-fluorophenyl)-N-[(1-methylpiperidin-4-yl)methyl]oxamide
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C15H19ClFN3O2
  1
1
IC50 > 100000 nM
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CP0214332
 Compound Info 
N'-(4-azidophenyl)-N-(2,2,6,6-tetramethylpiperidin-4-yl)oxamide
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C17H24N6O2
  1
1
IC50 > 100000 nM
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CP0223620
 Compound Info 
N'-(4-chloro-2-methoxyphenyl)-N-(2,2,6,6-tetramethylpiperidin-4-yl)oxamide
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C18H26ClN3O3
  1
1
IC50 > 100000 nM
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CP0223621
 Compound Info 
N'-[4-chloro-2-(trifluoromethyl)phenyl]-N-(2,2,6,6-tetramethylpiperidin-4-yl)oxamide
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C18H23ClF3N3O2
  1
1
IC50 > 100000 nM
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CP0223622
 Compound Info 
N-(4-chloro-3-fluorophenyl)-N'-[1-(3-oxo-4H-1,4-benzoxazin-6-yl)ethyl]oxamide
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C18H15ClFN3O4
  1
1
IC50 > 100000 nM
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CP0223623
 Compound Info 
N-(4-chloro-3-fluorophenyl)-N'-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-3-yl)oxamide
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C14H13ClFN5O2
  1
1
IC50 > 100000 nM
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CP0225663
 Compound Info 
N'-(4-chloro-3-fluorophenyl)-N-[2-(4-methylpiperazin-1-yl)-2-thiophen-2-ylethyl]oxamide
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C19H22ClFN4O2S
  1
1
IC50 > 100000 nM
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CP0225665
 Compound Info 
3-(4-aminophenyl)-N-(4-chlorophenyl)-3-oxopropanamide
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C15H13ClN2O2
  1
1
IC50 > 100000 nM
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CP0228397
 Compound Info 
1-(2-(1H-imidazol-5-yl)ethyl)-3-(3,4-dichlorophenyl)urea
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C12H12Cl2N4O
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0228399
 Compound Info 
(S)-N-(4-bromophenyl)-2-(3-methoxyphenylamino)propanamide
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C16H17BrN2O2
  1
1
IC50 > 100000 nM
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CP0228401
 Compound Info 
N-(4-bromophenyl)-N'-naphthalen-1-yloxamide
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C18H13BrN2O2
  1
1
IC50 > 100000 nM
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CP0228421
 Compound Info 
N'-(4-chloro-2-methylphenyl)-N-(2,2,6,6-tetramethylpiperidin-4-yl)oxamide
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C18H26ClN3O2
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0228424
 Compound Info 
N'-(4-bromophenyl)-N-(2,2,6,6-tetramethylpiperidin-4-yl)propanediamide
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C18H26BrN3O2
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0228468
 Compound Info 
N'-(1H-pyrrolo[2,3-b]pyridin-3-yl)-N-(2,2,6,6-tetramethylpiperidin-4-yl)oxamide
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C18H25N5O2
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0232522
 Compound Info 
2-(4-chlorophenoxy)-N-(2,6-dioxo-1,2,3,6-tetrahydropyrimidin-4-yl)acetamide
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C12H10ClN3O4
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0234509
 Compound Info 
N-(4-chlorophenyl)-2-(1H-indol-3-yl)-2-oxoacetamide
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C16H11ClN2O2
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0234510
 Compound Info 
2-(5-chloropyridin-2-ylamino)-2-oxoethyl 1H-indazole-3-carboxylate
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C15H11ClN4O3
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0234511
 Compound Info 
N-(4-chlorophenyl)-7,7-dimethyl-2,5-dioxo-6,8-dihydro-1H-quinoline-3-carboxamide
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C18H17ClN2O3
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0234512
 Compound Info 
N'-(4-bromophenyl)-N-(3,4-dihydro-1H-isochromen-1-ylmethyl)oxamide
   Show/Hide
C18H17BrN2O3
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0234513
 Compound Info 
N-(4-bromophenyl)-3-(3-methylpiperidin-1-yl)propanamide
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C15H21BrN2O
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0237644
 Compound Info 
4-(2-(1H-indol-6-ylamino)-2-oxoacetamido)-2,2,6,6-tetramethylpiperidinium
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C19H26N4O2
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0237645
 Compound Info 
N'-(4-bromophenyl)-N-(furan-2-ylmethyl)oxamide
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C13H11BrN2O3
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0237647
 Compound Info 
N-(4-bromophenyl)-2-[(1,3-dimethylpyrazol-4-yl)methyl-methylamino]acetamide
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C15H19BrN4O
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0239700
 Compound Info 
N'-(4-chlorophenyl)-N-[(3-methoxyphenyl)methyl]oxamide
   Show/Hide
C16H15ClN2O3
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0239701
 Compound Info 
N-(4-bromo-3-methylphenyl)-2-(1H-indol-3-yl)-2-oxoacetamide
   Show/Hide
C17H13BrN2O2
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0239739
 Compound Info 
N'-(4-chloro-3-fluorophenyl)-N-[[4-(methylcarbamoyl)phenyl]methyl]oxamide
   Show/Hide
C17H15ClFN3O3
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0239741
 Compound Info 
N'-(4-chloro-3-fluorophenyl)-N-(1,4,5,6,7,8-hexahydrocyclohepta[c]pyrazol-3-ylmethyl)oxamide
   Show/Hide
C17H18ClFN4O2
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0239742
 Compound Info 
N'-(4-chloro-3-fluorophenyl)-N-[2-(furan-2-yl)-2-pyrrolidin-1-ylethyl]oxamide
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C18H19ClFN3O3
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0239748
 Compound Info 
1-(4-chlorophenyl)-3-(9H-purin-6-yl)urea
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C12H9ClN6O
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0257953
 Compound Info 
2-(4-chloro-3-methylphenoxy)-N-(1H-1,2,4-triazol-5-ylmethyl)acetamide
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C12H13ClN4O2
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0272722
 Compound Info 
N'-(4-chloro-3-fluorophenyl)-N-[2-(2-methylpiperidin-1-yl)propyl]oxamide
   Show/Hide
C17H23ClFN3O2
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0272724
 Compound Info 
N'-(4-chloro-2-ethoxyphenyl)-N-(2,2,6,6-tetramethylpiperidin-4-yl)oxamide
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C19H28ClN3O3
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0272725
 Compound Info 
3,4-dichloro-N-(1,3-dioxoisoindolin-5-yl)benzamide
   Show/Hide
C15H8Cl2N2O3
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0281507
 Compound Info 
N-(1-benzoylpiperidin-4-yl)-N'-(4-chloro-3-fluorophenyl)oxamide
   Show/Hide
C20H19ClFN3O3
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0282020
 Compound Info 
N-(4-chloro-3-fluorophenyl)-N'-(1H-indazol-4-yl)oxamide
   Show/Hide
C15H10ClFN4O2
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0282021
 Compound Info 
N-(4-chloro-3-fluorophenyl)-N'-(1-methylpiperidin-3-yl)oxyoxamide
   Show/Hide
C14H17ClFN3O3
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0282023
 Compound Info 
N'-(4-chloro-3-propan-2-yloxyphenyl)-N-(2,2,6,6-tetramethylpiperidin-4-yl)oxamide
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C20H30ClN3O3
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0282028
 Compound Info 
N'-(4-chloro-3-fluorophenyl)-N-(1-propan-2-ylpiperidin-4-yl)oxamide
   Show/Hide
C16H21ClFN3O2
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0282034
 Compound Info 
4-(2-(4-chlorophenoxy)acetyl)-1-methyl-1,4-diazepan-1-ium
   Show/Hide
C14H19ClN2O2
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0282035
 Compound Info 
N-(4-chlorophenyl)-3-(2-hydroxy-3-methylphenyl)-1H-pyrazole-5-carboxamide
   Show/Hide
C17H14ClN3O2
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0282781
 Compound Info 
N'-(4-chloro-3-fluorophenyl)-N-[[1-(2-morpholin-4-ylethyl)pyrrolidin-3-yl]methyl]oxamide
   Show/Hide
C19H26ClFN4O3
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0282783
 Compound Info 
N'-(4-chloro-3-fluorophenyl)-N-(1-methylpiperidin-3-yl)oxamide
   Show/Hide
C14H17ClFN3O2
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0282784
 Compound Info 
N'-(4-chloro-3-fluorophenyl)-N-(1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl)oxamide
   Show/Hide
C18H22ClFN2O2
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0282786
 Compound Info 
4-(3-(2,4-dichlorophenyl)ureido)-1-methylpiperidinium
   Show/Hide
C13H17Cl2N3O
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0282806
 Compound Info 
N'-(4-chloro-3-fluorophenyl)-N-(2,2,6,6-tetramethyloxan-4-yl)oxamide
   Show/Hide
C17H22ClFN2O3
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0282818
 Compound Info 
N'-naphthalen-2-yl-N-(2,2,6,6-tetramethylpiperidin-4-yl)oxamide
   Show/Hide
C21H27N3O2
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0283380
 Compound Info 
N'-(4-chloro-3-fluorophenyl)-N-[[4-(methylsulfamoylmethyl)phenyl]methyl]oxamide
   Show/Hide
C17H17ClFN3O4S
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0283386
 Compound Info 
N'-(4-chloro-3-fluorophenyl)-N-[2-(dimethylamino)-2-(furan-2-yl)ethyl]oxamide
   Show/Hide
C16H17ClFN3O3
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0285133
 Compound Info 
N-(1,3-benzodioxol-5-ylmethyl)-N'-(4-bromophenyl)oxamide
   Show/Hide
C16H13BrN2O4
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0285135
 Compound Info 
(3S)-1-(3-(4-bromophenylamino)-3-oxopropyl)-3-(ethoxycarbonyl)piperidinium
   Show/Hide
C17H23BrN2O3
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0288895
 Compound Info 
(S)-N1-(1-benzylpyrrolidin-3-yl)-N2-(4-chloro-3-fluorophenyl)oxalamide
   Show/Hide
C19H19ClFN3O2
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0288935
 Compound Info 
N'-(2-propan-2-ylphenyl)-N-(2,2,6,6-tetramethylpiperidin-4-yl)oxamide
   Show/Hide
C20H31N3O2
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0288937
 Compound Info 
3,6-dichloro-N-(2-oxo-1,2-dihydropyrimidin-4-yl)benzo[b]thiophene-2-carboxamide
   Show/Hide
C13H7Cl2N3O2S
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0292435
 Compound Info 
N'-[4-(4-phenyltriazol-1-yl)phenyl]-N-(2,2,6,6-tetramethylpiperidin-4-yl)oxamide
   Show/Hide
C25H30N6O2
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0293016
 Compound Info 
N-(4-chloro-3-fluorophenyl)-N'-[1-(4-sulfamoylphenyl)ethyl]oxamide
   Show/Hide
C16H15ClFN3O4S
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0293018
 Compound Info 
N'-(2,4-dichlorophenyl)-N-(2,2,6,6-tetramethylpiperidin-4-yl)oxamide
   Show/Hide
C17H23Cl2N3O2
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0293021
 Compound Info 
N'-(4-chloro-3-fluorophenyl)-N-[4,4,4-trifluoro-3-hydroxy-3-(1-methylimidazol-2-yl)butyl]oxamide
   Show/Hide
C16H15ClF4N4O3
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0293026
 Compound Info 
N'-(4-chloro-3-fluorophenyl)-N-(1-methylpiperidin-4-yl)oxamide
   Show/Hide
C14H17ClFN3O2
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0293027
 Compound Info 
N-(4-chloro-3-fluorophenyl)-N'-methyl-N'-(2,2,6,6-tetramethylpiperidin-4-yl)oxamide
   Show/Hide
C18H25ClFN3O2
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0293028
 Compound Info 
N'-(4-chlorophenyl)-N'-methyl-N-(2,2,6,6-tetramethylpiperidin-4-yl)oxamide
   Show/Hide
C18H26ClN3O2
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0296370
 Compound Info 
N'-(4-chloro-3-methoxyphenyl)-N-(2,2,6,6-tetramethylpiperidin-4-yl)oxamide
   Show/Hide
C18H26ClN3O3
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0296372
 Compound Info 
N'-[4-chloro-2-(2-methylpropoxy)phenyl]-N-(2,2,6,6-tetramethylpiperidin-4-yl)oxamide
   Show/Hide
C21H32ClN3O3
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0296373
 Compound Info 
2-(4-chlorophenoxy)-N-(2-oxo-2,3-dihydro-1H-benzo[d]imidazol-5-yl)acetamide
   Show/Hide
C15H12ClN3O3
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0296375
 Compound Info 
N-(4-chlorophenyl)-2-[(2-oxo-5,6,7,8-tetrahydro-1H-quinazolin-4-yl)sulfanyl]acetamide
   Show/Hide
C16H16ClN3O2S
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0296386
 Compound Info 
N-(4-chloro-3-fluorophenyl)-2-[(2,2,6,6-tetramethylpiperidin-4-yl)amino]acetamide
   Show/Hide
C17H25ClFN3O
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0304498
 Compound Info 
2-(4-chlorophenoxy)-N-(5-(dimethylamino)-2-methylphenyl)acetamide
   Show/Hide
C17H19ClN2O2
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0304499
 Compound Info 
(2R,6S)-4-(3-(4-bromophenylamino)-3-oxopropyl)-2,6-dimethylmorpholin-4-ium
   Show/Hide
C15H21BrN2O2
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0304538
 Compound Info 
N'-(4-chloro-3-fluorophenyl)-N-[2-(diethylamino)-4-methylpentyl]oxamide
   Show/Hide
C18H27ClFN3O2
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0304539
 Compound Info 
N'-(4-chloro-3-fluorophenyl)-N-(2-methyl-2-morpholin-4-ylpropyl)oxamide
   Show/Hide
C16H21ClFN3O3
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0304541
 Compound Info 
N'-(4-chloro-3-fluorophenyl)-N-(1-propylpiperidin-4-yl)oxamide
   Show/Hide
C16H21ClFN3O2
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0311443
 Compound Info 
N'-(4-chloro-3-phenylmethoxyphenyl)-N-(2,2,6,6-tetramethylpiperidin-4-yl)oxamide
   Show/Hide
C24H30ClN3O3
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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   TS
CP0311444
 Compound Info 
N-(4-chlorophenyl)-2-oxo-5,6,7,8-tetrahydro-1H-quinoline-3-carboxamide
   Show/Hide
C16H15ClN2O2
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0311453
 Compound Info 
N'-(4-chloro-3-fluorophenyl)-N-(4,5,6,7-tetrahydro-1H-indazol-5-yl)oxamide
   Show/Hide
C15H14ClFN4O2
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0311454
 Compound Info 
N'-(4-chloro-3-fluorophenyl)-N-[(1-ethylpiperidin-4-yl)methyl]oxamide
   Show/Hide
C16H21ClFN3O2
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0314007
 Compound Info 
N'-(3-phenylmethoxyphenyl)-N-(2,2,6,6-tetramethylpiperidin-4-yl)oxamide
   Show/Hide
C24H31N3O3
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0314008
 Compound Info 
(S)-N-(4-chlorophenyl)-3-(4-hydroxy-4,5,5-trimethyl-2-oxooxazolidin-3-yl)propanamide
   Show/Hide
C15H19ClN2O4
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0369087
 Compound Info 
N-(4-chloro-3-fluorophenyl)-N'-(4,5-diethyl-1H-pyrazol-3-yl)oxamide
   Show/Hide
C15H16ClFN4O2
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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   TS
CP0369088
 Compound Info 
N'-(4-chloro-3-fluorophenyl)-N-[(1-methylpiperidin-3-yl)methyl]oxamide
   Show/Hide
C15H19ClFN3O2
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0369089
 Compound Info 
4-(3-((4-(4,4-dimethylpent-1-en-2-yl)cyclohexyl)methyl)-2-methylenebut-3-enyl)-1,2-dimethylbenzene
   Show/Hide
C18H23ClFN3O4
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0369113
 Compound Info 
N'-[4-[4-(2-phenylethyl)triazol-1-yl]phenyl]-N-(2,2,6,6-tetramethylpiperidin-4-yl)oxamide
   Show/Hide
C27H34N6O2
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0369114
 Compound Info 
N'-[4-[4-(5-hydroxypentyl)triazol-1-yl]phenyl]-N-(2,2,6,6-tetramethylpiperidin-4-yl)oxamide
   Show/Hide
C24H36N6O3
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0370655
 Compound Info 
N'-(4-bromophenyl)-N-(2,3-dihydro-1,4-benzodioxin-3-ylmethyl)oxamide
   Show/Hide
C17H15BrN2O4
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0371081
 Compound Info 
2,2,6,6-tetramethyl-4-(2-(4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)hydrazono)piperidinium
   Show/Hide
C17H27N5O
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0371082
 Compound Info 
N-(4-chlorophenyl)-N'-(3-methoxyphenyl)oxamide
   Show/Hide
C15H13ClN2O3
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0371083
 Compound Info 
2-(azepan-1-yl)-N-(4-bromophenyl)acetamide
   Show/Hide
C14H19BrN2O
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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CP0499758
 Compound Info 
(S)-N-(4-chlorophenyl)-2-(4,6-diaminopyrimidin-2-ylthio)propanamide
   Show/Hide
C13H14ClN5OS
  1
1
IC50 > 100000 nM
 Bioactivity Info 
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Biochemical Assays
Compound ID Compound Name Compound Formula
CP0304542
 Compound Info 
N'-(4-chloro-3-fluorophenyl)-N-(1,2,2,6,6-pentamethylpiperidin-4-yl)oxamide
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C18H25ClFN3O2
  1
1 Kd = 300 nM
CP0144831
 Compound Info 
N-(5-azaspiro[3.5]nonan-8-yl)-N'-(4-chloro-3-fluorophenyl)oxamide
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C16H19ClFN3O2
  1
1 Kd = 600 nM
CP0282807
 Compound Info 
N'-(4-chloro-3-fluorophenyl)-N-(2,2,6,6-tetramethylpiperidin-4-yl)oxamide
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C17H23ClFN3O2
  1
1 Kd = 760 nM
CP0282806
 Compound Info 
N'-(4-chloro-3-fluorophenyl)-N-(2,2,6,6-tetramethyloxan-4-yl)oxamide
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C17H22ClFN2O3
  1
1 Kd = 1000 nM
CP0293020
 Compound Info 
N'-(4-chloro-3-fluorophenyl)-N-(1,2,3,4-tetrahydroisoquinolin-1-ylmethyl)oxamide
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C18H17ClFN3O2
  1
1 Kd = 1200 nM
CP0049403
 Compound Info 
4-(2-(4-chloro-3-fluorophenylamino)-2-oxoacetamido)-1,2,2,6,6-pentamethylpiperidine 1-oxide
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C18H25ClFN3O3
  1
1 Kd = 1300 nM
CP0282780
 Compound Info 
N'-(4-chloro-3-fluorophenyl)-N-[2-[(2S,6R)-2,6-dimethylpiperidin-1-yl]ethyl]oxamide
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C17H23ClFN3O2
  1
1 Kd = 1600 nM
CP0283381
 Compound Info 
N'-(4-chloro-3-fluorophenyl)-N-[(1-cyclopropylpyrrolidin-3-yl)methyl]oxamide
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C16H19ClFN3O2
  1
1 Kd = 1700 nM
CP0282028
 Compound Info 
N'-(4-chloro-3-fluorophenyl)-N-(1-propan-2-ylpiperidin-4-yl)oxamide
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C16H21ClFN3O2
  1
1 Kd = 1900 nM
CP0228423
 Compound Info 
N'-(4-chloro-3-fluorophenyl)-N-[(1-ethylpyrrolidin-2-yl)methyl]oxamide
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C15H19ClFN3O2
  1
1 Kd = 2100 nM
CP0283382
 Compound Info 
N'-(4-chloro-3-fluorophenyl)-N-[(2,2,6,6-tetramethylpiperidin-4-yl)methyl]oxamide
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C18H25ClFN3O2
  1
1 Kd = 2200 nM
CP0296385
 Compound Info 
N'-(4-chloro-3-fluorophenyl)-N-[2-(1-propan-2-ylpiperidin-2-yl)ethyl]oxamide
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C18H25ClFN3O2
  1
1 Kd = 2300 nM
CP0228422
 Compound Info 
N'-(4-chloro-3-fluorophenyl)-N-(1-cyclohexylpyrrolidin-3-yl)oxamide
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C18H23ClFN3O2
  1
1 Kd = 2400 nM
CP0369088
 Compound Info 
N'-(4-chloro-3-fluorophenyl)-N-[(1-methylpiperidin-3-yl)methyl]oxamide
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C15H19ClFN3O2
  1
1 Kd = 2500 nM
CP0282779
 Compound Info 
N-[[(4S,5S)-5-(aminomethyl)-2,2-dimethyl-1,3-dioxolan-4-yl]methyl]-N'-(4-chloro-3-fluorophenyl)oxamide
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C15H19ClFN3O4
  1
1 Kd = 2600 nM
CP0108795
 Compound Info 
N'-(4-chloro-3-fluorophenyl)-N-(piperidin-4-ylmethyl)oxamide
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C14H17ClFN3O2
  1
1 Kd = 3000 nM
CP0144832
 Compound Info 
N-[[(3aS,6aS)-2,3,4,5,6,6a-hexahydro-1H-cyclopenta[c]pyrrol-3a-yl]methyl]-N'-(4-chloro-3-fluorophenyl)oxamide
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C16H19ClFN3O2
  1
1 Kd = 3100 nM
CP0296382
 Compound Info 
N'-(4-chloro-3-fluorophenyl)-N-[[1-(2-hydroxyethyl)piperidin-3-yl]methyl]oxamide
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C16H21ClFN3O3
  1
1 Kd = 3200 nM
CP0144833
 Compound Info 
N'-(4-chloro-3-fluorophenyl)-N-(1-propylpiperidin-3-yl)oxamide
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C16H21ClFN3O2
  1
1 Kd = 3300 nM
CP0311454
 Compound Info 
N'-(4-chloro-3-fluorophenyl)-N-[(1-ethylpiperidin-4-yl)methyl]oxamide
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C16H21ClFN3O2
  1
1 Kd = 3400 nM
CP0214321
 Compound Info 
N'-(4-chlorophenyl)-N-(2,2,6,6-tetramethylpiperidin-4-yl)oxamide
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C17H24ClN3O2
  1
1 Kd = 3700 nM
CP0108705
 Compound Info 
N'-(4-chloro-3-fluorophenyl)-N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]oxamide
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C14H14ClFN4O2
  1
1 Kd = 4000 nM
CP0282783
 Compound Info 
N'-(4-chloro-3-fluorophenyl)-N-(1-methylpiperidin-3-yl)oxamide
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C14H17ClFN3O2
  1
1 Kd = 4200 nM
CP0304541
 Compound Info 
N'-(4-chloro-3-fluorophenyl)-N-(1-propylpiperidin-4-yl)oxamide
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C16H21ClFN3O2
  1
1 Kd = 4200 nM
CP0214324
 Compound Info 
N'-(4-chloro-3-fluorophenyl)-N-[(1-methylpiperidin-4-yl)methyl]oxamide
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C15H19ClFN3O2
  1
1 Kd = 4300 nM
CP0293026
 Compound Info 
N'-(4-chloro-3-fluorophenyl)-N-(1-methylpiperidin-4-yl)oxamide
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C14H17ClFN3O2
  1
1 Kd = 9400 nM