General Information of the Protein
Protein ID
PT02466
Protein Name
Opioid growth factor receptor-like protein 1
Gene Name
OGFRL1
Sequence
MGNLLGGVSFREPTTVEDCDSTWQTDSEPEPEEPGPGGGSEGPGQESEQPAQPPEQAGGRPGASPAPDEDAEAAGAEQGGDSTEATAKPKRSFYAARDLYKYRHQYPNFKDIRYQNDLSNLRFYKNKIPFKPDGVYIEEVLSKWKGDYEKLEHNHTYIQWLFPLREQGLNFYAKELTTYEIEEFKKTKEAIRRFLLAYKMMLEFFGIKLTDKTGNVARAVNWQERFQHLNESQHNYLRITRILKSLGELGYESFKSPLVKFILHEALVENTIPNIKQSALEYFVYTIRDRRERRKLLRFAQKHYTPSENFIWGPPRKEQSEGSKAQKMSSPLASSHNSQTSMHKKAKDSKNSSSAVHLNSKTAEDKKVAPKEPVEETDRPSPEPSNEAAKPRNTEKDSNAENMNSQPEKTVTTPTEKKESVSPENNEEGGNDNQDNENPGNTNCHDVVLVQ
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Organism
Homo sapiens, Human
Protein Classification
Membrane receptor
Uniprot ID
Primary ID:
Q5TC84

Secondarily ID:
Q2TAC1
Q8NEQ4
Q9H7B5
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HGNC ID
HGNC:21378
Map of Molecular Bioactivity Related to the Protein
Map of Molecular Bioactivity Related to the Protein

Protein
Cell Line
Compound

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Protein
Cell Line ID: CL000006 , HEK293
Compound ID Compound Name Compound Formula
CP0086136
US8476271, 405
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C27H35N3O3
 2
1
EC50 = 0.55 nM
   TI
   LI
   LO
   TS
2
Ki = 1.1 nM
   TI
   LI
   LO
   TS
CP0109897
US8846929, 362
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C26H33N3O3
 2
1
EC50 = 4.03 nM
   TI
   LI
   LO
   TS
2
Ki = 2.4 nM
   TI
   LI
   LO
   TS
CP0129542
US8476271, 97
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C25H31N3O3
 2
1
EC50 = 57.2 nM
   TI
   LI
   LO
   TS
2
Ki = 5.7 nM
   TI
   LI
   LO
   TS
CP0279176
US8476271, 18
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C27H37N3O3
 2
1
EC50 = 62.6 nM
   TI
   LI
   LO
   TS
2
Ki = 9 nM
   TI
   LI
   LO
   TS
CP0478850
US9145408, 369
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C26H34N4O3
 2
1
EC50 = 545 nM
   TI
   LI
   LO
   TS
2
Ki = 178 nM
   TI
   LI
   LO
   TS
CP0223449
US8846929, 356
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C28H39N3O3
 2
1
EC50 = 686 nM
   TI
   LI
   LO
   TS
2
Ki = 43.1 nM
   TI
   LI
   LO
   TS
CP0413438
US9145408, 360
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C25H31N3O3
 2
1
EC50 = 1667.1 nM
   TI
   LI
   LO
   TS
2
Ki = 202.8 nM
   TI
   LI
   LO
   TS
CP0400515
US8969358, 101
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C33H41N3O4
 1
1
Ki = 228.55 nM
   TI
   LI
   LO
   TS
CP0881219
US9096606, 5
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C34H40NO4S+
 1
1
Ki = 18166.45 nM
   TI
   LI
   LO
   TS
CP0442217
US9096606, 23
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C35H44F2NO4+
 1
1
Ki > 20000 nM
   TI
   LI
   LO
   TS
CP0858784
US9096606, 8
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C34H44NO5+
 1
1
Ki > 20000 nM
   TI
   LI
   LO
   TS
CP0881759
US9096606, 6
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C33H42NO4+
 1
1
Ki > 20000 nM
   TI
   LI
   LO
   TS
CP0906694
US9096606, 3
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C34H44NO4+
 1
1
Ki > 20000 nM
   TI
   LI
   LO
   TS
CP0924248
US9096606, 2
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C34H41ClNO6+
 1
1
Ki > 20000 nM
   TI
   LI
   LO
   TS
CP0935636
US9096606, 4
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C32H39FNO4+
 1
1
Ki > 20000 nM
   TI
   LI
   LO
   TS
CP0955002
US9096606, 1
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C33H40Cl2NO4+
 1
1
Ki > 20000 nM
   TI
   LI
   LO
   TS