| Compound ID |
Compound Name |
Compound Formula |
|
CP0546991
|
3-[[(2S)-2-[(4-benzoylbenzoyl)amino]-2-(4-phenylmethoxyphenyl)acetyl]amino]benzamide
Show/Hide
|
C36H29N3O5
|
1
|
| 1 |
EC50 = 390 nM
|
|
|
|
CP0492600
|
N-[(1S)-2-[[4-(diaminomethylideneamino)phenyl]methylamino]-2-oxo-1-(4-phenylmethoxyphenyl)ethyl]hexanamide;2,2,2-trifluoroacetic acid
Show/Hide
|
C31H36F3N5O5
|
1
|
| 1 |
EC50 = 490 nM
|
|
|
|
CP0369204
|
N-[(1S)-2-[[4-(diaminomethylideneamino)phenyl]methylamino]-2-oxo-1-(4-phenylmethoxyphenyl)ethyl]heptanamide;2,2,2-trifluoroacetic acid
Show/Hide
|
C32H38F3N5O5
|
1
|
| 1 |
EC50 = 520 nM
|
|
|
|
CP0543002
|
3-(cyclohexylmethoxy)-N-(1-hydroxy-3H-2,1-benzoxaborol-6-yl)benzamide
Show/Hide
|
C21H24BNO4
|
1
|
| 1 |
EC50 = 540 nM
|
|
|
|
CP0570836
|
3-[[(2S)-2-[[4-(4-chlorophenoxy)benzoyl]amino]-2-(4-phenylmethoxyphenyl)acetyl]amino]benzamide
Show/Hide
|
C35H28ClN3O5
|
1
|
| 1 |
EC50 = 580 nM
|
|
|
|
CP0531603
|
3-[[(2S)-2-[(4-phenoxybenzoyl)amino]-2-(4-phenylmethoxyphenyl)acetyl]amino]benzamide
Show/Hide
|
C35H29N3O5
|
1
|
| 1 |
EC50 = 730 nM
|
|
|
|
CP0369205
|
N-[(1S)-2-[[4-(diaminomethylideneamino)phenyl]methylamino]-2-oxo-1-(4-phenylmethoxyphenyl)ethyl]octanamide;2,2,2-trifluoroacetic acid
Show/Hide
|
C33H40F3N5O5
|
1
|
| 1 |
EC50 = 830 nM
|
|
|
|
CP0491975
|
3-[[(2S)-2-[[4-(3-chlorophenoxy)benzoyl]amino]-2-(4-phenylmethoxyphenyl)acetyl]amino]benzamide
Show/Hide
|
C35H28ClN3O5
|
1
|
| 1 |
EC50 = 1000 nM
|
|
|
|
CP0546990
|
4-[[[(2S)-2-[(4-phenoxybenzoyl)amino]-2-(4-phenylmethoxyphenyl)acetyl]amino]methyl]benzamide
Show/Hide
|
C36H31N3O5
|
1
|
| 1 |
EC50 = 1000 nM
|
|
|
|
CP0552992
|
3-[[(2S)-2-[[4-(4-cyanophenoxy)benzoyl]amino]-2-(4-phenylmethoxyphenyl)acetyl]amino]benzamide
Show/Hide
|
C36H28N4O5
|
1
|
| 1 |
EC50 = 1000 nM
|
|
|
|
CP0577235
|
N-(1-hydroxy-3H-2,1-benzoxaborol-6-yl)-3-[(3-methoxyphenyl)methoxy]benzamide
Show/Hide
|
C22H20BNO5
|
1
|
| 1 |
EC50 = 1100 nM
|
|
|
|
CP0491966
|
3-[[(2S)-2-(4-phenylmethoxyphenyl)-2-[[4-[4-(trifluoromethyl)phenoxy]benzoyl]amino]acetyl]amino]benzamide
Show/Hide
|
C36H28F3N3O5
|
1
|
| 1 |
EC50 = 1200 nM
|
|
|
|
CP0491967
|
3-[[(2S)-2-[(4-benzoylbenzoyl)amino]-2-[4-[(3-methoxyphenyl)methoxy]phenyl]acetyl]amino]benzamide
Show/Hide
|
C37H31N3O6
|
1
|
| 1 |
EC50 = 1200 nM
|
|
|
|
CP0552402
|
3-[[(2S)-2-[[4-(4-chlorophenyl)benzoyl]amino]-2-(4-phenylmethoxyphenyl)acetyl]amino]benzamide
Show/Hide
|
C35H28ClN3O4
|
1
|
| 1 |
EC50 = 1200 nM
|
|
|
|
CP0531604
|
3-[[(2S)-2-[[4-(1,3-benzodioxol-5-yloxy)benzoyl]amino]-2-(4-phenylmethoxyphenyl)acetyl]amino]benzamide
Show/Hide
|
C36H29N3O7
|
1
|
| 1 |
EC50 = 1500 nM
|
|
|
|
CP0491974
|
3-[[(2S)-2-[(3-phenoxybenzoyl)amino]-2-(4-phenylmethoxyphenyl)acetyl]amino]benzamide
Show/Hide
|
C35H29N3O5
|
1
|
| 1 |
EC50 = 1700 nM
|
|
|
|
CP0491976
|
3-[[(2S)-2-[[5-(2,5-dimethylphenoxy)-2,2-dimethylpentanoyl]amino]-2-(4-phenylmethoxyphenyl)acetyl]amino]benzamide
Show/Hide
|
C37H41N3O5
|
1
|
| 1 |
EC50 = 1700 nM
|
|
|
|
CP0547008
|
3-[[(2S)-2-[(4-phenylbenzoyl)amino]-2-(4-phenylmethoxyphenyl)acetyl]amino]benzamide
Show/Hide
|
C35H29N3O4
|
1
|
| 1 |
EC50 = 1700 nM
|
|
|
|
CP0557760
|
3-[[(2S)-2-[[4-(furan-2-yl)benzoyl]amino]-2-(4-phenylmethoxyphenyl)acetyl]amino]benzamide
Show/Hide
|
C33H27N3O5
|
1
|
| 1 |
EC50 = 1700 nM
|
|
|
|
CP0121441
|
N-[(1S)-2-[[4-(diaminomethylideneamino)phenyl]methylamino]-2-oxo-1-(4-phenylmethoxyphenyl)ethyl]-4-phenylmethoxybenzamide;2,2,2-trifluoroacetic acid
Show/Hide
|
C39H36F3N5O6
|
1
|
| 1 |
EC50 = 2100 nM
|
|
|
|
CP0537494
|
3-[[(2S)-2-[4-[(3-methoxyphenyl)methoxy]phenyl]-2-[(4-phenoxybenzoyl)amino]acetyl]amino]benzamide
Show/Hide
|
C36H31N3O6
|
1
|
| 1 |
EC50 = 2100 nM
|
|
|
|
CP0268128
|
4-cyclohexyloxy-N-[(1S)-2-[[4-(diaminomethylideneamino)phenyl]methylamino]-2-oxo-1-(4-phenylmethoxyphenyl)ethyl]benzamide;2,2,2-trifluoroacetic acid
Show/Hide
|
C38H40F3N5O6
|
1
|
| 1 |
EC50 = 2200 nM
|
|
|
|
CP0547006
|
3-[[(2S)-2-[[4-(2-methoxyphenoxy)benzoyl]amino]-2-(4-phenylmethoxyphenyl)acetyl]amino]benzamide
Show/Hide
|
C36H31N3O6
|
1
|
| 1 |
EC50 = 2200 nM
|
|
|
|
CP0547010
|
3-[[(2S)-2-[(4-morpholin-4-ylbenzoyl)amino]-2-(4-phenylmethoxyphenyl)acetyl]amino]benzamide
Show/Hide
|
C33H32N4O5
|
1
|
| 1 |
EC50 = 2200 nM
|
|
|
|
CP0559450
|
3-[[(2S)-2-[4-[(2,6-dichlorophenyl)methoxy]phenyl]-2-[(4-phenoxybenzoyl)amino]acetyl]amino]benzamide
Show/Hide
|
C35H27Cl2N3O5
|
1
|
| 1 |
EC50 = 2200 nM
|
|
|
|
CP0570835
|
3-[[(2S)-2-(octanoylamino)-2-(4-phenylmethoxyphenyl)acetyl]amino]benzamide
Show/Hide
|
C30H35N3O4
|
1
|
| 1 |
EC50 = 2200 nM
|
|
|
|
CP0162723
|
N-[(1S)-2-[[4-(diaminomethylideneamino)phenyl]methylamino]-2-oxo-1-(4-phenylmethoxyphenyl)ethyl]decanamide;2,2,2-trifluoroacetic acid
Show/Hide
|
C35H44F3N5O5
|
1
|
| 1 |
EC50 = 2300 nM
|
|
|
|
CP0537495
|
3-[[(2S)-2-[4-[(2,6-dichlorophenyl)methoxy]phenyl]-2-(hexanoylamino)acetyl]amino]benzamide
Show/Hide
|
C28H29Cl2N3O4
|
1
|
| 1 |
EC50 = 2400 nM
|
|
|
|
CP0272845
|
3-[(2,6-dichlorophenyl)methoxy]-N-(1-hydroxy-3H-2,1-benzoxaborol-6-yl)benzamide
Show/Hide
|
C21H16BCl2NO4
|
1
|
| 1 |
EC50 = 2400 nM
|
|
|
|
CP0543001
|
N-(1-hydroxy-3H-2,1-benzoxaborol-6-yl)-6-phenylmethoxypyridine-2-carboxamide
Show/Hide
|
C20H17BN2O4
|
1
|
| 1 |
EC50 = 2400 nM
|
|
|
|
CP0568966
|
N-(1-hydroxy-3H-2,1-benzoxaborol-6-yl)-3-phenylmethoxybenzamide
Show/Hide
|
C21H18BNO4
|
1
|
| 1 |
EC50 = 2400 nM
|
|
|
|
CP0544642
|
N-(1-hydroxy-3H-2,1-benzoxaborol-6-yl)-3-[(3-methylphenyl)methoxy]benzamide
Show/Hide
|
C22H20BNO4
|
1
|
| 1 |
EC50 = 2500 nM
|
|
|
|
CP0268126
|
N-[(1S)-2-[[4-(diaminomethylideneamino)phenyl]methylamino]-2-oxo-1-(4-phenylmethoxyphenyl)ethyl]pentanamide;2,2,2-trifluoroacetic acid
Show/Hide
|
C30H34F3N5O5
|
1
|
| 1 |
EC50 = 2800 nM
|
|
|
|
CP0423117
|
N-[(1S)-2-[[4-(diaminomethylideneamino)phenyl]methylamino]-2-oxo-1-(4-phenylmethoxyphenyl)ethyl]-4-[(3-methoxyphenyl)methoxy]benzamide;2,2,2-trifluoroacetic acid
Show/Hide
|
C40H38F3N5O7
|
1
|
| 1 |
EC50 = 2900 nM
|
|
|
|
CP0531598
|
3-[[(2S)-2-[(4-phenoxybenzoyl)amino]-2-(4-phenoxyphenyl)acetyl]amino]benzamide
Show/Hide
|
C34H27N3O5
|
1
|
| 1 |
EC50 = 2900 nM
|
|
|
|
CP0495122
|
3-[(4-cyanophenyl)methoxy]-N-(1-hydroxy-3H-2,1-benzoxaborol-6-yl)benzamide
Show/Hide
|
C22H17BN2O4
|
1
|
| 1 |
EC50 = 2900 nM
|
|
|
|
CP0162721
|
N-[(1S)-2-[[4-(diaminomethylideneamino)phenyl]methylamino]-2-oxo-1-[4-[[4-(trifluoromethyl)phenyl]methoxy]phenyl]ethyl]hexanamide;2,2,2-trifluoroacetic acid
Show/Hide
|
C32H35F6N5O5
|
1
|
| 1 |
EC50 = 3000 nM
|
|
|
|
CP0524381
|
N-[(1S)-2-[[4-(diaminomethylideneamino)phenyl]methylamino]-2-oxo-1-(4-phenylmethoxyphenyl)ethyl]-4-phenoxybenzamide;2,2,2-trifluoroacetic acid
Show/Hide
|
C38H34F3N5O6
|
1
|
| 1 |
EC50 = 3000 nM
|
|
|
|
CP0570002
|
N-(1-hydroxy-3H-2,1-benzoxaborol-6-yl)-2-(3-phenoxyphenyl)propanamide
Show/Hide
|
C22H20BNO4
|
1
|
| 1 |
EC50 = 3100 nM
|
|
|
|
CP0343737
|
N-(1-hydroxy-3H-2,1-benzoxaborol-6-yl)-4-phenoxybenzamide
Show/Hide
|
C20H16BNO4
|
1
|
| 1 |
EC50 = 3500 nM
|
|
|
|
CP0547007
|
3-[[(2S)-2-[[4-(2,3-dihydro-1,4-benzodioxin-6-yloxy)benzoyl]amino]-2-(4-phenylmethoxyphenyl)acetyl]amino]benzamide
Show/Hide
|
C37H31N3O7
|
1
|
| 1 |
EC50 = 3800 nM
|
|
|
|
CP0537496
|
3-[[(2S)-2-[[4-[(3-oxo-1,2-dihydroinden-4-yl)oxy]benzoyl]amino]-2-(4-phenylmethoxyphenyl)acetyl]amino]benzamide
Show/Hide
|
C38H31N3O6
|
1
|
| 1 |
EC50 = 3900 nM
|
|
|
|
CP0531602
|
4-[[[(2S)-2-[(4-phenylmethoxybenzoyl)amino]-2-(4-phenylmethoxyphenyl)acetyl]amino]methyl]benzamide
Show/Hide
|
C37H33N3O5
|
1
|
| 1 |
EC50 = 4000 nM
|
|
|
|
CP0343735
|
benzyl N-(1-hydroxy-3H-2,1-benzoxaborol-6-yl)carbamate
Show/Hide
|
C15H14BNO4
|
1
|
| 1 |
EC50 = 4000 nM
|
|
|
|
CP0567960
|
3-[(4-chlorophenyl)methoxy]-N-(1-hydroxy-3H-2,1-benzoxaborol-6-yl)benzamide
Show/Hide
|
C21H17BClNO4
|
1
|
| 1 |
EC50 = 4100 nM
|
|
|
|
CP0268160
|
N-[(1S)-2-[[3-(aminomethyl)phenyl]methylamino]-2-oxo-1-(4-phenylmethoxyphenyl)ethyl]hexanamide
Show/Hide
|
C29H35N3O3
|
1
|
| 1 |
EC50 = 4200 nM
|
|
|
|
CP0552991
|
N-[(1S)-2-(3-carbamoylanilino)-2-oxo-1-(4-phenylmethoxyphenyl)ethyl]naphthalene-2-carboxamide
Show/Hide
|
C33H27N3O4
|
1
|
| 1 |
EC50 = 4500 nM
|
|
|
|
CP0419355
|
3-[[(2S)-2-(hexanoylamino)-2-(4-phenylmethoxyphenyl)acetyl]amino]benzamide
Show/Hide
|
C28H31N3O4
|
1
|
| 1 |
EC50 = 4600 nM
|
|
|
|
CP0571743
|
3-(benzylamino)-N-(1-hydroxy-3H-2,1-benzoxaborol-6-yl)benzamide
Show/Hide
|
C21H19BN2O3
|
1
|
| 1 |
EC50 = 5200 nM
|
|
|
|
CP0537493
|
N-[(1S)-2-(3-carbamoylanilino)-2-oxo-1-(4-phenylmethoxyphenyl)ethyl]-2,3-dihydro-1,4-benzodioxine-6-carboxamide
Show/Hide
|
C31H27N3O6
|
1
|
| 1 |
EC50 = 5400 nM
|
|
|
|
CP0162720
|
N-[(1S)-2-[[6-(diaminomethylideneamino)pyridin-3-yl]methylamino]-2-oxo-1-(4-phenylmethoxyphenyl)ethyl]hexanamide;2,2,2-trifluoroacetic acid
Show/Hide
|
C30H35F3N6O5
|
1
|
| 1 |
EC50 = 5900 nM
|
|
|
|
CP0272842
|
N-(1-hydroxy-3H-2,1-benzoxaborol-6-yl)-2-phenylmethoxybenzamide
Show/Hide
|
C21H18BNO4
|
1
|
| 1 |
EC50 = 6100 nM
|
|
|
|
CP0565236
|
N-[(1S)-2-[(4-carbamoylphenyl)methylamino]-2-oxo-1-(4-phenylmethoxyphenyl)ethyl]-5-thiophen-2-ylthiophene-2-carboxamide
Show/Hide
|
C32H27N3O4S2
|
1
|
| 1 |
EC50 = 6200 nM
|
|
|
|
CP0801855
|
(S)-N-(1-(4-(benzyloxy)phenyl)-2-(4-(guanidinomethyl)-benzylamino)-2-oxoethyl)hexanamide trifluoroacetic acid salt
Show/Hide
|
C32H38F3N5O5
|
1
|
| 1 |
EC50 = 6300 nM
|
|
|
|
CP0491968
|
4-[[[(2S)-2-(hexanoylamino)-2-(4-phenylmethoxyphenyl)acetyl]amino]methyl]benzamide
Show/Hide
|
C29H33N3O4
|
1
|
| 1 |
EC50 = 6300 nM
|
|
|
|
CP0544637
|
N-(1-hydroxy-3H-2,1-benzoxaborol-6-yl)-3-methoxybenzamide
Show/Hide
|
C15H14BNO4
|
1
|
| 1 |
EC50 = 6400 nM
|
|
|
|
CP0569607
|
N-(1-hydroxy-3H-2,1-benzoxaborol-6-yl)-3-phenoxybenzamide
Show/Hide
|
C20H16BNO4
|
1
|
| 1 |
EC50 = 6400 nM
|
|
|
|
CP0491972
|
N-[(1S)-2-[(4-carbamoylphenyl)methylamino]-2-oxo-1-(4-phenylmethoxyphenyl)ethyl]-1-benzothiophene-2-carboxamide
Show/Hide
|
C32H27N3O4S
|
1
|
| 1 |
EC50 = 6600 nM
|
|
|
|
CP0403576
|
N-[(1S)-2-[[4-[(dimethylamino)methyl]phenyl]methylamino]-2-oxo-1-(4-phenylmethoxyphenyl)ethyl]hexanamide
Show/Hide
|
C31H39N3O3
|
1
|
| 1 |
EC50 = 6700 nM
|
|
|
|
CP0773666
|
(S)-N-(2-(1H-Indazol-5-ylamino)-1-(4-(benzyloxy)phenyl)-2-oxoethyl)hexanamide
Show/Hide
|
C28H30N4O3
|
1
|
| 1 |
EC50 = 6900 nM
|
|
|
|
CP0491952
|
4-[[(2S)-2-(hexanoylamino)-2-(4-phenylmethoxyphenyl)acetyl]amino]benzamide
Show/Hide
|
C28H31N3O4
|
1
|
| 1 |
EC50 = 7000 nM
|
|
|
|
CP0423114
|
4-(4-chlorophenyl)-N-[(1S)-2-[[4-(diaminomethylideneamino)phenyl]methylamino]-2-oxo-1-(4-phenylmethoxyphenyl)ethyl]benzamide;2,2,2-trifluoroacetic acid
Show/Hide
|
C38H33ClF3N5O5
|
1
|
| 1 |
EC50 = 7100 nM
|
|
|
|
CP0068092
|
(3,4-Dihydroxy-5-nitro-phenyl)-p-tolyl-methanone
Show/Hide
|
C14H11NO5
|
1
|
| 1 |
EC50 = 7100 nM
|
|
|
|
CP0121439
|
N-[(1S)-2-[[4-(diaminomethylideneamino)phenyl]methylamino]-2-oxo-1-(4-phenylmethoxyphenyl)ethyl]-3-phenoxybenzamide;2,2,2-trifluoroacetic acid
Show/Hide
|
C38H34F3N5O6
|
1
|
| 1 |
EC50 = 7300 nM
|
|
|
|
CP0559447
|
4-[[[(2S)-2-(hexanoylamino)-2-[4-[(3-methoxyphenyl)methoxy]phenyl]acetyl]amino]methyl]benzamide
Show/Hide
|
C30H35N3O5
|
1
|
| 1 |
EC50 = 7300 nM
|
|
|
|
CP0268129
|
N-[(1S)-2-[[4-(diaminomethylideneamino)phenyl]methylamino]-2-oxo-1-(4-phenylmethoxyphenyl)ethyl]-4-phenylbenzamide;2,2,2-trifluoroacetic acid
Show/Hide
|
C38H34F3N5O5
|
1
|
| 1 |
EC50 = 7600 nM
|
|
|
|
CP0423115
|
N-[(1S)-2-[6-(diaminomethylideneamino)hexylamino]-2-oxo-1-(4-phenylmethoxyphenyl)ethyl]hexanamide
Show/Hide
|
C28H41N5O3
|
1
|
| 1 |
EC50 = 7700 nM
|
|
|
|
CP0562156
|
4-[2-[[(2S)-2-(hexanoylamino)-2-(4-phenylmethoxyphenyl)acetyl]amino]ethyl]benzamide
Show/Hide
|
C30H35N3O4
|
1
|
| 1 |
EC50 = 7700 nM
|
|
|
|
CP0557761
|
4-[[[(2S)-2-(heptanoylamino)-2-(4-phenylmethoxyphenyl)acetyl]amino]methyl]benzamide
Show/Hide
|
C30H35N3O4
|
1
|
| 1 |
EC50 = 7900 nM
|
|
|
|
CP0531599
|
3-[[(2S)-2-(4-phenylmethoxyphenyl)-2-[(4-pyrimidin-5-ylbenzoyl)amino]acetyl]amino]benzamide
Show/Hide
|
C33H27N5O4
|
1
|
| 1 |
EC50 = 8100 nM
|
|
|
|
CP0491965
|
4-[[[(2S)-2-[4-[(2,6-dichlorophenyl)methoxy]phenyl]-2-(hexanoylamino)acetyl]amino]methyl]benzamide
Show/Hide
|
C29H31Cl2N3O4
|
1
|
| 1 |
EC50 = 8300 nM
|
|
|
|
CP0562151
|
N-[(1S)-2-[(4-carbamoylphenyl)methylamino]-2-oxo-1-(4-phenylmethoxyphenyl)ethyl]thiophene-2-carboxamide
Show/Hide
|
C28H25N3O4S
|
1
|
| 1 |
EC50 = 8400 nM
|
|
|
|
CP0547002
|
4-[2-[(2S)-2-(hexanoylamino)-2-(4-phenylmethoxyphenyl)acetyl]hydrazinyl]benzamide
Show/Hide
|
C28H32N4O4
|
1
|
| 1 |
EC50 = 8700 nM
|
|
|
|
CP0543000
|
N-(1-hydroxy-3H-2,1-benzoxaborol-6-yl)-4-phenylmethoxybenzamide
Show/Hide
|
C21H18BNO4
|
1
|
| 1 |
EC50 = 8800 nM
|
|
|
|
CP0544638
|
4-chloro-N-(1-hydroxy-3H-2,1-benzoxaborol-6-yl)benzenesulfonamide
Show/Hide
|
C13H11BClNO4S
|
1
|
| 1 |
EC50 = 9200 nM
|
|
|
|
CP0329893
|
N-[(1S)-2-[[4-(diaminomethylideneamino)phenyl]methylamino]-2-oxo-1-(4-phenylmethoxyphenyl)ethyl]-5-thiophen-2-ylthiophene-2-carboxamide;2,2,2-trifluoroacetic acid
Show/Hide
|
C34H30F3N5O5S2
|
1
|
| 1 |
EC50 = 9300 nM
|
|
|
|
CP0491964
|
4-[[[(2S)-2-(hexanoylamino)-2-[4-[[4-(trifluoromethyl)phenyl]methoxy]phenyl]acetyl]amino]methyl]benzamide
Show/Hide
|
C30H32F3N3O4
|
1
|
| 1 |
EC50 = 9800 nM
|
|
|
|
CP0310857
|
N-[(1R)-2-[[4-(diaminomethylideneamino)phenyl]methylamino]-2-oxo-1-(4-phenylmethoxyphenyl)ethyl]hexanamide;2,2,2-trifluoroacetic acid
Show/Hide
|
C31H36F3N5O5
|
1
|
| 1 |
EC50 = 9900 nM
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CP0531600
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N-[(1S)-2-[2-(4-hydroxyphenyl)ethylamino]-2-oxo-1-(4-phenylmethoxyphenyl)ethyl]hexanamide
Show/Hide
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C29H34N2O4
|
1
|
| 1 |
EC50 = 10000 nM
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CP0531601
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4-[[[(2S)-2-(heptylsulfonylamino)-2-(4-phenylmethoxyphenyl)acetyl]amino]methyl]benzamide
Show/Hide
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C30H37N3O5S
|
1
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| 1 |
EC50 = 11000 nM
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CP0419357
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4-[[[(2S)-2-(4-phenylmethoxyphenyl)-2-(3-phenylpropanoylamino)acetyl]amino]methyl]benzamide
Show/Hide
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C32H31N3O4
|
1
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| 1 |
EC50 = 12000 nM
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CP0568645
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[3-[(3-phenylmethoxybenzoyl)amino]phenyl]boronic acid
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C20H18BNO4
|
1
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| 1 |
EC50 = 12500 nM
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CP0323962
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N-[(1S)-2-[(6-aminopyridin-3-yl)methylamino]-2-oxo-1-(4-phenylmethoxyphenyl)ethyl]hexanamide;2,2,2-trifluoroacetic acid
Show/Hide
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C29H33F3N4O5
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1
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| 1 |
EC50 = 13000 nM
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CP0403579
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N-[(1S)-2-(6-aminohexylamino)-2-oxo-1-(4-phenylmethoxyphenyl)ethyl]hexanamide
Show/Hide
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C27H39N3O3
|
1
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| 1 |
EC50 = 13000 nM
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CP0491951
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N-[(1S)-2-oxo-1-(4-phenylmethoxyphenyl)-2-piperidin-1-ylethyl]hexanamide
Show/Hide
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C26H34N2O3
|
1
|
| 1 |
EC50 = 13000 nM
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|
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CP0571116
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3-benzamido-N-(1-hydroxy-3H-2,1-benzoxaborol-6-yl)benzamide
Show/Hide
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C21H17BN2O4
|
1
|
| 1 |
EC50 = 13100 nM
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|
|
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CP0491971
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4-[[[(2S)-2-(pentanoylamino)-2-(4-phenylmethoxyphenyl)acetyl]amino]methyl]benzamide
Show/Hide
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C28H31N3O4
|
1
|
| 1 |
EC50 = 14000 nM
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|
|
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CP0557758
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N-[(1S)-2-[(4-acetamidophenyl)methylamino]-2-oxo-1-(4-phenylmethoxyphenyl)ethyl]hexanamide
Show/Hide
|
C30H35N3O4
|
1
|
| 1 |
EC50 = 14000 nM
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|
|
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CP0544641
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[4-[[(3-phenylmethoxybenzoyl)amino]methyl]phenyl]boronic acid
Show/Hide
|
C21H20BNO4
|
1
|
| 1 |
EC50 = 14000 nM
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|
|
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CP0495121
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4-[(4-chlorophenyl)methoxy]-N-(1-hydroxy-3H-2,1-benzoxaborol-6-yl)benzamide
Show/Hide
|
C21H17BClNO4
|
1
|
| 1 |
EC50 = 14500 nM
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|
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CP0557776
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3-[[(2S)-2-[[4-(morpholine-4-carbonyl)benzoyl]amino]-2-(4-phenylmethoxyphenyl)acetyl]amino]benzamide
Show/Hide
|
C34H32N4O6
|
1
|
| 1 |
EC50 = 15000 nM
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|
|
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CP0100922
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N-[(1R)-2-[[4-(diaminomethylideneamino)phenyl]methylamino]-1-[4-[(3,4-dichlorophenyl)methoxy]phenyl]-2-oxoethyl]hexanamide;2,2,2-trifluoroacetic acid
Show/Hide
|
C31H34Cl2F3N5O5
|
1
|
| 1 |
EC50 = 16000 nM
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|
|
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CP0271592
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N-[(2S)-1-[[(2S)-6-amino-1-[[(1R)-2-amino-2-oxo-1-(4-phenylmethoxyphenyl)ethyl]amino]-1-oxohexan-2-yl]amino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]benzamide
Show/Hide
|
C34H44N8O5
|
1
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| 1 |
EC50 = 16000 nM
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|
|
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CP0575574
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N-(1-hydroxy-3H-2,1-benzoxaborol-6-yl)-4-morpholin-4-ylbenzamide
Show/Hide
|
C18H19BN2O4
|
1
|
| 1 |
EC50 = 17100 nM
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|
|
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CP0552401
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N-[(1S)-2-[4-(hydroxymethyl)anilino]-2-oxo-1-(4-phenylmethoxyphenyl)ethyl]hexanamide
Show/Hide
|
C28H32N2O4
|
1
|
| 1 |
EC50 = 18000 nM
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|
|
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CP0567961
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N-(1-hydroxy-3H-2,1-benzoxaborol-6-yl)hexanamide
Show/Hide
|
C13H18BNO3
|
1
|
| 1 |
EC50 = 19200 nM
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|
|
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CP0339644
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(2S)-N-[[4-(diaminomethylideneamino)phenyl]methyl]-2-(4-phenylmethoxyphenyl)-2-[[2-(4-phenylphenyl)acetyl]amino]acetamide;2,2,2-trifluoroacetic acid
Show/Hide
|
C39H36F3N5O5
|
1
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| 1 |
EC50 = 20000 nM
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|
|
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CP0419354
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1-[(2S)-2-(hexanoylamino)-2-(4-phenylmethoxyphenyl)acetyl]-N-phenylpiperidine-4-carboxamide
Show/Hide
|
C33H39N3O4
|
1
|
| 1 |
EC50 = 20000 nM
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|
|
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CP0259659
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3-(4-fluorophenyl)-N-(1-hydroxy-3H-2,1-benzoxaborol-6-yl)-5-methyl-1,2-oxazole-4-carboxamide
Show/Hide
|
C18H14BFN2O4
|
1
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| 1 |
EC50 = 21600 nM
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|
|
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CP0241169
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1-(1-hydroxy-3H-2,1-benzoxaborol-6-yl)-3-phenylurea
Show/Hide
|
C14H13BN2O3
|
1
|
| 1 |
EC50 = 22500 nM
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|
|
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CP0559451
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N-[(1S)-2-(3-carbamoylanilino)-2-oxo-1-(4-phenylmethoxyphenyl)ethyl]-3-(morpholine-4-carbonyl)benzamide
Show/Hide
|
C34H32N4O6
|
1
|
| 1 |
EC50 = 23000 nM
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|
|
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CP0423677
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N-[(1S)-2-[(4-methoxyphenyl)methylamino]-2-oxo-1-(4-phenylmethoxyphenyl)ethyl]hexanamide
Show/Hide
|
C29H34N2O4
|
1
|
| 1 |
EC50 = 28000 nM
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|
|
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CP0552990
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4-(aminomethyl)-N-[(1S)-2-[(4-carbamoylphenyl)methylamino]-2-oxo-1-(4-phenylmethoxyphenyl)ethyl]benzamide
Show/Hide
|
C31H30N4O4
|
1
|
| 1 |
EC50 = 29000 nM
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|
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CP0388406
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(2S)-N-[[4-(diaminomethylideneamino)phenyl]methyl]-2-[4-[(2,6-dichlorophenyl)methoxy]phenyl]-2-[[2-(4-phenylphenyl)acetyl]amino]acetamide;2,2,2-trifluoroacetic acid
Show/Hide
|
C39H34Cl2F3N5O5
|
1
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| 1 |
EC50 = 39000 nM
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|
|
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CP0576058
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4-chloro-N-(1-hydroxy-3H-2,1-benzoxaborol-6-yl)-N-methylbenzenesulfonamide
Show/Hide
|
C14H13BClNO4S
|
1
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| 1 |
EC50 > 50000 nM
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