Brief Information of the Cell Line and Protein
Cell Line ID: CL000656 , NCTC 2544
 Cell Line Info 
Synonyms
NCTC-2544
NCTC2544
NCTC strain 2544
Category Cancer cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0461
Protein ID: PT04124 , Proteinase-activated receptor 2
 Protein Info 
Gene Name F2RL1
Organism Homo sapiens, Human
Protein Classification Membrane receptor
Uniprot ID P55085
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000656
 Cell Line Info 
 Protein ID: PT04124
 Protein Info 
 
Compound ID Compound Name Compound Formula
CP0415492
 Compound Info 
N-[(2S)-1-[[(2S,3S)-1-[[2-[[(2S)-5-(diaminomethylideneamino)-1-[[(2S)-1-[[(2S)-1,5-diamino-1-oxopentan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-1-oxopentan-2-yl]amino]-2-oxoethyl]amino]-3-methyl-1-oxopentan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]furan-2-carboxamide
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C36H63N11O8
  1
1
IC50 = 100 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0389117
 Compound Info 
(2S)-6-amino-N-[(2S)-1-(benzhydrylamino)-1-oxo-3-phenylpropan-2-yl]-2-[[2-[[1-[(2,6-dichlorophenyl)methyl]-3-(pyrrolidin-1-ylmethyl)indol-5-yl]carbamoylamino]acetyl]amino]hexanamide
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C51H56Cl2N8O4
  2
1
IC50 = 1100 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
2
Ki = 600 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0407850
 Compound Info 
(2S)-6-amino-N-[(2R)-1-(benzhydrylamino)-1-oxo-3-phenylpropan-2-yl]-2-[[2-[[1-[(2,6-dichlorophenyl)methyl]-3-(pyrrolidin-1-ylmethyl)indol-5-yl]carbamoylamino]acetyl]amino]hexanamide
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C51H56Cl2N8O4
  1
1
Ki = 627 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0417382
 Compound Info 
(2S)-4-amino-N-[(2R)-1-anilino-1-oxo-3-phenylpropan-2-yl]-2-[[2-[[1-[(2,6-dichlorophenyl)methyl]-3-(pyrrolidin-1-ylmethyl)indol-5-yl]carbamoylamino]acetyl]amino]butanamide
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C42H46Cl2N8O4
  1
1
Ki = 1940 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS