Brief Information of the Cell Line and Protein
Cell Line ID: CL000789 , HG5LN
Category Cancer cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0030
Protein ID: PT02658 , Nuclear receptor ROR-alpha
Gene Name RORA
Organism Homo sapiens, Human
Protein Classification Transcription factor
Uniprot ID P35398
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000789  Protein ID: PT02658
 
Compound ID Compound Name Compound Formula
CP0447696
4-[3-(2-chloro-6-methylphenoxy)-5-(dimethylcarbamoyl)indazol-1-yl]benzoic acid
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C24H20ClN3O4
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0452052
4-[3-[2-chloro-6-(trifluoromethyl)phenoxy]-5-(dimethylcarbamoyl)indazol-1-yl]benzoic acid
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C24H17ClF3N3O4
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0405429
N-(4-ethylphenyl)-N-(2-methylpropyl)-3-(methylsulfonimidoyl)-4-(oxan-4-ylmethoxy)benzenesulfonamide
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C25H36N2O5S2
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0440833
BDBM50461078
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C25H36N2O5S2
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS