Brief Information of the Cell Line and Protein
Cell Line ID: CL000482 , NCI-H929
Synonyms
NCI H929
NCIH929
H929
H-929
Category Cancer cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_1600
Protein ID: PT02583 , Proteasome subunit beta type-1
Gene Name PSMB1
Organism Homo sapiens, Human
Protein Classification Enzyme
Uniprot ID P20618
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000482  Protein ID: PT02583
 
Compound ID Compound Name Compound Formula
CP0261361
(2S)-N-[(2S)-1-[[(E,2S)-1-[4-(aminomethyl)phenyl]-4-methylsulfonylbut-3-en-2-yl]amino]-4-methyl-1-oxopentan-2-yl]-2-[[(2S)-2-azido-3-phenylpropanoyl]amino]-4-methylpentanamide
   Show/Hide
C33H47N7O5S
 1
1
IC50 = 2200 nM
   TI
   LI
   LO
   TS
CP0065810
(2S)-2-[[(2S)-3-[4-(aminomethyl)phenyl]-2-[[(2S)-2-azido-3-phenylpropanoyl]amino]propanoyl]amino]-N-[(E,2S)-1-[4-(aminomethyl)phenyl]-4-methylsulfonylbut-3-en-2-yl]-4-methylpentanamide
   Show/Hide
C37H48N8O5S
 1
1
IC50 = 17400 nM
   TI
   LI
   LO
   TS
CP0128289
(2S)-N-[(E,2S)-1-[4-(aminomethyl)phenyl]-4-methylsulfonylbut-3-en-2-yl]-2-[[(2S)-3-(4-aminophenyl)-2-[[(2S)-2-azido-3-phenylpropanoyl]amino]propanoyl]amino]-4-methylpentanamide
   Show/Hide
C36H46N8O5S
 1
1
IC50 = 22000 nM
   TI
   LI
   LO
   TS
CP0145054
(2S)-N-[(E,2S)-1-[4-(aminomethyl)phenyl]-4-methylsulfonylbut-3-en-2-yl]-2-[[(2S)-2-[[(2S)-2-azido-3-phenylpropanoyl]amino]-3-pyridin-4-ylpropanoyl]amino]-4-methylpentanamide
   Show/Hide
C35H44N8O5S
 1
1
IC50 > 30000 nM
   TI
   LI
   LO
   TS
CP0427458
N-[(2S)-1-[[(2S)-1-[[(2S)-5-(diaminomethylideneamino)-1-[(2R)-2-methyloxiran-2-yl]-1-oxopentan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]-3-hydroxy-2-methylbenzamide
   Show/Hide
C25H38N6O7
 1
1
IC50 > 30000 nM
   TI
   LI
   LO
   TS
CP0427459
N-[(2S)-1-[[(2S)-1-[[(E,2S)-1-[4-(aminomethyl)phenyl]-4-methylsulfonylbut-3-en-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]-3-hydroxy-2-methylbenzamide
   Show/Hide
C28H38N4O7S
 1
1
IC50 > 30000 nM
   TI
   LI
   LO
   TS