Compound ID |
Compound Name |
Compound Formula |
CP0440068
|
2-[4-[4-[5-[(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)amino]pyridin-2-yl]phenyl]cyclohexyl]acetic acid
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|
C26H29N3O4
|
1
|
1 |
EC50 = 8 nM
|
|
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CP0455441
|
2-[4-[4-[5-[(5-cyclobutyl-1,3,4-thiadiazol-2-yl)amino]pyridin-2-yl]phenyl]cyclohexyl]acetic acid
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|
C25H28N4O2S
|
1
|
1 |
EC50 = 8 nM
|
|
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CP0391157
|
2-[4-[4-[4-[(5-cyclobutyl-1,3,4-oxadiazol-2-yl)amino]phenyl]phenyl]-2-oxabicyclo[2.2.2]octan-1-yl]acetic acid
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|
C27H29N3O4
|
1
|
1 |
EC50 = 12 nM
|
|
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CP0462265
|
2-[4-[4-[5-[(5-cyclobutyl-1,3,4-oxadiazol-2-yl)amino]pyridin-2-yl]phenyl]cyclohexyl]acetic acid
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|
C25H28N4O3
|
1
|
1 |
EC50 = 12 nM
|
|
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CP0391156
|
2-[4-[4-[5-[(5-ethyl-1,3,4-oxadiazol-2-yl)amino]pyridin-2-yl]phenyl]cyclohexyl]acetic acid
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|
C23H26N4O3
|
1
|
1 |
EC50 = 27 nM
|
|
|
CP0479246
|
2-[4-[4-[4-[(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)amino]phenyl]phenyl]-2-oxabicyclo[2.2.2]octan-1-yl]acetic acid
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|
C28H30N2O5
|
1
|
1 |
EC50 = 56 nM
|
|
|
CP0455442
|
LCQ-908-NXA
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|
C25H24F3N3O2
|
1
|
1 |
EC50 = 71 nM
|
|
|
CP0411042
|
2-[4-[4-[5-[(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)amino]pyridin-2-yl]phenyl]-2-oxabicyclo[2.2.2]octan-1-yl]acetic acid
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|
C27H29N3O5
|
1
|
1 |
EC50 = 98 nM
|
|
|
CP0462264
|
2-[4-[4-[5-[(5-methyl-1,3,4-oxadiazol-2-yl)amino]pyridin-2-yl]phenyl]cyclohexyl]acetic acid
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|
C22H24N4O3
|
1
|
1 |
EC50 = 206 nM
|
|
|
CP0459254
|
2-[4-[4-[5-[(5-cyclobutyl-1,3,4-oxadiazol-2-yl)amino]pyridin-2-yl]phenyl]-2-oxabicyclo[2.2.2]octan-1-yl]acetic acid
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|
C26H28N4O4
|
1
|
1 |
EC50 = 413 nM
|
|
|
CP0533414
|
2-[1-[4-[5-[(5-propan-2-yl-1,3,4-oxadiazol-2-yl)amino]pyridin-2-yl]phenyl]piperidin-4-yl]acetic acid
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|
C23H27N5O3
|
1
|
1 |
EC50 = 2300 nM
|
|
|
CP0485296
|
N-[2-[[1-phenyl-3-(trifluoromethyl)pyrazole-4-carbonyl]amino]ethyl]-6-(2,2,2-trifluoroethoxy)pyridine-3-carboxamide
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|
C21H17F6N5O3
|
1
|
1 |
IC50 = 44 nM
|
|
|
CP0383423
|
N-[2-[(4-ethoxybenzoyl)amino]ethyl]-1-phenyl-3-(trifluoromethyl)pyrazole-4-carboxamide
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|
C22H21F3N4O3
|
1
|
1 |
IC50 = 77 nM
|
|
|
CP0519371
|
6-Ethoxy-N-[2-({[1-phenyl-3-(trifluoromethyl)-1Hpyrazol-4-yl]carbonyl}amino)ethyl]pyridine-3-carboxamide
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|
C21H20F3N5O3
|
1
|
1 |
IC50 = 87 nM
|
|
|
CP0462722
|
N-[2-[(4-ethoxybenzoyl)amino]ethyl]-1-pyridin-2-yl-3-(trifluoromethyl)pyrazole-4-carboxamide
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|
C21H20F3N5O3
|
1
|
1 |
IC50 = 91 nM
|
|
|
CP0453586
|
N-(3,4-dimethylphenyl)-2-(4-methoxy-2,6-dimethylphenyl)-3H-benzimidazole-5-carboxamide
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|
C25H25N3O2
|
1
|
1 |
IC50 = 120 nM
|
|
|
CP0244107
|
3-[4-[6-[5-(4-methoxyphenyl)-1,3,4-oxadiazol-2-yl]-1H-benzimidazol-2-yl]-3,5-dimethylphenyl]-2,2-dimethylpropanoic acid
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|
C29H28N4O4
|
1
|
1 |
IC50 = 151 nM
|
|
|
CP0513574
|
3-[4-[6-[5-(4-methoxyphenyl)-1,3,4-oxadiazol-2-yl]-1H-benzimidazol-2-yl]-3,5-dimethylphenyl]propanoic acid
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|
C27H24N4O4
|
1
|
1 |
IC50 = 181 nM
|
|
|
CP0485297
|
N-[2-[(4-ethoxybenzoyl)amino]ethyl]-3-methyl-1-phenylpyrazole-4-carboxamide
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|
C22H24N4O3
|
1
|
1 |
IC50 = 260 nM
|
|
|
CP0401552
|
6-Chloro-N-[2-({[1-phenyl-3-(trifluoromethyl)-1Hpyrazol-4-yl]carbonyl}amino)ethyl]pyridine-3-carboxamide
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|
C19H15ClF3N5O2
|
1
|
1 |
IC50 = 370 nM
|
|
|
CP0485295
|
1-(4-Ethoxyphenyl)-N-(2-{[(4-ethoxyphenyl)carbonyl]amino}ethyl)-3-(trifluoromethyl)-1Hpyrazole-4-carboxamide
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|
C24H25F3N4O4
|
1
|
1 |
IC50 = 380 nM
|
|
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CP0443584
|
3-[4-[6-[(4-tert-butylphenyl)carbamoyl]-1H-benzimidazol-2-yl]-3,5-dimethylphenyl]propanoic acid
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|
C29H31N3O3
|
1
|
1 |
IC50 = 390 nM
|
|
|
CP0910947
|
1-Phenyl-N-[2-({[4-(1H-pyrazol-1-yl)phenyl]carbonyl}amino)ethyl]-3-(trifluoromethyl)-1Hpyrazole-4-carboxamide hydrochloride
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|
C23H20ClF3N6O2
|
1
|
1 |
IC50 = 400 nM
|
|
|
CP0502365
|
1-(3-Ethoxyphenyl)-N-(2-{[(4-ethoxyphenyl)carbonyl]amino}ethyl)-3-(trifluoromethyl)-1Hpyrazole-4-carboxamide
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|
C24H25F3N4O4
|
1
|
1 |
IC50 = 600 nM
|
|
|
CP0374310
|
N-[2-[(4-ethoxybenzoyl)amino]ethyl]-1-(2-hydroxyphenyl)-3-(trifluoromethyl)pyrazole-4-carboxamide
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|
C22H21F3N4O4
|
1
|
1 |
IC50 = 610 nM
|
|
|
CP0510120
|
1-Cyclohexyl-N-(2-{[(4-ethoxyphenyl)carbonyl]amino}-ethyl)-3-(trifluoromethyl)-1H-pyrazole-4-carboxamide
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|
C22H27F3N4O3
|
1
|
1 |
IC50 = 650 nM
|
|
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CP0497302
|
1-Benzyl-N-(2-{[(4-ethoxyphenyl)carbonyl]amino}-ethyl)-3-(trifluoromethyl)-1H-pyrazole-4-carboxamide
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|
C23H23F3N4O3
|
1
|
1 |
IC50 = 770 nM
|
|
|
CP0513575
|
3-[3,5-dimethyl-4-[6-(quinolin-2-ylcarbamoyl)-1H-benzimidazol-2-yl]phenyl]propanoic acid
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|
C28H24N4O3
|
1
|
1 |
IC50 = 913 nM
|
|
|
CP0547900
|
3-[3,5-dimethyl-4-[6-(quinolin-2-ylcarbamoyl)-1H-benzimidazol-2-yl]phenyl]-2,2-dimethylpropanoic acid
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|
C30H28N4O3
|
1
|
1 |
IC50 = 954 nM
|
|
|
CP0383424
|
N-[2-[(4-ethoxybenzoyl)amino]ethyl]-4-methyl-1-phenylpyrazole-3-carboxamide
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|
C22H24N4O3
|
1
|
1 |
IC50 = 1200 nM
|
|
|
CP0383469
|
5-Chloro-N-[2-({[1-phenyl-3-(trifluoromethyl)-1Hpyrazol-4-yl]carbonyl}amino)ethyl]pyridine-2-carboxamide
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|
C19H15ClF3N5O2
|
1
|
1 |
IC50 = 1200 nM
|
|
|
CP0374309
|
1-(4-Chlorophenyl)-N-(2-{[(4-ethoxyphenyl)carbonyl]amino}ethyl)-3-(trifluoromethyl)-1Hpyrazole-4-carboxamide
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|
C22H20ClF3N4O3
|
1
|
1 |
IC50 = 1500 nM
|
|
|
CP0461832
|
2-[4-[6-[(3,4-dimethylphenyl)carbamoyl]-1H-benzimidazol-2-yl]-3,5-dimethylanilino]acetic acid
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|
C26H26N4O3
|
1
|
1 |
IC50 = 2000 nM
|
|
|
CP0473494
|
N-[2-[(4-ethoxybenzoyl)amino]ethyl]-1-pyridin-3-yl-3-(trifluoromethyl)pyrazole-4-carboxamide
Show/Hide
|
C21H20F3N5O3
|
1
|
1 |
IC50 = 3400 nM
|
|
|
CP0374311
|
N-[2-[(3-ethoxybenzoyl)amino]ethyl]-1-phenyl-3-(trifluoromethyl)pyrazole-4-carboxamide
Show/Hide
|
C22H21F3N4O3
|
1
|
1 |
IC50 = 5100 nM
|
|
|
CP0461831
|
3-[4-[6-[(3,4-dimethylphenyl)carbamoyl]-1H-benzimidazol-2-yl]-3,5-dimethylphenyl]propanoic acid
Show/Hide
|
C27H27N3O3
|
1
|
1 |
IC50 = 6500 nM
|
|
|
CP0401551
|
N-[2-[(4-ethoxybenzoyl)amino]ethyl]-1-pyridin-4-yl-3-(trifluoromethyl)pyrazole-4-carboxamide
Show/Hide
|
C21H20F3N5O3
|
1
|
1 |
IC50 > 10000 nM
|
|
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CP0489844
|
2-[4-[6-[(3,4-dimethylphenyl)carbamoyl]-1H-benzimidazol-2-yl]-3,5-dimethylphenoxy]acetic acid
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|
C26H25N3O4
|
1
|
1 |
IC50 > 10000 nM
|
|
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