Compound ID |
Compound Name |
Compound Formula |
CP0498361
|
naphthyridinone analog., 27
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|
C8H4ClFN2O2
|
1
|
1 |
IC50 = 3 nM
|
|
|
CP0506125
|
3-hydroxyquinolin-2(1H)-one, 3
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|
C9H6FNO2
|
1
|
1 |
IC50 = 3 nM
|
|
|
CP0044107
|
3-hydroxyquinolin-2(1H)-one, 10
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|
C9H6ClNO2
|
1
|
1 |
IC50 = 4 nM
|
|
|
CP0176014
|
3-hydroxyquinolin-2(1H)-one, 2
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|
C9H7NO2
|
1
|
1 |
IC50 = 4 nM
|
|
|
CP0203193
|
3-hydroxyquinolin-2(1H)-one, 26
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|
C9H5ClFNO2
|
1
|
1 |
IC50 = 5 nM
|
|
|
CP0281664
|
naphthyridinone analog.,18
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|
C8H6N2O2
|
1
|
1 |
IC50 = 8 nM
|
|
|
CP0281665
|
3-hydroxyquinolin-2(1H)-one, 6
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|
C9H6FNO2
|
1
|
1 |
IC50 = 8 nM
|
|
|
CP0296216
|
3-hydroxyquinolin-2(1H)-one, 15
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|
C11H11NO2
|
1
|
1 |
IC50 = 8 nM
|
|
|
CP0044110
|
4H-furo[3,2-b]pyrrole-5-carboxylic acid
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|
C7H5NO3
|
1
|
1 |
IC50 = 9 nM
|
|
|
CP0296215
|
3-hydroxyquinolin-2(1H)-one, 5
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|
C9H6FNO2
|
1
|
1 |
IC50 = 9 nM
|
|
|
CP0371190
|
3-hydroxyquinolin-2(1H)-one, 4
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|
C9H6FNO2
|
1
|
1 |
IC50 = 10 nM
|
|
|
CP0418011
|
3-hydroxyquinolin-2(1H)-one, 14
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|
C10H9NO2
|
1
|
1 |
IC50 = 16 nM
|
|
|
CP0498363
|
naphthyridinone analog.,19
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|
C8H6N2O2
|
1
|
1 |
IC50 = 32 nM
|
|
|
CP0496669
|
3-hydroxyquinolin-2(1H)-one, 7
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|
C9H6ClNO2
|
1
|
1 |
IC50 = 33 nM
|
|
|
CP0498360
|
3-hydroxyquinolin-2(1H)-one, 11
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|
C10H9NO2
|
1
|
1 |
IC50 = 38 nM
|
|
|
CP0491077
|
3-hydroxyquinolin-2(1H)-one, 8
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|
C9H6ClNO2
|
1
|
1 |
IC50 = 100 nM
|
|
|
CP0418010
|
naphthyridinone analog.,21
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|
C8H6N2O2
|
1
|
1 |
IC50 = 128 nM
|
|
|
CP0498932
|
3-hydroxyquinolin-2(1H)-one, 9
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|
C9H6ClNO2
|
1
|
1 |
IC50 = 155 nM
|
|
|
CP0418012
|
3-hydroxyquinolin-2(1H)-one, 12
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|
C10H9NO2
|
1
|
1 |
IC50 = 197 nM
|
|
|
CP0496668
|
naphthyridinone analog.,20
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|
C8H6N2O2
|
1
|
1 |
IC50 = 784 nM
|
|
|
CP0496667
|
3-hydroxyquinolin-2(1H)-one, 13
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|
C10H9NO2
|
1
|
1 |
IC50 = 2750 nM
|
|
|
CP0514636
|
3-hydroxyquinolin-2(1H)-one, 25
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|
C10H9NO2
|
1
|
1 |
IC50 = 3260 nM
|
|
|
CP0453822
|
3-hydroxyquinolin-2(1H)-one, 17
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|
C11H11NO2
|
1
|
1 |
IC50 = 14400 nM
|
|
|
CP0471935
|
3-hydroxyquinolin-2(1H)-one, 23
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|
C10H9NO2
|
1
|
1 |
IC50 = 17300 nM
|
|
|
CP0400860
|
3-hydroxyquinolin-2(1H)-one, 16
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|
C11H11NO2
|
1
|
1 |
IC50 = 22600 nM
|
|
|
CP0418009
|
3-methoxyquinolin-2(1H)-one, 24
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|
C10H9NO2
|
1
|
1 |
IC50 > 26200 nM
|
|
|
CP0505016
|
pyridopyrazinone, 22
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|
C7H5N3O2
|
1
|
1 |
IC50 > 50000 nM
|
|
|