Brief Information of the Cell Line and Protein
Cell Line ID: CL000314 , HEK293T/17
Synonyms
HEK-293T/17
HEK 293T/17
293T/17
Category Transformed cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_1926
Protein ID: PT02200 , Glutamate receptor ionotropic, kainate 1
Gene Name GRIK1
Organism Rattus norvegicus, Rat
Protein Classification Ion channel
Uniprot ID P22756
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000314  Protein ID: PT02200
 
Compound ID Compound Name Compound Formula
CP0417183
(2S,4R)-4-(2-carboxyphenoxy)pyrrolidine-2-carboxylic acid;hydrochloride
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C12H14ClNO5
 1
1
Ki = 2270 nM
   TI
   LI
   LO
   TS
CP0398995
(2S,4S)-4-(4-carboxyphenoxy)pyrrolidine-2-carboxylic acid;hydrochloride
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C12H14ClNO5
 1
1
Ki > 100000 nM
   TI
   LI
   LO
   TS
CP0398997
(2S,4R)-4-(2-carboxynaphthalen-1-yl)oxypyrrolidine-2-carboxylic acid
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C16H15NO5
 1
1
Ki > 100000 nM
   TI
   LI
   LO
   TS
CP0409584
(2S,4R)-4-[3-(carboxymethyl)phenoxy]pyrrolidine-2-carboxylic acid
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C13H15NO5
 1
1
Ki > 100000 nM
   TI
   LI
   LO
   TS
CP0411195
(2S,4R)-4-[(3-carboxyphenyl)methyl]pyrrolidine-2-carboxylic acid;hydrochloride
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C13H16ClNO4
 1
1
Ki > 100000 nM
   TI
   LI
   LO
   TS
CP0411198
(2S,4S)-4-(3-carboxyphenyl)sulfanylpyrrolidine-2-carboxylic acid
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C12H13NO4S
 1
1
Ki > 100000 nM
   TI
   LI
   LO
   TS
CP0411212
(2S,4R)-4-(4-carboxyphenoxy)pyrrolidine-2-carboxylic acid;hydrochloride
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C12H14ClNO5
 1
1
Ki > 100000 nM
   TI
   LI
   LO
   TS
CP0417180
(2S,4S)-4-(3-carboxyphenoxy)pyrrolidine-2-carboxylic acid;hydrochloride
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C12H14ClNO5
 1
1
Ki > 100000 nM
   TI
   LI
   LO
   TS
CP0447492
(2S,4R)-4-(3-carboxyphenyl)sulfanylpyrrolidine-2-carboxylic acid
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C12H13NO4S
 1
1
Ki > 100000 nM
   TI
   LI
   LO
   TS
CP0479812
4-[(3R,5S)-5-carboxypyrrolidin-3-yl]oxybenzene-1,3-dicarboxylic acid
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C13H13NO7
 1
1
Ki = 100000 nM
   TI
   LI
   LO
   TS
CP0481247
(2S,4S)-4-(2-carboxyphenyl)sulfanylpyrrolidine-2-carboxylic acid
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C12H13NO4S
 1
1
Ki > 100000 nM
   TI
   LI
   LO
   TS
CP0482120
(2S,4S)-4-(2-carboxyphenoxy)pyrrolidine-2-carboxylic acid;hydrochloride
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C12H14ClNO5
 1
1
Ki > 100000 nM
   TI
   LI
   LO
   TS