Brief Information of the Cell Line and Protein
Cell Line ID: CL000017 , HeLa
Synonyms
HELA
Hela
He La
He-La
HeLa-CCL2
Henrietta Lacks cells
Helacyton gartleri
Category Cancer cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0030
Protein ID: PT02059 , C-X-C chemokine receptor type 4
Gene Name CXCR4
Organism Homo sapiens, Human
Protein Classification Membrane receptor
Uniprot ID P61073
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000017  Protein ID: PT02059
 
Compound ID Compound Name Compound Formula
CP0559907
US9314468, Table 8, Compound 2
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C28H31N5
 1
1
IC50 = 5.5 nM
   TI
   LI
   LO
   TS
CP0567742
US9314468, Table 8, Compound 3
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C31H38N6O2
 1
1
IC50 = 5.6 nM
   TI
   LI
   LO
   TS
CP0529254
US9314468, Table 8, Compound 1
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C31H41N7
 1
1
IC50 = 5.7 nM
   TI
   LI
   LO
   TS
CP0563329
US9314468, Table 8, Compound 4
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C27H32N6O
 1
1
IC50 = 5.8 nM
   TI
   LI
   LO
   TS
CP0555371
US9314468, Table 8, Compound 5
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C28H36N6
 1
1
IC50 = 7.3 nM
   TI
   LI
   LO
   TS
CP0557222
US9314468, Table 8, Compound 6
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C31H40N6O
 1
1
IC50 = 7.7 nM
   TI
   LI
   LO
   TS
CP0512338
US9314468, Table 8, Compound 7
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C27H30IN5O2
 1
1
IC50 = 8.1 nM
   TI
   LI
   LO
   TS
CP0564063
US9314468, Table 8, Compound 8
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C32H43N7
 1
1
IC50 = 8.3 nM
   TI
   LI
   LO
   TS
CP0499712
US9314468, Table 8, Compound 9
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C34H45N7O
 1
1
IC50 = 9.3 nM
   TI
   LI
   LO
   TS
CP0557223
US9314468, Table 8, Compound 10
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C33H42N6O2
 1
1
IC50 = 9.9 nM
   TI
   LI
   LO
   TS
CP0557224
US9314468, Table 8, Compound 11
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C32H41N7O
 1
1
IC50 = 11 nM
   TI
   LI
   LO
   TS
CP0499710
US9314468, Table 8, Compound 12
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C32H41N7O
 1
1
IC50 = 12 nM
   TI
   LI
   LO
   TS
CP0499713
US9314468, Table 8, Compound 14
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C30H38N6O
 1
1
IC50 = 12 nM
   TI
   LI
   LO
   TS
CP0523363
US9314468, Table 8, Compound 13
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C32H40N6O2
 1
1
IC50 = 12 nM
   TI
   LI
   LO
   TS
CP0537002
US9314468, Table 8, Compound 15
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C34H43N7O2
 1
1
IC50 = 15 nM
   TI
   LI
   LO
   TS
CP0545939
US9314468, Table 8, Compound 16
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C30H36N6O2
 1
1
IC50 = 26 nM
   TI
   LI
   LO
   TS