| Compound ID |
Compound Name |
Compound Formula |
|
CP0381075
|
2-((R)-3-(2-Bromo-1H-indol-3-yl)-2-{2-cyclopropyl-2-[((2S,6R)-2,6-dimethyl-piperidine-1-carbonyl)-amino]-acetylamino}-propionylamino)-hexanoic acid
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|
C30H42BrN5O5
|
1
|
| 1 |
IC50 = 1.1 nM
|
|
|
|
CP0875845
|
Sodium salt 2-[2-{2-[(2,6-dimethyl-piperidine-1-carbonyl)-amino]-4,4-dimethyl-pentanoylamino}-3-(1-methoxymethyl-1H-indol-3-yl)-propionylamino]-hexanoate
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|
C34H52N5NaO6
|
1
|
| 1 |
IC50 = 1.2 nM
|
|
|
|
CP0423125
|
2-((R)-3-(2-Bromo-1H-indol-3-yl)-2-{2-[((2S,6R)-2,6-dimethyl-piperidine-1-carbonyl)-amino]-4-methyl-pentanoylamino}-propionylamino)-3-ethylsulfanyl-propionic acid
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|
C30H44BrN5O5S
|
1
|
| 1 |
IC50 = 3.6 nM
|
|
|
|
CP0374683
|
2-[(R)-2-{2-Cyclopropyl-2-[((2R,6S)-2,6-dimethyl-piperidine-1-carbonyl)-amino]-acetylamino}-3-(2-methyl-1H-indol-3-yl)-propionylamino]-4-methylsulfanyl-butyric acid
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|
C30H43N5O5S
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0523274
|
2-((R)-3-(2-Cyano-1H-indol-3-yl)-2-{2-[((2S,6R)-2,6-dimethyl-piperidine-1-carbonyl)-amino]-3-methyl-butyrylamino}-propionylamino)-hexanoic acid
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|
C31H44N6O5
|
1
|
| 1 |
IC50 = 5 nM
|
|
|
|
CP0395445
|
2-[(3R,6S,9R,12S,15S)-6-[(2-bromo-1H-indol-3-yl)methyl]-12-cyclopentyl-9-cyclopropyl-2,5,8,11,14-pentaoxo-1,4,7,10,13-pentazabicyclo[13.3.0]octadecan-3-yl]acetic acid
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|
C32H39BrN6O7
|
1
|
| 1 |
IC50 = 29 nM
|
|
|
|
CP0448751
|
2-[(3R,6S,9R,12R,15S)-6-[(2-cyano-1H-indol-3-yl)methyl]-12-(2-methylsulfanylpropan-2-yl)-2,5,8,11,14-pentaoxo-9-propan-2-yl-1,4,7,10,13-pentazabicyclo[13.3.0]octadecan-3-yl]acetic acid
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|
C32H41N7O7S
|
1
|
| 1 |
IC50 = 29 nM
|
|
|
|
CP0376484
|
2-[(3R,6S,9R,12S,15S)-12-cyclopentyl-9-cyclopropyl-6-[(2-methyl-1H-indol-3-yl)methyl]-2,5,8,11,14-pentaoxo-1,4,7,10,13-pentazabicyclo[13.3.0]octadecan-3-yl]acetic acid
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|
C33H42N6O7
|
1
|
| 1 |
IC50 = 130 nM
|
|
|
