| Compound ID |
Compound Name |
Compound Formula |
|
CP0562941
|
3-(cyclopropylmethyl)-7-[3-(4-fluorophenyl)cyclobutyl]oxy-8-(trifluoromethyl)-[1,2,4]triazolo[4,3-a]pyridine
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|
C21H19F4N3O
|
1
|
| 1 |
EC50 = 0.4 nM
|
|
|
|
CP0566106
|
3-(cyclopropylmethyl)-7-(4-phenylcyclohexyl)oxy-8-(trifluoromethyl)-[1,2,4]triazolo[4,3-a]pyridine
Show/Hide
|
C23H24F3N3O
|
1
|
| 1 |
EC50 = 0.4 nM
|
|
|
|
CP0512450
|
3-(cyclopropylmethyl)-7-(3-phenylcyclobutyl)oxy-8-(trifluoromethyl)-[1,2,4]triazolo[4,3-a]pyridine
Show/Hide
|
C21H20F3N3O
|
1
|
| 1 |
EC50 = 0.5 nM
|
|
|
|
CP0445301
|
7-[[2-(4-chlorophenyl)cyclopropyl]methoxy]-3-(cyclopropylmethyl)-8-(trifluoromethyl)-[1,2,4]triazolo[4,3-a]pyridine
Show/Hide
|
C21H19ClF3N3O
|
1
|
| 1 |
EC50 = 1.3 nM
|
|
|
|
CP0326353
|
7-[[(1S,2S)-2-(4-chlorophenyl)cyclopropyl]methoxy]-3-(cyclopropylmethyl)-8-(trifluoromethyl)-[1,2,4]triazolo[4,3-a]pyridine
Show/Hide
|
C21H19ClF3N3O
|
3
|
| 1 |
EC50 = 1.4 nM
|
|
|
| 2 |
EC50 = 530 nM
|
|
|
| 3 |
Ki = 1 nM
|
|
|
|
CP0388460
|
3-(cyclopropylmethyl)-7-[[2-(4-fluorophenyl)cyclopropyl]methoxy]-8-(trifluoromethyl)-[1,2,4]triazolo[4,3-a]pyridine
Show/Hide
|
C21H19F4N3O
|
1
|
| 1 |
EC50 = 1.7 nM
|
|
|
|
CP0388459
|
3-(cyclopropylmethyl)-7-[(1-phenylcyclohexyl)methoxy]-8-(trifluoromethyl)-[1,2,4]triazolo[4,3-a]pyridine
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|
C24H26F3N3O
|
1
|
| 1 |
EC50 = 1.8 nM
|
|
|
|
CP0035205
|
2-[[(3R,4R)-4-[2-fluoro-4-(trifluoromethyl)phenyl]-3-methylpiperidin-1-yl]methyl]-1-methylimidazo[4,5-b]pyridine
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|
C21H22F4N4
|
1
|
| 1 |
EC50 = 3 nM
|
|
|
|
CP0454448
|
(1S,2S,4S,5R,6S)-2-amino-4-[(3-hydroxybenzoyl)amino]bicyclo[3.1.0]hexane-2,6-dicarboxylic acid
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|
C15H16N2O6
|
2
|
| 1 |
EC50 = 3.77 nM
|
|
|
| 2 |
Ki = 31.5 nM
|
|
|
|
CP0473376
|
7-[[(1R,2R)-2-(4-chlorophenyl)cyclopropyl]methoxy]-3-(cyclopropylmethyl)-8-(trifluoromethyl)-[1,2,4]triazolo[4,3-a]pyridine
Show/Hide
|
C21H19ClF3N3O
|
1
|
| 1 |
EC50 = 4 nM
|
|
|
|
CP0070606
|
(5R)-3-(4-(1-cyclohexylethoxy)benzyl)-5-methyloxazolidin-2-one
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|
C19H27NO3
|
1
|
| 1 |
EC50 = 5 nM
|
|
|
|
CP0512453
|
7-[2-(4-chlorophenyl)-2-methylpropoxy]-3-(cyclopropylmethyl)-8-(trifluoromethyl)-[1,2,4]triazolo[4,3-a]pyridine
Show/Hide
|
C21H21ClF3N3O
|
1
|
| 1 |
EC50 = 5.5 nM
|
|
|
|
CP0563807
|
3-(cyclopropylmethyl)-7-(2,2-difluoro-2-phenylethoxy)-8-(trifluoromethyl)-[1,2,4]triazolo[4,3-a]pyridine
Show/Hide
|
C19H16F5N3O
|
1
|
| 1 |
EC50 = 6.1 nM
|
|
|
|
CP0396672
|
(1S,2S,4S,5R,6S)-2-amino-4-[(4-hydroxybenzoyl)amino]bicyclo[3.1.0]hexane-2,6-dicarboxylic acid
Show/Hide
|
C15H16N2O6
|
2
|
| 1 |
EC50 = 6.32 nM
|
|
|
| 2 |
Ki = 54.7 nM
|
|
|
|
CP0455190
|
8-chloro-3-(cyclopropylmethyl)-7-[(4-phenylphenyl)methoxy]-[1,2,4]triazolo[4,3-a]pyridine
Show/Hide
|
C23H20ClN3O
|
1
|
| 1 |
EC50 = 6.8 nM
|
|
|
|
CP0396670
|
(1S,2S,4S,5R,6S)-2-amino-4-[(4-chlorobenzoyl)amino]bicyclo[3.1.0]hexane-2,6-dicarboxylic acid
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|
C15H15ClN2O5
|
2
|
| 1 |
EC50 = 6.97 nM
|
|
|
| 2 |
Ki = 137 nM
|
|
|
|
CP0076675
|
(1S,2S,5R,6S)-2-Amino-bicyclo[3.1.0]hexane-2,6-dicarboxylic acid
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|
C8H11NO4
|
2
|
| 1 |
EC50 = 7 nM
|
|
|
| 2 |
Ki = 71.7 nM
|
|
|
|
CP0389521
|
(1S,2S,4S,5R,6S)-2-amino-4-[(2-hydroxybenzoyl)amino]bicyclo[3.1.0]hexane-2,6-dicarboxylic acid
Show/Hide
|
C15H16N2O6
|
2
|
| 1 |
EC50 = 7.44 nM
|
|
|
| 2 |
Ki = 58.2 nM
|
|
|
|
CP0497870
|
3-(4-(1-cyclohexylethoxy)benzyl)-5-methyloxazolidin-2-one
Show/Hide
|
C19H27NO3
|
1
|
| 1 |
EC50 = 7.9 nM
|
|
|
|
CP0447261
|
(1S,2S,4S,5R,6S)-2-amino-4-[(3-chlorobenzoyl)amino]bicyclo[3.1.0]hexane-2,6-dicarboxylic acid
Show/Hide
|
C15H15ClN2O5
|
2
|
| 1 |
EC50 = 8.37 nM
|
|
|
| 2 |
Ki = 85.3 nM
|
|
|
|
CP0388455
|
3-(cyclopropylmethyl)-7-[2-(4-fluorophenyl)propoxy]-8-(trifluoromethyl)-[1,2,4]triazolo[4,3-a]pyridine
Show/Hide
|
C20H19F4N3O
|
1
|
| 1 |
EC50 = 10 nM
|
|
|
|
CP0388458
|
3-(cyclopropylmethyl)-7-[2-(4-fluorophenyl)-2-methylpropoxy]-8-(trifluoromethyl)-[1,2,4]triazolo[4,3-a]pyridine
Show/Hide
|
C21H21F4N3O
|
1
|
| 1 |
EC50 = 11 nM
|
|
|
|
CP0461681
|
8-chloro-7-[(2-chlorophenyl)methoxy]-3-(cyclopropylmethyl)-[1,2,4]triazolo[4,3-a]pyridine
Show/Hide
|
C17H15Cl2N3O
|
1
|
| 1 |
EC50 = 11 nM
|
|
|
|
CP0508177
|
8-chloro-3-(cyclopropylmethyl)-7-[(3-phenylphenyl)methoxy]-[1,2,4]triazolo[4,3-a]pyridine
Show/Hide
|
C23H20ClN3O
|
1
|
| 1 |
EC50 = 13 nM
|
|
|
|
CP0512449
|
7-[[1-(4-chlorophenyl)cyclopropyl]methoxy]-3-(cyclopropylmethyl)-8-(trifluoromethyl)-[1,2,4]triazolo[4,3-a]pyridine
Show/Hide
|
C21H19ClF3N3O
|
1
|
| 1 |
EC50 = 13 nM
|
|
|
|
CP0502184
|
3-(4-(cyclohexylmethoxy)benzyl)-5-methyloxazolidin-2-one
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|
C18H25NO3
|
1
|
| 1 |
EC50 = 15 nM
|
|
|
|
CP0388456
|
3-(cyclopropylmethyl)-7-[[1-(4-fluorophenyl)cyclopropyl]methoxy]-8-(trifluoromethyl)-[1,2,4]triazolo[4,3-a]pyridine
Show/Hide
|
C21H19F4N3O
|
1
|
| 1 |
EC50 = 16 nM
|
|
|
|
CP0476634
|
(1S,2S,4S,5R,6S)-2-amino-4-[(4-methoxybenzoyl)amino]bicyclo[3.1.0]hexane-2,6-dicarboxylic acid
Show/Hide
|
C16H18N2O6
|
2
|
| 1 |
EC50 = 16 nM
|
|
|
| 2 |
Ki = 188 nM
|
|
|
|
CP0508175
|
8-chloro-7-[(3-chlorophenyl)methoxy]-3-(cyclopropylmethyl)-[1,2,4]triazolo[4,3-a]pyridine
Show/Hide
|
C17H15Cl2N3O
|
1
|
| 1 |
EC50 = 17 nM
|
|
|
|
CP0396668
|
(1S,2S,4S,5R,6S)-2-amino-4-[(2-fluorobenzoyl)amino]bicyclo[3.1.0]hexane-2,6-dicarboxylic acid
Show/Hide
|
C15H15FN2O5
|
2
|
| 1 |
EC50 = 17.1 nM
|
|
|
| 2 |
Ki = 218 nM
|
|
|
|
CP0461682
|
8-chloro-3-(cyclopropylmethyl)-7-(1,2,3,4-tetrahydronaphthalen-2-yloxy)-[1,2,4]triazolo[4,3-a]pyridine
Show/Hide
|
C20H20ClN3O
|
1
|
| 1 |
EC50 = 18 nM
|
|
|
|
CP0465824
|
(1S,2S,4S,5R,6S)-2-amino-4-[(3-fluorobenzoyl)amino]bicyclo[3.1.0]hexane-2,6-dicarboxylic acid
Show/Hide
|
C15H15FN2O5
|
2
|
| 1 |
EC50 = 18.1 nM
|
|
|
| 2 |
Ki = 214 nM
|
|
|
|
CP0390069
|
(1S,2S,4S,5R,6S)-2-amino-4-[(4-fluorobenzoyl)amino]bicyclo[3.1.0]hexane-2,6-dicarboxylic acid
Show/Hide
|
C15H15FN2O5
|
2
|
| 1 |
EC50 = 19.1 nM
|
|
|
| 2 |
Ki = 330 nM
|
|
|
|
CP0447263
|
(1S,2S,4S,5R,6S)-2-amino-4-benzamidobicyclo[3.1.0]hexane-2,6-dicarboxylic acid
Show/Hide
|
C15H16N2O5
|
2
|
| 1 |
EC50 = 19.8 nM
|
|
|
| 2 |
Ki = 294 nM
|
|
|
|
CP0512451
|
8-chloro-3-(cyclopropylmethyl)-7-[(2-phenylphenyl)methoxy]-[1,2,4]triazolo[4,3-a]pyridine
Show/Hide
|
C23H20ClN3O
|
1
|
| 1 |
EC50 = 20 nM
|
|
|
|
CP0390062
|
(1S,2S,4S,5R,6S)-2,4-diaminobicyclo[3.1.0]hexane-2,6-dicarboxylic acid
Show/Hide
|
C8H12N2O4
|
2
|
| 1 |
EC50 = 21.2 nM
|
|
|
| 2 |
Ki = 4410 nM
|
|
|
|
CP0388051
|
(5S)-3-(4-(1-cyclohexylethoxy)benzyl)-5-methyloxazolidin-2-one
Show/Hide
|
C19H27NO3
|
1
|
| 1 |
EC50 = 22.1 nM
|
|
|
|
CP0510532
|
(R)-3-((2'-ethoxybiphenyl-4-yl)methyl)-5-methyloxazolidin-2-one
Show/Hide
|
C19H21NO3
|
1
|
| 1 |
EC50 = 26 nM
|
|
|
|
CP0465823
|
(1S,2S,4S,5R,6S)-2-amino-4-[(2-methoxybenzoyl)amino]bicyclo[3.1.0]hexane-2,6-dicarboxylic acid
Show/Hide
|
C16H18N2O6
|
2
|
| 1 |
EC50 = 26.5 nM
|
|
|
| 2 |
Ki = 151 nM
|
|
|
|
CP0491369
|
(R)-3-((2'-chlorobiphenyl-4-yl)methyl)-5-methyloxazolidin-2-one
Show/Hide
|
C17H16ClNO2
|
1
|
| 1 |
EC50 = 28 nM
|
|
|
|
CP0388454
|
3-(cyclopropylmethyl)-7-phenylmethoxy-8-(trifluoromethyl)-[1,2,4]triazolo[4,3-a]pyridine
Show/Hide
|
C18H16F3N3O
|
1
|
| 1 |
EC50 = 28 nM
|
|
|
|
CP0512452
|
8-chloro-3-(cyclopropylmethyl)-7-(naphthalen-2-ylmethoxy)-[1,2,4]triazolo[4,3-a]pyridine
Show/Hide
|
C21H18ClN3O
|
1
|
| 1 |
EC50 = 29 nM
|
|
|
|
CP0293829
|
(R)-3-((3'-chloro-4'-fluorobiphenyl-4-yl)methyl)-5-methyloxazolidin-2-one
Show/Hide
|
C17H15ClFNO2
|
1
|
| 1 |
EC50 = 30 nM
|
|
|
|
CP0092081
|
2-[[(3R,4R)-4-[2-fluoro-4-(trifluoromethoxy)phenyl]-3-methylpiperidin-1-yl]methyl]-1-methylimidazo[4,5-b]pyridine
Show/Hide
|
C21H22F4N4O
|
1
|
| 1 |
EC50 = 31 nM
|
|
|
|
CP0174720
|
(R)-3-((2'-fluoro-4'-(trifluoromethoxy)biphenyl-4-yl)methyl)-5-methyloxazolidin-2-one
Show/Hide
|
C18H15F4NO3
|
1
|
| 1 |
EC50 = 32 nM
|
|
|
|
CP0508179
|
8-chloro-3-(cyclopropylmethyl)-7-(2-phenylethoxy)-[1,2,4]triazolo[4,3-a]pyridine
Show/Hide
|
C18H18ClN3O
|
1
|
| 1 |
EC50 = 32 nM
|
|
|
|
CP0388052
|
(R)-3-((2'-fluorobiphenyl-4-yl)methyl)-5-methyloxazolidin-2-one
Show/Hide
|
C17H16FNO2
|
1
|
| 1 |
EC50 = 35 nM
|
|
|
|
CP0443359
|
(R)-3-((2'-methoxybiphenyl-4-yl)methyl)-5-methyloxazolidin-2-one
Show/Hide
|
C18H19NO3
|
1
|
| 1 |
EC50 = 41 nM
|
|
|
|
CP0447264
|
(1S,2S,4S,5R,6S)-2-amino-4-[(2-chlorobenzoyl)amino]bicyclo[3.1.0]hexane-2,6-dicarboxylic acid
Show/Hide
|
C15H15ClN2O5
|
2
|
| 1 |
EC50 = 42.5 nM
|
|
|
| 2 |
Ki = 391 nM
|
|
|
|
CP0464987
|
1-Methyl-2-((4-(4-(trifluoromethyl)phenyl)piperidin-1-yl)methyl)-1H-imidazo[4,5-b]pyridine
Show/Hide
|
C20H21F3N4
|
1
|
| 1 |
EC50 = 43 nM
|
|
|
|
CP0356641
|
(1S,2S,4S,5R,6S)-2-amino-4-[(3-methoxybenzoyl)amino]bicyclo[3.1.0]hexane-2,6-dicarboxylic acid
Show/Hide
|
C16H18N2O6
|
2
|
| 1 |
EC50 = 47.5 nM
|
|
|
| 2 |
Ki = 412 nM
|
|
|
|
CP0515804
|
(R)-3-((4'-methoxybiphenyl-4-yl)methyl)-5-methyloxazolidin-2-one
Show/Hide
|
C18H19NO3
|
1
|
| 1 |
EC50 = 53 nM
|
|
|
|
CP0388453
|
8-chloro-7-[(4-chlorophenyl)methoxy]-3-(cyclopropylmethyl)-[1,2,4]triazolo[4,3-a]pyridine
Show/Hide
|
C17H15Cl2N3O
|
1
|
| 1 |
EC50 = 60 nM
|
|
|
|
CP0070609
|
(R)-3-((2',4'-difluorobiphenyl-4-yl)methyl)-5-methyloxazolidin-2-one
Show/Hide
|
C17H15F2NO2
|
1
|
| 1 |
EC50 = 70 nM
|
|
|
|
CP0388053
|
3-(4-(1-cyclohexylethoxy)benzyl)-1,3-oxazinan-2-one
Show/Hide
|
C19H27NO3
|
1
|
| 1 |
EC50 = 75 nM
|
|
|
|
CP0510509
|
(R)-3-((4'-chlorobiphenyl-4-yl)methyl)-5-methyloxazolidin-2-one
Show/Hide
|
C17H16ClNO2
|
1
|
| 1 |
EC50 = 76 nM
|
|
|
|
CP0347800
|
2-[[(3R,4R)-4-[2-methoxy-4-(trifluoromethyl)phenyl]-3-methylpiperidin-1-yl]methyl]-1-methylimidazo[4,5-b]pyridine
Show/Hide
|
C22H25F3N4O
|
1
|
| 1 |
EC50 = 76 nM
|
|
|
|
CP0479008
|
(R)-3-((4'-fluorobiphenyl-4-yl)methyl)-5-methyloxazolidin-2-one
Show/Hide
|
C17H16FNO2
|
1
|
| 1 |
EC50 = 84 nM
|
|
|
|
CP0523244
|
(5R)-3-((6-(1-cyclohexylethoxy)pyridin-3-yl)methyl)-5-methyloxazolidin-2-one
Show/Hide
|
C18H26N2O3
|
1
|
| 1 |
EC50 = 88 nM
|
|
|
|
CP0504169
|
(R)-3-((4'-ethoxybiphenyl-4-yl)methyl)-5-methyloxazolidin-2-one
Show/Hide
|
C19H21NO3
|
1
|
| 1 |
EC50 = 97 nM
|
|
|
|
CP0372007
|
3-(4-(cyclohexylmethoxy)benzyl)-1,3-oxazinan-2-one
Show/Hide
|
C18H25NO3
|
1
|
| 1 |
EC50 = 117 nM
|
|
|
|
CP0515805
|
(R)-3-(biphenyl-4-ylmethyl)-5-methyloxazolidin-2-one
Show/Hide
|
C17H17NO2
|
1
|
| 1 |
EC50 = 142 nM
|
|
|
|
CP0510512
|
(R)-3-((3'-chlorobiphenyl-4-yl)methyl)-5-methyloxazolidin-2-one
Show/Hide
|
C17H16ClNO2
|
1
|
| 1 |
EC50 = 158 nM
|
|
|
|
CP0565501
|
8-chloro-3-(cyclopropylmethyl)-7-phenylmethoxy-[1,2,4]triazolo[4,3-a]pyridine
Show/Hide
|
C17H16ClN3O
|
1
|
| 1 |
EC50 = 180 nM
|
|
|
|
CP0386090
|
(R)-5-methyl-3-((4'-(trifluoromethoxy)biphenyl-4-yl)methyl)oxazolidin-2-one
Show/Hide
|
C18H16F3NO3
|
1
|
| 1 |
EC50 = 183 nM
|
|
|
|
CP0523245
|
3-(4-(2-cyclohexylethoxy)benzyl)-5-methyloxazolidin-2-one
Show/Hide
|
C19H27NO3
|
1
|
| 1 |
EC50 = 203 nM
|
|
|
|
CP0388457
|
8-[[8-chloro-3-(cyclopropylmethyl)-[1,2,4]triazolo[4,3-a]pyridin-7-yl]oxymethyl]isoquinoline
Show/Hide
|
C20H17ClN4O
|
1
|
| 1 |
EC50 = 230 nM
|
|
|
|
CP0515806
|
3-(4-(cyclohexyloxy)benzyl)-5-methyloxazolidin-2-one
Show/Hide
|
C17H23NO3
|
1
|
| 1 |
EC50 = 236 nM
|
|
|
|
CP0385921
|
(1S,2S,4S,5R,6S)-4-acetamido-2-aminobicyclo[3.1.0]hexane-2,6-dicarboxylic acid
Show/Hide
|
C10H14N2O5
|
2
|
| 1 |
EC50 = 257 nM
|
|
|
| 2 |
Ki = 898 nM
|
|
|
|
CP0468499
|
3-(4-(benzyloxy)benzyl)-5-methyloxazolidin-2-one
Show/Hide
|
C18H19NO3
|
1
|
| 1 |
EC50 = 262 nM
|
|
|
|
CP0515807
|
(R)-3-((3'-methoxybiphenyl-4-yl)methyl)-5-methyloxazolidin-2-one
Show/Hide
|
C18H19NO3
|
1
|
| 1 |
EC50 = 275 nM
|
|
|
|
CP0515808
|
(R)-3-((3'-fluorobiphenyl-4-yl)methyl)-5-methyloxazolidin-2-one
Show/Hide
|
C17H16FNO2
|
1
|
| 1 |
EC50 = 280 nM
|
|
|
|
CP0174718
|
(R)-3-((6-(2-fluoro-4-(trifluoromethoxy)phenyl)pyridin-3-yl)methyl)-5-methyloxazolidin-2-one
Show/Hide
|
C17H14F4N2O3
|
1
|
| 1 |
EC50 = 380 nM
|
|
|
|
CP0523246
|
3-(4-(cyclohexylmethoxy)benzyl)-1,8-dioxa-3-azaspiro[4.5]decan-2-one
Show/Hide
|
C21H29NO4
|
1
|
| 1 |
EC50 = 384 nM
|
|
|
|
CP0519556
|
(1S,2S,4S,5R,6S)-2-amino-4-(benzylamino)bicyclo[3.1.0]hexane-2,6-dicarboxylic acid
Show/Hide
|
C15H18N2O4
|
2
|
| 1 |
EC50 = 508 nM
|
|
|
| 2 |
Ki = 11200 nM
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CP0515809
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3-(4-(cyclohexylmethoxy)benzyl)oxazolidin-2-one
Show/Hide
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C17H23NO3
|
1
|
| 1 |
EC50 = 590 nM
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|
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CP0515810
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(R)-3-((6-(3-chloro-4-fluorophenyl)pyridin-3-yl)methyl)-5-methyloxazolidin-2-one
Show/Hide
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C16H14ClFN2O2
|
1
|
| 1 |
EC50 = 595 nM
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|
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CP0508178
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8-chloro-3-(cyclopropylmethyl)-7-[(3-pyrimidin-5-ylphenyl)methoxy]-[1,2,4]triazolo[4,3-a]pyridine
Show/Hide
|
C21H18ClN5O
|
1
|
| 1 |
EC50 = 720 nM
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|
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CP0454449
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(1S,2S,4S,5R,6S)-2-amino-4-(3-phenylpropanoylamino)bicyclo[3.1.0]hexane-2,6-dicarboxylic acid
Show/Hide
|
C17H20N2O5
|
3
|
| 1 |
EC50 = 893 nM
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|
|
| 2 |
IC50 = 5540 nM
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|
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| 3 |
Ki = 595 nM
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CP0498533
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(R)-3-((5-(3,4-difluorophenyl)pyridin-2-yl)methyl)-5-methyloxazolidin-2-one
Show/Hide
|
C16H14F2N2O2
|
1
|
| 1 |
EC50 = 1800 nM
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|
|
|
CP0002355
|
(2S)-2-aminopentanedioic acid
Show/Hide
|
C5H9NO4
|
2
|
| 1 |
EC50 = 1800 nM
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|
|
| 2 |
Ki = 1819.7 nM
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CP0438458
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8-chloro-6-morpholin-4-yl-2-propylisoquinolin-1-one
Show/Hide
|
C16H19ClN2O2
|
1
|
| 1 |
EC50 = 2511.89 nM
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|
|
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CP0573980
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3-cycloheptyl-7-(2,6-dichlorophenyl)-[1,2,4]triazolo[4,3-a]pyridine
Show/Hide
|
C19H19Cl2N3
|
1
|
| 1 |
EC50 = 2700 nM
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|
|
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CP0386091
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(R)-3-((4'-((dimethylamino)methyl)biphenyl-4-yl)methyl)-5-methyloxazolidin-2-one
Show/Hide
|
C20H24N2O2
|
1
|
| 1 |
EC50 = 3060 nM
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|
|
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CP0396669
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(1S,2S,4S,5R,6S)-2-amino-4-(cyclohexanecarbonylamino)bicyclo[3.1.0]hexane-2,6-dicarboxylic acid
Show/Hide
|
C15H22N2O5
|
3
|
| 1 |
EC50 = 3390 nM
|
|
|
| 2 |
IC50 = 12000 nM
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|
|
| 3 |
Ki = 1520 nM
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CP0070608
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(R)-3-((6-(3,4-difluorophenyl)pyridin-3-yl)methyl)-5-methyloxazolidin-2-one
Show/Hide
|
C16H14F2N2O2
|
1
|
| 1 |
EC50 = 3400 nM
|
|
|
|
CP0386092
|
(R)-5-methyl-3-(4-(pyrimidin-5-yl)benzyl)oxazolidin-2-one
Show/Hide
|
C15H15N3O2
|
1
|
| 1 |
EC50 = 4380 nM
|
|
|
|
CP0504170
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(R)-5-methyl-3-(4-(pyridin-4-yl)benzyl)oxazolidin-2-one
Show/Hide
|
C16H16N2O2
|
1
|
| 1 |
EC50 = 4790 nM
|
|
|
|
CP0510519
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(R)-3-((2'-((dimethylamino)methyl)biphenyl-4-yl)methyl)-5-methyloxazolidin-2-one
Show/Hide
|
C20H24N2O2
|
1
|
| 1 |
EC50 = 6360 nM
|
|
|
|
CP0504171
|
(R)-5-methyl-3-(4-(pyridin-3-yl)benzyl)oxazolidin-2-one
Show/Hide
|
C16H16N2O2
|
1
|
| 1 |
EC50 = 7550 nM
|
|
|
|
CP0479010
|
5-methyl-3-(4-(tetrahydro-2H-pyran-4-yloxy)benzyl)oxazolidin-2-one
Show/Hide
|
C16H21NO4
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0504172
|
(5R)-5-methyl-3-(4-(1-(piperidin-1-yl)ethyl)benzyl)oxazolidin-2-one
Show/Hide
|
C18H26N2O2
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0515811
|
3-(4-(pyridin-3-ylmethoxy)benzyl)-1,3-oxazinan-2-one
Show/Hide
|
C17H18N2O3
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0515812
|
(R)-3-(4-((cyclohexyl(methyl)amino)methyl)benzyl)-5-methyloxazolidin-2-one
Show/Hide
|
C19H28N2O2
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0077643
|
5-methyl-2-(phenoxymethyl)-6,7-dihydro-[1,3]thiazolo[5,4-c]pyridin-4-one
Show/Hide
|
C14H14N2O2S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0133913
|
7-(benzyloxy)-2,3-dihydro-4H-chromen-4-one
Show/Hide
|
C16H14O3
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0379848
|
7-(phenoxymethyl)chroman-4-one
Show/Hide
|
C16H14O3
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0379852
|
2-(2-phenylethynyl)-5,6-dihydro-4H-1,3-benzothiazol-7-one
Show/Hide
|
C15H11NOS
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0397096
|
4-oxochroman-7-yl benzoate
Show/Hide
|
C16H12O4
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0871656
|
Trans-1-Amino-2-carboxymethyl-cyclopropanecarboxylic acid
Show/Hide
|
C6H9NO4
|
2
|
| 1 |
EC50 = 10000 nM
|
|
|
| 2 |
Ki = 10471.29 nM
|
|
|
|
CP0099614
|
5-(5-fluoropyridin-2-yl)-2-(phenoxymethyl)-6,7-dihydropyrazolo[1,5-a]pyrazin-4-one
Show/Hide
|
C18H15FN4O2
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0395090
|
5-(4-fluorophenyl)-2-phenylmethoxy-6,7-dihydropyrazolo[1,5-a]pyrazin-4-one
Show/Hide
|
C19H16FN3O2
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0069484
|
(+/-)-trans-ACPD
Show/Hide
|
C7H11NO4
|
1
|
| 1 |
EC50 = 13000 nM
|
|
|
|
CP0466650
|
8-chloro-3-(cyclopropylmethyl)-7-(pyridin-3-ylmethoxy)-[1,2,4]triazolo[4,3-a]pyridine
Show/Hide
|
C16H15ClN4O
|
1
|
| 1 |
EC50 > 15000 nM
|
|
|
|
CP0049004
|
(1S,3R)-1-aminocyclopentane-1,3-dicarboxylic acid;hydrate
Show/Hide
|
C7H11NO4
|
1
|
| 1 |
EC50 = 18000 nM
|
|
|
|
CP0876173
|
Cis-1-Amino-2-carboxymethyl-cyclopropanecarboxylic acid
Show/Hide
|
C6H9NO4
|
2
|
| 1 |
EC50 = 23000 nM
|
|
|
| 2 |
Ki = 22387.21 nM
|
|
|
|
CP0390064
|
(1S,2S,4S,5R,6S)-2-amino-4-[(2-cyclohexylacetyl)amino]bicyclo[3.1.0]hexane-2,6-dicarboxylic acid
Show/Hide
|
C16H24N2O5
|
3
|
| 1 |
EC50 > 25000 nM
|
|
|
| 2 |
IC50 = 7660 nM
|
|
|
| 3 |
Ki = 627 nM
|
|
|
|
CP0103369
|
2-Amino-4-(4-hydroxy-[1,2,5]thiadiazol-3-yl)-butyric acid
Show/Hide
|
C6H9N3O3S
|
1
|
| 1 |
EC50 = 37000 nM
|
|
|
|
CP0268363
|
2-Amino-4-(4-hydroxy-[1,2,5]thiadiazol-3-yl)-butyric acid
Show/Hide
|
C6H9N3O3S
|
1
|
| 1 |
EC50 = 40000 nM
|
|
|
|
CP0464373
|
8-chloro-3-(cyclopropylmethyl)-7-(pyridin-2-ylmethoxy)-[1,2,4]triazolo[4,3-a]pyridine
Show/Hide
|
C16H15ClN4O
|
1
|
| 1 |
EC50 > 3000 nM
|
|
|
