Compound ID |
Compound Name |
Compound Formula |
CP0057346
|
3-(2-aminopropyl)-1H-indol-5-ol
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C11H14N2O
|
1
|
1 |
EC50 = 1.8 nM
|
|
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CP0001238
|
14C-5-hydroxy tryptamine creatinine disulfate
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C10H12N2O
|
1
|
1 |
EC50 = 2.8 nM
|
|
|
CP0099665
|
2-(5-Methoxy-1H-indol-3-yl)-1-methyl-ethylamine
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C12H16N2O
|
1
|
1 |
EC50 = 3.1 nM
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|
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CP0044585
|
1-((S)-2-aminopropyl)-1H-indazol-6-ol
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|
C10H13N3O
|
1
|
1 |
EC50 = 3.7 nM
|
|
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CP0394695
|
phenyl 2-[[8-[(2R)-2-aminopropyl]-2,3,6,7-tetrahydrofuro[2,3-f][1]benzofuran-4-yl]methoxy]acetate
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|
C22H25NO5
|
1
|
1 |
EC50 = 4.5 nM
|
|
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CP0431209
|
1-(2-aminoethyl)-1H-indazol-6-ol
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|
C9H11N3O
|
1
|
1 |
EC50 = 4.5 nM
|
|
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CP0422213
|
1-((S)-2-aminopropyl)-7-chloro-1H-indazol-6-ol
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|
C10H12ClN3O
|
1
|
1 |
EC50 = 4.9 nM
|
|
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CP0372474
|
1-((S)-2-aminopropyl)-7-fluoro-1H-indazol-6-ol
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|
C10H12FN3O
|
1
|
1 |
EC50 = 5.5 nM
|
|
|
CP0386221
|
(2S)-1-(6-methoxy-1H-indazol-1-yl)propan-2-amine
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|
C11H15N3O
|
1
|
1 |
EC50 = 6.7 nM
|
|
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CP0431212
|
1-((S)-2-aminopropyl)-7-methyl-1H-indazol-6-ol
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|
C11H15N3O
|
1
|
1 |
EC50 = 7.3 nM
|
|
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CP0373329
|
(R)-2-[8-(2-methoxy-ethoxymethyl)-2,3,6,7-tetrahydro-benzo[1,2-b;4,5-b']difuran-4-yl]-1-methyl-ethylamine
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|
C17H25NO4
|
1
|
1 |
EC50 = 8.6 nM
|
|
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CP0373330
|
(R)-2-(8-methoxymethyl-2,3,6,7-tetrahydro-benzo[1,2-b;4,5-b']difuran-4-yl)-1-methyl-ethylamine
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|
C15H21NO3
|
1
|
1 |
EC50 = 12.6 nM
|
|
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CP0057042
|
(R)-1-(4-iodo-2,5-dimethoxyphenyl)propan-2-amine
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|
C11H16INO2
|
1
|
1 |
EC50 = 30.2 nM
|
|
|
CP0442976
|
(1R,2R)-2-amino-1-(8-bromo-2,3,6,7-tetrahydro-benzo[1,2-b;4,5-b']difuran-4-yl)-propan-1-ol
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|
C13H16BrNO3
|
1
|
1 |
EC50 = 39 nM
|
|
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CP0071154
|
2-(5-methoxy-1H-indol-3-yl)-N,N-dimethyl-ethanamine
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|
C13H18N2O
|
1
|
1 |
EC50 = 77.8 nM
|
|
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CP0394899
|
(R)-1-methyl-2-[8-(3-methyl-[1,2,4]oxadiazol-5-ylmethyl)-benzo[1,2-b;4,5-b']difuran-4-yl]-ethylamine
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|
C17H17N3O3
|
1
|
1 |
EC50 = 82 nM
|
|
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CP0372472
|
1-((R)-2-aminopropyl)-1H-indazol-6-ol
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|
C10H13N3O
|
1
|
1 |
EC50 = 87.3 nM
|
|
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CP0394693
|
(R)-1-methyl-2-[8-(3-methyl-[1,2,4]oxadiazol-5-ylmethyl)-2,3,6,7-tetrahydro-benzo[1,2-b;4,5-b']difuran-4-yl]-ethylamine
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|
C17H21N3O3
|
1
|
1 |
EC50 = 689 nM
|
|
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CP0031743
|
1H-imidazo[4,5-c]pyridine derivative
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|
C18H26N4O2S
|
1
|
1 |
Ki = 0.37 nM
|
|
|
CP0046703
|
1-(2-{4-[5-chloro-1-(4-fluorophenyl)-1H-indol-3-yl]piperidin-1-yl}ethyl)imidazolidin-2-one
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|
C24H26ClFN4O
|
1
|
1 |
Ki = 0.51 nM
|
|
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CP0005956
|
1-(8-Chloro-dibenzo[b,f]oxepin-10-yl)-4-methyl-piperazine
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|
C19H19ClN2O
|
1
|
1 |
Ki = 3 nM
|
|
|
CP0003324
|
1-(8-Chloro-5H-dibenzo[a,d]cyclohepten-10-yl)-4-methyl-piperazine
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|
C20H21ClN2
|
1
|
1 |
Ki = 6 nM
|
|
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CP0008953
|
1-(2-Chloro-dibenzo[b,f]oxepin-10-yl)-4-methyl-piperazine
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|
C19H19ClN2O
|
1
|
1 |
Ki = 6 nM
|
|
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CP0010829
|
1-Dibenzo[b,f]oxepin-10-yl-4-methyl-piperazine
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|
C19H20N2O
|
1
|
1 |
Ki = 6 nM
|
|
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CP0002406
|
1-(2-Chloro-5H-dibenzo[a,d]cyclohepten-10-yl)-4-methyl-piperazine
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|
C20H21ClN2
|
1
|
1 |
Ki = 7 nM
|
|
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CP0874541
|
4-Dibenzo[b,f]oxepin-10-yl-1-methyl-piperidine hydrochloride
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|
C20H22ClNO
|
1
|
1 |
Ki = 8 nM
|
|
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CP0885801
|
4-Dibenzo[b,f]oxepin-10-yl-1-ethyl-1,2,3,6-tetrahydro-pyridine hydrochloride
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|
C21H22ClNO
|
1
|
1 |
Ki = 14 nM
|
|
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CP0005197
|
1-Methyl-4-(5-methylene-5H-dibenzo[a,d]cyclohepten-10-yl)-piperazine
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|
C21H22N2
|
1
|
1 |
Ki = 18 nM
|
|
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CP0005613
|
8-Chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,f][1,4]oxazepine
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|
C18H18ClN3O
|
1
|
1 |
Ki = 19 nM
|
|
|
CP0391139
|
4-Dibenzo[b,f]oxepin-10-yl-1-methyl-1,2,3,6-tetrahydro-pyridine
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|
C20H19NO
|
1
|
1 |
Ki = 20 nM
|
|
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CP0183655
|
1-Methyl-4-(5-methyl-5H-dibenzo[a,d]cyclohepten-10-yl)-piperazine
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|
C21H24N2
|
1
|
1 |
Ki = 36 nM
|
|
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CP0406243
|
1-(2-{4-[5-(2-Ethyl-2H-[1,2,3]triazol-4-yl)-1-(4-fluoro-phenyl)-1H-indol-3-yl]-piperidin-1-yl}-ethyl)-imidazolidin-2-one
Show/Hide
|
C28H32FN7O
|
1
|
1 |
Ki = 37 nM
|
|
|
CP0448256
|
1-(2-{4-[1-(4-Fluoro-phenyl)-5-(2-methyl-2H-pyrazol-3-yl)-1H-indol-3-yl]-piperidin-1-yl}-ethyl)-imidazolidin-2-one
Show/Hide
|
C28H31FN6O
|
1
|
1 |
Ki = 45 nM
|
|
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CP0490676
|
1-(2-{4-[1-(4-Fluoro-phenyl)-5-pyridin-3-yl-1H-indol-3-yl]-piperidin-1-yl}-ethyl)-imidazolidin-2-one
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|
C29H30FN5O
|
1
|
1 |
Ki = 50 nM
|
|
|
CP0845312
|
1-Allyl-4-dibenzo[b,f]oxepin-10-yl-1,2,3,6-tetrahydro-pyridine hydrochloride
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|
C22H22ClNO
|
1
|
1 |
Ki = 51 nM
|
|
|
CP0384143
|
1-(2-{4-[1-(4-Fluoro-phenyl)-5-(2-methyl-2H-[1,2,3]triazol-4-yl)-1H-indol-3-yl]-piperidin-1-yl}-ethyl)-imidazolidin-2-one
Show/Hide
|
C27H30FN7O
|
1
|
1 |
Ki = 73 nM
|
|
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CP0004912
|
1-[5-Eth-(Z)-ylidene-5H-dibenzo[a,d]cyclohepten-10-yl]-4-methyl-piperazine
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|
C22H24N2
|
1
|
1 |
Ki = 110 nM
|
|
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CP0453890
|
1-(2-{4-[1-(4-Fluoro-phenyl)-5-pyrimidin-5-yl-1H-indol-3-yl]-piperidin-1-yl}-ethyl)-imidazolidin-2-one
Show/Hide
|
C28H29FN6O
|
1
|
1 |
Ki = 120 nM
|
|
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CP0492027
|
1-(2-{4-[1-(4-Fluoro-phenyl)-5-(1-methyl-1H-imidazol-2-yl)-1H-indol-3-yl]-piperidin-1-yl}-ethyl)-imidazolidin-2-one
Show/Hide
|
C28H31FN6O
|
1
|
1 |
Ki = 130 nM
|
|
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CP0376628
|
1-(2-{4-[1-(4-Fluoro-phenyl)-5-(3-methyl-3H-[1,2,3]triazol-4-yl)-1H-indol-3-yl]-piperidin-1-yl}-ethyl)-imidazolidin-2-one
Show/Hide
|
C27H30FN7O
|
1
|
1 |
Ki = 140 nM
|
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CP0392710
|
1-(2-{4-[1-(4-Fluoro-phenyl)-5-(2H-[1,2,3]triazol-4-yl)-1H-indol-3-yl]-piperidin-1-yl}-ethyl)-imidazolidin-2-one
Show/Hide
|
C26H28FN7O
|
1
|
1 |
Ki = 150 nM
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CP0404715
|
1-(2-{4-[1-(4-Fluoro-phenyl)-5-(1-methyl-1H-tetrazol-5-yl)-1H-indol-3-yl]-piperidin-1-yl}-ethyl)-imidazolidin-2-one
Show/Hide
|
C26H29FN8O
|
1
|
1 |
Ki = 180 nM
|
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CP0459887
|
1-(2-{4-[1-(4-Fluoro-phenyl)-5-(2-methyl-2H-[1,2,4]triazol-3-yl)-1H-indol-3-yl]-piperidin-1-yl}-ethyl)-imidazolidin-2-one
Show/Hide
|
C27H30FN7O
|
1
|
1 |
Ki = 190 nM
|
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CP0228798
|
1-(2-{4-[1-(4-Fluoro-phenyl)-5-(2-methyl-2H-tetrazol-5-yl)-1H-indol-3-yl]-piperidin-1-yl}-ethyl)-imidazolidin-2-one
Show/Hide
|
C26H29FN8O
|
1
|
1 |
Ki = 330 nM
|
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CP0277576
|
1-(2-{4-[1-(4-Fluoro-phenyl)-5-(1-methyl-1H-pyrazol-3-yl)-1H-indol-3-yl]-piperidin-1-yl}-ethyl)-imidazolidin-2-one
Show/Hide
|
C28H31FN6O
|
1
|
1 |
Ki = 330 nM
|
|
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CP0000272
|
1-(2-Chloro-5-isopropylidene-5H-dibenzo[a,d]cyclohepten-10-yl)-4-methyl-piperazine
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|
C23H25ClN2
|
1
|
1 |
Ki = 370 nM
|
|
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CP0011263
|
1-(5-Isopropylidene-5H-dibenzo[a,d]cyclohepten-10-yl)-4-methyl-piperazine
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|
C23H26N2
|
1
|
1 |
Ki = 390 nM
|
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CP0382930
|
1-(2-{4-[5-(1-Ethyl-1H-[1,2,3]triazol-4-yl)-1-(4-fluoro-phenyl)-1H-indol-3-yl]-piperidin-1-yl}-ethyl)-imidazolidin-2-one
Show/Hide
|
C28H32FN7O
|
1
|
1 |
Ki = 500 nM
|
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CP0502318
|
1-(2-{4-[1-(4-Fluoro-phenyl)-5-(1-methyl-1H-pyrazol-4-yl)-1H-indol-3-yl]-piperidin-1-yl}-ethyl)-imidazolidin-2-one
Show/Hide
|
C28H31FN6O
|
1
|
1 |
Ki = 1000 nM
|
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CP0429995
|
1-(2-{4-[1-(4-Fluoro-phenyl)-5-(4-methyl-4H-[1,2,4]triazol-3-yl)-1H-indol-3-yl]-piperidin-1-yl}-ethyl)-imidazolidin-2-one
Show/Hide
|
C27H30FN7O
|
1
|
1 |
Ki = 1100 nM
|
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CP0382893
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1-(2-{4-[1-(4-Fluoro-phenyl)-5-pyrimidin-2-yl-1H-indol-3-yl]-piperidin-1-yl}-ethyl)-imidazolidin-2-one
Show/Hide
|
C28H29FN6O
|
1
|
1 |
Ki = 1200 nM
|
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CP0126860
|
1-(2-{4-[1-(4-Fluoro-phenyl)-5-(1-methyl-1H-[1,2,3]triazol-4-yl)-1H-indol-3-yl]-piperidin-1-yl}-ethyl)-imidazolidin-2-one
Show/Hide
|
C27H30FN7O
|
1
|
1 |
Ki = 1500 nM
|
|
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CP0072419
|
(SNAP-8719)[4-(4-Amino-6,7-dimethoxy-quinazolin-2-yl)-octahydro-quinoxalin-1-yl]-furan-2-yl-methanone
Show/Hide
|
C22H28F3N3O2
|
1
|
1 |
Ki = 2600 nM
|
|
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CP0151333
|
1-(2-{4-[1-(4-Fluoro-phenyl)-5-(1-methyl-1H-[1,2,4]triazol-3-yl)-1H-indol-3-yl]-piperidin-1-yl}-ethyl)-imidazolidin-2-one
Show/Hide
|
C27H30FN7O
|
1
|
1 |
Ki = 2900 nM
|
|
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CP0040814
|
[4-(4-amino-6,7-dimethoxyquinazolin-2-yl)piperazin-1-yl]-(furan-2-yl)methanone
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|
C19H21N5O4
|
1
|
1 |
Ki > 4200 nM
|
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|