Brief Information of the Cell Line and Protein
Cell Line ID: CL000997 , SAE
 Cell Line Info 
Synonyms
Squalus Acanthias Embryo
Category Spontaneously immortalized cell line
Organism
Squalus acanthias (Spiny dogfish)
Protein ID: PT01462 , Bromodomain-containing protein 4
 Protein Info 
Gene Name BRD4
Organism Homo sapiens, Human
Protein Classification Epigenetic regulator
Uniprot ID O60885
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000997
 Cell Line Info 
 Protein ID: PT01462
 Protein Info 
 
Compound ID Compound Name Compound Formula
CP0202113
 Compound Info 
6-[(2-amino-4-hydroxy-5-methylphenyl)diazenyl]-3,4-dihydro-1H-quinolin-2-one
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C16H16N4O2
  4
1
IC50 = 490 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
2
IC50 = 510 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
3
IC50 = 530 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
4
IC50 = 580 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0033805
 Compound Info 
4-[(2-amino-4-hydroxy-5-methylphenyl)diazenyl]-N-cyclopentylbenzenesulfonamide
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C18H22N4O3S
  4
1
IC50 = 730 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
2
IC50 = 790 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
3
IC50 = 810 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
4
IC50 = 860 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0004236
 Compound Info 
(+)-JQ1
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C23H25ClN4O2S
  4
1
IC50 = 1380 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
2
IC50 = 1490 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
3
IC50 = 1510 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
4
IC50 = 1630 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0058410
 Compound Info 
2-[4-(2-hydroxyethoxy)-3,5-dimethylphenyl]-5,7-dimethoxy-3H-quinazolin-4-one
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C20H22N2O5
  4
1
IC50 = 2630 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
2
IC50 = 2740 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
3
IC50 = 3730 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
4
IC50 = 3850 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0424094
 Compound Info 
2-(5-tert-butyl-1,2-oxazol-3-yl)-5-(3-chloro-5-fluorophenyl)-1,3,4-oxadiazole
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C15H13ClFN3O2
  4
1
IC50 = 3900 nM
 Bioactivity Info 
   TI
   LI
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   TS
2
IC50 = 4300 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
3
IC50 = 7700 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
4
IC50 = 7900 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS