Compound ID |
Compound Name |
Compound Formula |
CP0554605
|
2-[1-[(2R)-2-(5-fluoro-2-methoxyphenyl)-2-[[(1S,5R)-8-oxabicyclo[3.2.1]octan-3-yl]oxy]ethyl]-5-methyl-2,4-dioxo-6-(triazol-2-yl)thieno[2,3-d]pyrimidin-3-yl]-2-methyl-N-(1-methylcyclopropyl)sulfonylpropanamide
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|
C33H39FN6O8S2
|
1
|
1 |
EC50 = 0.3 nM
|
|
|
CP0578524
|
1-[1-[(2R)-2-[2-(difluoromethoxy)-5-fluorophenyl]-2-[[(1S,5R)-8-oxabicyclo[3.2.1]octan-3-yl]oxy]ethyl]-5-methyl-2,4-dioxo-6-(triazol-2-yl)thieno[2,3-d]pyrimidin-3-yl]-N-(1-methylcyclopropyl)sulfonylcyclopropane-1-carboxamide
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|
C33H35F3N6O8S2
|
1
|
1 |
EC50 = 0.9 nM
|
|
|
CP0537257
|
(2R)-2-[1-[(2R)-2-(2-methoxyphenyl)-2-[[(1S,5R)-8-oxabicyclo[3.2.1]octan-3-yl]oxy]ethyl]-5-methyl-6-(1,3-oxazol-2-yl)-2,4-dioxothieno[2,3-d]pyrimidin-3-yl]-N-(1-methylcyclopropyl)sulfonylpropanamide
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|
C33H38N4O9S2
|
1
|
1 |
EC50 = 1 nM
|
|
|
CP0554604
|
2-[1-[(2R)-2-(2-methoxyphenyl)-2-[[(1S,5R)-8-oxabicyclo[3.2.1]octan-3-yl]oxy]ethyl]-5-methyl-6-(1,3-oxazol-2-yl)-2,4-dioxothieno[2,3-d]pyrimidin-3-yl]-2-methyl-N-(1-methylcyclopropyl)sulfonylpropanamide
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|
C34H40N4O9S2
|
1
|
1 |
EC50 = 1 nM
|
|
|
CP0554606
|
1-[1-[(2R)-2-(2-methoxyphenyl)-2-[[(1S,5R)-8-oxabicyclo[3.2.1]octan-3-yl]oxy]ethyl]-5-methyl-2,4-dioxo-6-(triazol-2-yl)thieno[2,3-d]pyrimidin-3-yl]-N-(1-methylcyclopropyl)sulfonylcyclopropane-1-carboxamide
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|
C33H38N6O8S2
|
1
|
1 |
EC50 = 1 nM
|
|
|
CP0563057
|
2-[1-[(2R)-2-(2-methoxyphenyl)-2-[[(1S,5R)-8-oxabicyclo[3.2.1]octan-3-yl]oxy]ethyl]-5-methyl-2,4-dioxo-6-(triazol-2-yl)thieno[2,3-d]pyrimidin-3-yl]-2-methyl-N-(1-methylcyclopropyl)sulfonylpropanamide
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|
C33H40N6O8S2
|
1
|
1 |
EC50 = 1 nM
|
|
|