| Compound ID |
Compound Name |
Compound Formula |
|
CP0542631
|
N-[3-[(6R)-4-amino-2-cyano-6-methyl-7H-pyrazolo[1,5-a]pyrazin-6-yl]-4-fluorophenyl]-5-(difluoromethoxy)pyridine-2-carboxamide
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|
C21H16F3N7O2
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0572071
|
N-[3-[(6R)-4-amino-2-cyano-6-methyl-7H-pyrazolo[1,5-a]pyrazin-6-yl]-4-fluorophenyl]-5-cyanopyridine-2-carboxamide
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|
C21H15FN8O
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0558300
|
N-[3-[(6R)-4-amino-2-cyano-6-methyl-7H-pyrazolo[1,5-a]pyrazin-6-yl]-4-fluorophenyl]-5-(fluoromethoxy)pyrazine-2-carboxamide
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|
C20H16F2N8O2
|
1
|
| 1 |
IC50 = 1.2 nM
|
|
|
|
CP0549717
|
N-[3-[(6R)-4-amino-2-cyano-6-methyl-7H-pyrazolo[1,5-a]pyrazin-6-yl]-4-fluorophenyl]-5-methoxypyrazine-2-carboxamide
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|
C20H17FN8O2
|
1
|
| 1 |
IC50 = 1.3 nM
|
|
|
|
CP0569898
|
N-[3-[(6R)-4-amino-2-cyano-6-methyl-7H-pyrazolo[1,5-a]pyrazin-6-yl]-4-fluorophenyl]-5-(difluoromethyl)pyrazine-2-carboxamide
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|
C20H15F3N8O
|
1
|
| 1 |
IC50 = 2.5 nM
|
|
|
|
CP0579632
|
N-[3-[(6R)-4-amino-2-cyano-6-methyl-7H-pyrazolo[1,5-a]pyrazin-6-yl]-4-fluorophenyl]-5-fluoropyridine-2-carboxamide
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|
C20H15F2N7O
|
1
|
| 1 |
IC50 = 2.6 nM
|
|
|
|
CP0283775
|
N-[3-[(6R)-8-amino-3-cyano-6-methyl-5H-imidazo[1,2-a]pyrazin-6-yl]-4-fluorophenyl]-5-cyanopyridine-2-carboxamide
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|
C21H15FN8O
|
1
|
| 1 |
IC50 = 3.3 nM
|
|
|
|
CP0558299
|
N-[3-[(6R)-8-amino-3-cyano-6-methyl-5H-imidazo[1,2-a]pyrazin-6-yl]-4-fluorophenyl]-5-chloropyridine-2-carboxamide
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|
C20H15ClFN7O
|
1
|
| 1 |
IC50 = 3.6 nM
|
|
|
|
CP0567739
|
N-[3-[(6R)-4-amino-2-cyano-6-methyl-7H-pyrazolo[1,5-a]pyrazin-6-yl]-4-fluorophenyl]-2-methyl-1,3-oxazole-4-carboxamide
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|
C19H16FN7O2
|
1
|
| 1 |
IC50 = 4.8 nM
|
|
|
|
CP0569897
|
N-[3-[(6R)-8-amino-3-cyano-6-methyl-5H-imidazo[1,2-a]pyrazin-6-yl]-4-fluorophenyl]-5-methoxypyrazine-2-carboxamide
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|
C20H17FN8O2
|
1
|
| 1 |
IC50 = 6.3 nM
|
|
|
|
CP0549715
|
N-[3-[(6R)-8-amino-2-cyano-6-methyl-5H-imidazo[1,2-a]pyrazin-6-yl]-4-fluorophenyl]-5-cyanopyridine-2-carboxamide
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|
C21H15FN8O
|
1
|
| 1 |
IC50 = 8.5 nM
|
|
|
|
CP0259790
|
N-[3-[(6R)-8-amino-3-cyano-6-methyl-5H-imidazo[1,2-a]pyrazin-6-yl]-4-fluorophenyl]-5-fluoropyridine-2-carboxamide
Show/Hide
|
C20H15F2N7O
|
1
|
| 1 |
IC50 = 12.6 nM
|
|
|
