Brief Information of the Cell Line and Protein
Cell Line ID: CL000790 , MR-5
Synonyms
MR 5
Category Cancer cell line
Organism
Homo sapiens (Human)
Protein ID: PT01032 , B1 bradykinin receptor
Gene Name BDKRB1
Organism Homo sapiens, Human
Protein Classification Membrane receptor
Uniprot ID P46663
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000790  Protein ID: PT01032
 
Compound ID Compound Name Compound Formula
CP0057919
(R)-N-(4-(4,5-dihydro-1H-imidazol-2-yl)phenethyl)-2-(1-(3,4-dichlorophenylsulfonyl)-3-oxo-1,2,3,4-tetrahydroquinoxalin-2-yl)acetamide
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C27H25Cl2N5O4S
 1
1
IC50 = 0.18 nM
   TI
   LI
   LO
   TS
CP0334933
(R)-1-(2-oxo-5-phenethyl-1-propyl-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl)-3-(4-(4-(pyridin-4-yl)piperazin-1-yl)phenyl)urea
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C36H39N7O2
 1
1
IC50 = 1.9 nM
   TI
   LI
   LO
   TS
CP0502742
4-bromo-5-[(2-chlorobenzoyl)amino]-N-[2-[1-(4-pyridinyl)-4-piperidinyl]ethyl]-1H-pyrazole-3-carboxamide
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C23H24BrClN6O2
 1
1
IC50 = 3.5 nM
   TI
   LI
   LO
   TS
CP0290513
[1-[4-(2,2-diphenylethylamino)-3-(morpholine-4-carbonyl)phenyl]sulfonylpiperidin-4-yl]-(4-methylpiperazin-1-yl)methanone
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C36H45N5O5S
 1
1
IC50 = 33 nM
   TI
   LI
   LO
   TS