| Compound ID |
Compound Name |
Compound Formula |
|
CP0431929
|
4-(5-cyano-2-(4-fluorophenyl)-6-methyl-1H-indol-3-yl)-N-(methylsulfonyl)butanamide
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|
C21H20FN3O3S
|
1
|
| 1 |
IC50 = 19 nM
|
|
|
|
CP0378378
|
4-[5-cyano-2-(4-fluorophenyl)-6-methyl-1H-indol-3-yl]-N-(dimethylsulfamoyl)butanamide
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|
C22H23FN4O3S
|
1
|
| 1 |
IC50 = 24 nM
|
|
|
|
CP0455698
|
3-[5-(4-Fluoro-phenylcarbamoyl)-1-oxy-pyridine-2-sulfonyl]-benzoic acid
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|
C19H13FN2O6S
|
1
|
| 1 |
IC50 = 32 nM
|
|
|
|
CP0034902
|
4-[5-cyano-2-(4-fluorophenyl)-1H-indol-3-yl]-N-(dimethylsulfamoyl)butanamide
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|
C21H21FN4O3S
|
1
|
| 1 |
IC50 = 50 nM
|
|
|
|
CP0511492
|
4-[5-cyano-2-(4-fluorophenyl)-6-methoxy-1H-indol-3-yl]-N-(dimethylsulfamoyl)butanamide
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|
C22H23FN4O4S
|
1
|
| 1 |
IC50 = 57 nM
|
|
|
|
CP0560217
|
4-(5-cyano-2-(4-fluorophenyl)-1H-indol-3-yl)-N-(ethylsulfonyl)butanamide
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|
C21H20FN3O3S
|
1
|
| 1 |
IC50 = 64 nM
|
|
|
|
CP0530800
|
4-[5-cyano-2-(4-fluorophenyl)-1H-indol-3-yl]-N-sulfamoylbutanamide
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|
C19H17FN4O3S
|
1
|
| 1 |
IC50 = 66 nM
|
|
|
|
CP0500719
|
4-(5-cyano-2-(4-fluorophenyl)-1H-indol-3-yl)-N-(methylsulfonyl)butanamide
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|
C20H18FN3O3S
|
1
|
| 1 |
IC50 = 72 nM
|
|
|
|
CP0497871
|
4-(5-cyano-2-(4-fluorophenyl)-1H-indol-3-yl)-N-(trifluoromethylsulfonyl)butanamide
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|
C20H15F4N3O3S
|
1
|
| 1 |
IC50 = 87 nM
|
|
|
|
CP0524612
|
6-Benzenesulfonyl-N-(4-fluoro-phenyl)-1-oxy-nicotinamide
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|
C18H13FN2O4S
|
1
|
| 1 |
IC50 = 90 nM
|
|
|
|
CP0467172
|
N-[6,7-dichloro-3-(5-thiophen-2-ylthiophen-2-yl)quinoxalin-2-yl]-N',N'-diethylbutane-1,4-diamine
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|
C24H26Cl2N4S2
|
1
|
| 1 |
IC50 = 110 nM
|
|
|
|
CP0530801
|
4-[5-cyano-2-(4-fluorophenyl)-1H-indol-3-yl]-N-[(methylamino)sulfonyl]butanamide
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|
C20H19FN4O3S
|
1
|
| 1 |
IC50 = 120 nM
|
|
|
|
CP0530803
|
1-(2-(5-bromo-2-(4-fluorophenyl)-1H-indol-3-yl)ethyl)-3-(phenylsulfonyl)urea
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|
C23H19BrFN3O3S
|
1
|
| 1 |
IC50 = 120 nM
|
|
|
|
CP0403851
|
N-(4-fluorophenyl)-6-methylsulfonyl-1-oxidopyridin-1-ium-3-carboxamide
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|
C13H11FN2O4S
|
1
|
| 1 |
IC50 = 130 nM
|
|
|
|
CP0428751
|
6-Ethanesulfonyl-N-(4-fluoro-phenyl)-1-oxy-nicotinamide
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|
C14H13FN2O4S
|
1
|
| 1 |
IC50 = 130 nM
|
|
|
|
CP0504980
|
1-(2-(5-cyano-2-(4-fluorophenyl)-1H-indol-3-yl)ethyl)-3-(phenylsulfonyl)urea
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|
C24H19FN4O3S
|
1
|
| 1 |
IC50 = 140 nM
|
|
|
|
CP0472005
|
4-(5-cyano-2-(4-fluorophenyl)-1H-indol-3-yl)-N-(morpholinosulfonyl)butanamide
Show/Hide
|
C23H23FN4O4S
|
1
|
| 1 |
IC50 = 150 nM
|
|
|
|
CP0378353
|
4-(5-cyano-2-(4-fluorophenyl)-6-methoxy-1H-indol-3-yl)-N-(methylsulfonyl)butanamide
Show/Hide
|
C21H20FN3O4S
|
1
|
| 1 |
IC50 = 160 nM
|
|
|
|
CP0431931
|
4-(5-bromo-2-(4-fluorophenyl)-1H-indol-3-yl)-N-(methylsulfonyl)butanamide
Show/Hide
|
C19H18BrFN2O3S
|
1
|
| 1 |
IC50 = 170 nM
|
|
|
|
CP0496565
|
4-(5-cyano-2-(4-fluorophenyl)-1H-indol-3-yl)-N-(isopropylsulfonyl)butanamide
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|
C22H22FN3O3S
|
1
|
| 1 |
IC50 = 220 nM
|
|
|
|
CP0431933
|
1-(2-(5-bromo-2-(4-fluorophenyl)-1H-indol-3-yl)ethyl)-3-(methylsulfonyl)urea
Show/Hide
|
C18H17BrFN3O3S
|
1
|
| 1 |
IC50 = 250 nM
|
|
|
|
CP0392907
|
4-[5-cyano-2-(4-fluorophenyl)-1H-indol-3-yl]-N-[(2-methoxyethyl)sulfamoyl]butanamide
Show/Hide
|
C22H23FN4O4S
|
1
|
| 1 |
IC50 = 260 nM
|
|
|
|
CP0457958
|
4-(5-cyano-2-(4-fluorophenyl)-1H-indol-3-yl)-N-(phenylsulfonyl)butanamide
Show/Hide
|
C25H20FN3O3S
|
1
|
| 1 |
IC50 = 260 nM
|
|
|
|
CP0448473
|
6-benzylsulfonyl-N-(4-fluorophenyl)-1-oxidopyridin-1-ium-3-carboxamide
Show/Hide
|
C19H15FN2O4S
|
1
|
| 1 |
IC50 = 280 nM
|
|
|
|
CP0391732
|
N-(4-fluorophenyl)-1-oxido-6-propan-2-ylsulfonylpyridin-1-ium-3-carboxamide
Show/Hide
|
C15H15FN2O4S
|
1
|
| 1 |
IC50 = 400 nM
|
|
|
|
CP0384031
|
1-(2-chlorophenylsulfonyl)-3-(2-(5-cyano-2-(4-fluorophenyl)-1H-indol-3-yl)ethyl)urea
Show/Hide
|
C24H18ClFN4O3S
|
1
|
| 1 |
IC50 = 400 nM
|
|
|
|
CP0410132
|
6-Cyclopentanesulfonyl-N-(4-fluoro-phenyl)-1-oxy-nicotinamide
Show/Hide
|
C17H17FN2O4S
|
1
|
| 1 |
IC50 = 460 nM
|
|
|
|
CP0530802
|
1-(2-(5-cyano-2-(4-fluorophenyl)-1H-indol-3-yl)ethyl)-3-(4-fluorophenylsulfonyl)urea
Show/Hide
|
C24H18F2N4O3S
|
1
|
| 1 |
IC50 = 520 nM
|
|
|
|
CP0560218
|
1-(2-(5-cyano-2-(4-fluorophenyl)-1H-indol-3-yl)ethyl)-3-(methylsulfonyl)urea
Show/Hide
|
C19H17FN4O3S
|
1
|
| 1 |
IC50 = 640 nM
|
|
|
|
CP0530799
|
4-[5-cyano-2-(4-fluorophenyl)-1H-indol-3-yl]-N-(phenylsulfamoyl)butanamide
Show/Hide
|
C25H21FN4O3S
|
1
|
| 1 |
IC50 = 880 nM
|
|
|
|
CP0403824
|
6-Chloro-N-(4-fluoro-phenyl)-1-oxy-nicotinamide
Show/Hide
|
C12H8ClFN2O2
|
1
|
| 1 |
IC50 = 1000 nM
|
|
|
|
CP0422339
|
N-(butylsulfamoyl)-4-[5-cyano-2-(4-fluorophenyl)-1H-indol-3-yl]butanamide
Show/Hide
|
C23H25FN4O3S
|
1
|
| 1 |
IC50 = 1100 nM
|
|
|
|
CP0511493
|
4-[5-cyano-2-(4-fluorophenyl)-1H-indol-3-yl]-N-(diethylsulfamoyl)butanamide
Show/Hide
|
C23H25FN4O3S
|
1
|
| 1 |
IC50 = 1100 nM
|
|
|
|
CP0497872
|
4-(5-cyano-2-(4-fluorophenyl)-1H-indol-3-yl)-N-(propylsulfonyl)butanamide
Show/Hide
|
C22H22FN3O3S
|
1
|
| 1 |
IC50 = 1300 nM
|
|
|
|
CP0496925
|
N-benzylsulfonyl-4-[5-cyano-2-(4-fluorophenyl)-1H-indol-3-yl]butanamide
Show/Hide
|
C26H22FN3O3S
|
1
|
| 1 |
IC50 = 1400 nM
|
|
|
|
CP0404136
|
N-(4-tert-butylphenyl)-6-chloro-1-oxidopyridin-1-ium-3-carboxamide
Show/Hide
|
C16H17ClN2O2
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0437756
|
6-Chloro-N-(4-methoxy-phenyl)-1-oxy-nicotinamide
Show/Hide
|
C13H11ClN2O3
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0458740
|
N-benzhydryl-6-chloro-1-oxidopyridin-1-ium-3-carboxamide
Show/Hide
|
C19H15ClN2O2
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0488101
|
6-Chloro-N-cyclohexyl-1-oxy-nicotinamide
Show/Hide
|
C12H15ClN2O2
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0496413
|
6-Chloro-N-(4-iodo-phenyl)-1-oxy-nicotinamide
Show/Hide
|
C12H8ClIN2O2
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0503474
|
6-Chloro-N-(4-fluoro-benzyl)-1-oxy-nicotinamide
Show/Hide
|
C13H10ClFN2O2
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0538247
|
6-Chloro-N-(2-hydroxy-phenyl)-1-oxy-nicotinamide
Show/Hide
|
C12H9ClN2O3
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0378354
|
4-(5-cyano-2-(4-fluorophenyl)-1H-indol-3-yl)-N-methyl-N-(methylsulfonyl)butanamide
Show/Hide
|
C21H20FN3O3S
|
1
|
| 1 |
IC50 > 2000 nM
|
|
|
