Brief Information of the Cell Line and Protein
Cell Line ID: CL000680 , HBL
Category Cancer cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_J075
Protein ID: PT00911 , Melanocyte-stimulating hormone receptor
Gene Name MC1R
Organism Homo sapiens, Human
Protein Classification Membrane receptor
Uniprot ID Q01726
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000680  Protein ID: PT00911
 
Compound ID Compound Name Compound Formula
CP0908213
US9447148, 9.13
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C52H65N15O9
 1
1
EC50 = 0.01 nM
   TI
   LI
   LO
   TS
CP0870725
US9447148, 9.15
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C45H60N14O8
 1
1
EC50 = 0.012 nM
   TI
   LI
   LO
   TS
CP0951277
US9447148, 9.6
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C50H69N15O9
 1
1
EC50 = 0.014 nM
   TI
   LI
   LO
   TS
CP0904782
US9447148, 9.12
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C52H65N15O9
 1
1
EC50 = 0.015 nM
   TI
   LI
   LO
   TS
CP0929640
US9447148, 9.43
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C51H70N16O10
 1
1
EC50 = 0.016 nM
   TI
   LI
   LO
   TS
CP0870723
US9447148, 9.5
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C46H62N14O8S2
 1
1
EC50 = 0.025 nM
   TI
   LI
   LO
   TS
CP0870724
US9447148, 9.7
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C49H67N15O9
 1
1
EC50 = 0.025 nM
   TI
   LI
   LO
   TS
CP0966841
US9447148, 9.19
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C45H58N14O8
 1
1
EC50 = 0.031 nM
   TI
   LI
   LO
   TS
CP0908211
US9447148, 9.8
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C49H67N15O9
 1
1
EC50 = 0.052 nM
   TI
   LI
   LO
   TS
CP0423973
US9447148, 9.63
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C38H62N12O8
 1
1
EC50 = 0.076 nM
   TI
   LI
   LO
   TS
CP0870717
US9447148, 9.25
   Show/Hide
C41H62N14O9
 1
1
EC50 = 0.08 nM
   TI
   LI
   LO
   TS
CP0474882
US9447148, 9.59
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C37H59ClN12O8
 1
1
EC50 = 0.1 nM
   TI
   LI
   LO
   TS
CP0904523
US9447148, 9.26
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C48H64N14O10
 1
1
EC50 = 0.107 nM
   TI
   LI
   LO
   TS
CP0423940
US9447148, 9.64
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C38H62N12O9
 1
1
EC50 = 0.12 nM
   TI
   LI
   LO
   TS
CP0870738
US9447148, 9.66
   Show/Hide
C48H67N13O9
 1
1
EC50 = 0.18 nM
   TI
   LI
   LO
   TS
CP0870722
US9447148, 9.4
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C47H63N15O9
 1
1
EC50 = 0.195 nM
   TI
   LI
   LO
   TS
CP0493416
US9447148, 9.56
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C37H60N12O8
 1
1
EC50 = 0.5 nM
   TI
   LI
   LO
   TS
CP0486280
US9447148, 9.60
   Show/Hide
C37H59FN12O8
 1
1
EC50 = 0.8 nM
   TI
   LI
   LO
   TS
CP0481221
US9447148, 9.57
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C37H59ClN12O8
 1
1
EC50 = 1 nM
   TI
   LI
   LO
   TS
CP0481223
US9447148, 9.62
   Show/Hide
C37H58F2N12O8
 1
1
EC50 = 1 nM
   TI
   LI
   LO
   TS
CP0548110
US9447148, 9.61
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C37H59FN12O8
 1
1
EC50 = 1 nM
   TI
   LI
   LO
   TS
CP0497596
US9447148, 9.58
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C37H59ClN12O8
 1
1
EC50 = 2 nM
   TI
   LI
   LO
   TS
CP0908214
US9447148, 9.14
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C40H51N13O7
 1
1
EC50 = 31 nM
   TI
   LI
   LO
   TS
CP0423941
US9447148, 9.65
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C37H57N11O8
 1
1
EC50 = 332 nM
   TI
   LI
   LO
   TS