General Information of the Compound
Compound ID
CP0679751
Compound Name
rac-2-{5-Chloro-2-[5,5-dimethyl-2-oxo-3-(2,2,2-trifluoroacetylamino)-2,3,4,5-tetrahydro-1H-1-benzazepin-8-ylamino]-pyrimidin-4-ylamino}-3-fluoro-N-methyl-benzamide 2,2,2-trifluoroacetic acid
    Show/Hide
Structure
Formula
C28H25ClF7N7O5
Molecular Weight
707.991
Canonical SMILES
CNC(=O)c1cccc(F)c1Nc1nc(Nc2ccc3c(c2)NC(=O)C(NC(=O)C(F)(F)F)CC3(C)C)ncc1Cl.O=C(O)C(F)(F)F
    Show/Hide
InChI
InChI=1S/C26H24ClF4N7O3.C2HF3O2/c1-25(2)10-18(36-23(41)26(29,30)31)22(40)35-17-9-12(7-8-14(17)25)34-24-33-11-15(27)20(38-24)37-19-13(21(39)32-3)5-4-6-16(19)28;3-2(4,5)1(6)7/h4-9,11,18H,10H2,1-3H3,(H,32,39)(H,35,40)(H,36,41)(H2,33,34,37,38);(H,6,7)
    Show/Hide
InChIKey
XFWJBSSSWQZGAD-UHFFFAOYSA-N
Physicochemical Property
logP
5.4161
Rotatable Bonds
6
Heavy Atom Count
48
Polar Areas
174.44
Hydrogen Bond Donor Count
6
Hydrogen Bond Acceptor Count
8
Complexity
48

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

    Show/Hide
Click to Show/Hide the External Link(s) of This Compound
PubChem ID
CID: 57390203
ChEMBL ID
CHEMBL1939320
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01201, Hepatocyte growth factor receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000282 GTL-16 Homo sapiens (Human)  1
1
IC50 = 16 nM
   TI
   LI
   LO
   TS