General Information of the Compound
Compound ID
CP0577419
Compound Name
N-(5-hydroxy-2-adamantyl)-2-[(2R)-2-methyl-4-(4-methylsulfonylphenyl)piperazin-1-yl]pyrimidine-4-carboxamide
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Structure
Formula
C27H35N5O4S
Molecular Weight
525.675
Canonical SMILES
C[C@@H]1CN(CCN1c1nccc(n1)C(=O)NC1C2CC3CC1CC(O)(C3)C2)c1ccc(cc1)S(C)(=O)=O
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InChI
InChI=1S/C27H35N5O4S/c1-17-16-31(21-3-5-22(6-4-21)37(2,35)36)9-10-32(17)26-28-8-7-23(29-26)25(33)30-24-19-11-18-12-20(24)15-27(34,13-18)14-19/h3-8,17-20,24,34H,9-16H2,1-2H3,(H,30,33)/t17-,18?,19?,20?,24?,27?/m1/s1
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InChIKey
FEGJQPCXQMHGGC-JPAYEOGSSA-N
Physicochemical Property
logP
2.2646
Rotatable Bonds
5
Heavy Atom Count
37
Polar Areas
115.73
Hydrogen Bond Donor Count
2
Hydrogen Bond Acceptor Count
8
Complexity
37

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 67464318
ChEMBL ID
CHEMBL4788862
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01107, 11-beta-hydroxysteroid dehydrogenase 1
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 8.5 nM
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